Herbicidal pyridinesulfonylureas

ABSTRACT

This invention relates to herbicidal pyridinesulfonylureas which are highly active as preemergence and postemergence herbicides.

CROSS-REFERENCE TO RELATED APPLICATION

This application is a division of prior Application Ser. No. 07/806,749,filed Dec. 13, 1991, now U.S. Pat. No. 5,209,770, granted May 11, 1993,which is a division of prior Application Ser. No. 07/507,926, filed Apr.12, 1990, now granted as U.S. Pat. No. 5,102,444, granted Apr. 7, 1992;which is in rum a continuation-in-part of Application Ser. No. 399,485,filed May 26, 1989, now abandoned; which in turn derives from PCTApplication Ser. No. US87/03111, filed Dec. 4, 1987; which in turn was acontinuation-in-part of U.S. application Ser. No. 07/039,491, filed Apr.16, 1987, now abandoned; which in turn was a continuation-in-part ofapplication Ser. No. 939,428, filed Dec. 8, 1986, now abandoned.

BACKGROUND OF THE INVENTION

Pyridinesulfonylureas of the instant application show high activity aspreemergence and postemergence herbicides. In particular, safety to cornis demonstrated by many of the herbicides.

EP-A-13,480 discloses herbicidal sulfonamides of the formula ##STR1##wherein R₁ is H, Cl, Br, F, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄alkylthio, NO₂ or CO₂ R₅.

U.S. Pat. No. 4,435,206, issued Mar. 6, 1984 and U.S. Pat. No.4,522,645, issued Jun. 11, 1983, disclose 2-pyridinesulfonylureassubstituted in the 3-position by R₁, wherein R₁ is H, Cl, Br, F, C₁ -C₄alkyl, C₁ -C₄ alkoxy, C₁ -C₄ alkylthio, NO₂, CF₃, CO₂ R₅ or SO₂ NR₆ R₇.

U.S. Pat. No. 4,339,267 discloses herbicidal sulfonamides of the formula##STR2## wherein R₄ is H, Cl, Br, F, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, NO₂,CO₂ R₆ or SR₁₃.

EP-A-30,433 discloses herbicidal sulfonamides of the formula ##STR3##wherein X is H;

R₁₄ is H or CH₃ ; and

R₃ is H, F, Cl, Br, CH₃, OCH₃, NO₂, CO₂ R₁₁ or S(O)_(n) R₁₂.

U.S. Pat. No. 4,456,469 discloses herbicidal sulfonamides of the formula##STR4## wherein R is C₁ -C₆ alkyl, C₃ -C₆ alkenyl, C₂ -C₄ alkoxyalkyl,C₅ -C₆ cycloalkyl, R'OCH₂ CH₂ OCH₂, R'OCH₂ CH₂ OCH₂ CH₂, ##STR5## CF₃,CF₃ CH₂, HGLCCF₂ or HCF₂ ; and Z is H, F, Cl, Br, CH₃, OCH₃ or SCH₃.

U.S. Pat. No. 4,487,626 discloses herbicidal sulfonamides of the formula##STR6## wherein A is ##STR7## and R₂ is H, F, Cl, Br, C₁ -C₄ alkyl, C₁-C₄ alkoxy, NO₂, CO₂ R₁₅, S(O)_(m) R₁₆, SO₂ NR₁₈ R₁₉ or SO₂ N(OCH₃)CH₃.

U.S. Pat. No. 4,421,550 discloses herbicidal sulfonamides of the formula##STR8## wherein Z is ##STR9## and R₁₆ is H, C₁ -C₄ alkyl, C₁ -C₄alkoxy, F, Cl, Br, CF₃, CO₂ R₂₀, SO₂ NR₁₀ R₁₁, SO₂ N(OCH₃)CH₃ orS(O)_(n) R₁₃.

U.S. Pat. No. 4,496,392 discloses herbicidal sulfonamides of the formula##STR10## wherein R₃ is Cl, SO₂ CH₃ or SO₂ N(CH₃)₂.

EP-A-84,224 discloses herbicidal sulfonamides of the formula ##STR11##wherein A is ##STR12## and R₁₆ is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, F, Cl,Br, CF₃, CO₂ R₉, SO₂ NR₁₀ R₁₁, SO₂ N(OCH₃)CH₃ or S(O)_(n) R₁₃.

EP-A-125,846 discloses herbicidal sulfonamides of the formula ##STR13##wherein J is ##STR14## and R₃ is Cl, SO₂ CH₃, SO₂ N(CH₃)₂, OCH₃, NO₂ orN(CH₃)₂.

EP-A-155,767 discloses herbicidal sulfonamides of the formula ##STR15##wherein J is ##STR16## and R₅ is H, CH₃, Cl, Br, CO₂ R₁₅, C(O)NR₁₆ R₁₇,SO₂ NR₁₆ R₁₇, SO₂ N(OCH₃)CH₃, SO₂ R₁₈ or NO₂.

EP-A-161,905 discloses herbicidal sulfonamides of the formula ##STR17##wherein R₄ is CH₃, CH₂ CH₃, OCH₃, OCH₂ CH₃, F, Cl, Br, SO₂ NR₁₆ R₁₇, SO₂N(OCH₃)CH₃, S(O)_(n) R₁₉, C₃ -C₄ alkenyloxy or C₃ -C₄ alkynyloxy.

EP-A-164 , 269 discloses herbicidal sulfonamides of the formula##STR18## wherein R₄ is CH₃, CH₂ CH₃, OCH₃, OCH₂ CH₃, F, Cl, Br, SO₂NR₁₁ R₁₂, SO₂ N(OCH₃)CH₃ or S(O)_(n) R₁₃.

EP-A-171,286 discloses herbicidal sulfonamides of the formula ##STR19##wherein R₄ is CH₃, CH₂ CH₃, OCH₃, OCH₂ CH₃, F, Cl, Br, SO₂ NR₁₈ R₁₉, SO₂N(OCH₃)CH₃, S(O)_(n) R₂₁, C₃ -C₄ alkenyloxy, CH₂ OCH₃ or CH₂ OCH₂ CH₃.

South African Patent Application 83/4305, published Dec. 14, 1983,discloses herbicidal sulfonamides of the formula ##STR20## wherein R₂ isH, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, NO₂, C₁ -C₃ alkoxy, C(W)R₈,SO₂ NR₆ R₇, S(O)_(n) -- C₁ -C₃ alkyl or C(O)R₉ ;

R₃ is H, halogen, C₁ -C₃ alkyl, OCH₃, NO₂ or CF₃ ;

R₅ is H, NO₂, F, Cl, Br, CH₃, CF₃, S(O)_(n) C₁ -C₃ alkyl, C(O)C₁ -C₄alkoxy or C₁ -C₃ alkoxy;

Y is O or S.

South African Patent Application 83/6639, published Mar. 8, 1984,discloses herbicidal sulfonamides of the formula ##STR21## wherein A isa C₃ -C₆ alkynyl radical, a C₁ -C₆ alkyl radical which is substituted byhalogen, C₁ -C₄ alkoxy, C₁ -C₄ alkylthio, C₁ -C₄ alkylsulfinyl, C₁ -C₄alkylsulfonyl, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkylthio, C₁ -C₄haloalkylsulfinyl or C₁ -C₄ haloalkylsulfonyl, or is a C₂ -C₄ alkenylradical which is unsubstituted or substituted as for C₁ -C₆ alkyl, or isa phenyl radical which is unsubstituted or substituted by halogen,cyano, nitro, C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, an --X--C₁ -C₄ alkyl, C₁-C₄ alkoxycarbonyl, amino, mono- or di(C₁ -C₄ alkyl)amino, carbamoyl,mono- or di-(C₁ -C₄ alkyl)carbamoyl, sulfamoyl, mono- or di-(C₁ -C₄alkyl)sulfamoyl radical;

R₁ is hydrogen, halogen, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkyl,C₁ -C₄ haloalkoxy, C₂ -C₅ alkoxyalkoxy, C₁ -C₅ alkylthio, C₁ -C₅alkylsulfinyl or C₁ -C₅ alkylsulfonyl; and

X is O, S, SO or SO₂.

U.S. Pat. No. 4,518,776 discloses a process for the preparation ofherbicidal sulfonamides of the formula ##STR22## wherein R₁, in part, isS(O)_(n) C₁ -C₄ alkyl, SO₂ di-C₁ -C₄ alkylamino or CO₂ -C₁ -C₂ alkyl;and

R₂ is H, halogen, CF₃, NO₂, C₁ -C₄ alkyl or C₁ -C₄ alkoxy.

This patent generically discloses some, but does not claim any,compounds of the instant invention.

EP-A-101,670, published Feb. 29, 1984, discloses a process for thepreparation of herbicidal sulfonamides of the formula ##STR23## whereinR₁ is Q-C₁ -C₄ alkyl, SO₂ -di-C₁ -C₄ alkylamino or CO₂ -C₁ -C₄ alkyl;

Q is S or S(O)_(n) ; and

R₂ is H, halogen, CF₃, NO₂, C₁ -C₄ alkyl or C₁ -C₄ alkoxy.

This application generically discloses some of the compounds of theinstant invention.

U.S. Pat. No. 4,521,597 discloses a process for the preparation ofherbicidal sulfonamides of the formula ##STR24## wherein R₃ is H, F, Cl,Br, NO₂, OCH₃ or CF₃ ;

R₅ is S(O)_(m) C₁ -C₅ alkyl, SO₂ NR₈ R₉ or COR₇ ; and

R₆ is H, F, CH₃ or OCH₃.

This patent generically discloses some, but does not claim any,compounds of the instant invention.

EP-A-184,385, published Jun. 11, 1986, discloses the following compoundfor selective weed control in tomatoes and turf. ##STR25##

U.S. Ser. No. 874,307 discloses herbicidalo-alkylcarbonyl-pyridinesulfonylureas.

U.S. Ser. No. 943,137 discloses herbicidalo-substituted-pyridinesulfonylureas.

SUMMARY OF THE INVENTION

This application pertains to novel compounds of Formula I,agriculturally suitable compositions containing them and theirmethod-of-use as preemergent and/or postemergent herbicides or plantgrowth regulants. ##STR26## wherein J is ##STR27## R is H or CH₃ ; W isO or S;

R₁ is R_(f) or R_(g) ;

R_(f) is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, NO₂, C₁ -C₃ alkoxy,C₁ -C₃ alkylthio or CN;

R_(g) is C₁ -C₃ haloalkyl, C₂ -C₃ alkyl, cyclopropyl, C₁ -C₃ alkylsubstituted by C₁ -C₃ alkoxy, OH, C₁ -C₂ alkylthio or CN, CN, W₂ R₁₁,amino, C₁ -C₃ alkylamino or C₁ -C₃ dialkylamino;

R₂ is C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl, C₃ -C₅ cycloalkylthio,C₃ -C₅ cycloalkylsulfinyl, C₃ -C₅ cycloalkylsulfonyl, SO₂ NH₂, SO₂NR_(d) R_(e), SO₂ NR'₇ R₈, SO₂ NR₇ R₈, OSO₂ R₈, SO₂ OR₈, N₃, P(W₁)(OC₁-C₂ alkyl)₂, CN, CO₂ R₉, CO₂ R'₉, CH₂ F, CF₂ H, CH₂ Cl, CCl₂ H or C₂ -C₄haloalkyl;

R₃ is C₁ -C₄ alkylsulfinyl, C₃ -C₅ cycloalkylthio, C₃ -C₅cycloalkylsulfinyl, C₃ -C₄ cycloalkylsulfonyl, SO₂ NH₂, SO₂ NR_(d)R_(e), SO₂ NR₇ R₈, SO₂ NR'₇ R₈, OSO₂ R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂alkyl)₂, CN, CO₂ R₉, CO₂ R'₉ or C₁ -C₄ haloalkyl;

R₄ is C₁ -C₄ alkylsulfinyl, C₃ -C₅ cycloalkylthio, C₃ -C₅cycloalkylsulfinyl, C₃ -C₄ cycloalkylsulfonyl, SO₂ NH₂, SO₂ NR_(d)R_(e), SO₂ NR₇ R₈, OSO₂ R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂ alkyl)₂, CN, CO₂R₉ or C₁ -C₄ haloalkyl;

R₅ is C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl, C₃ -C₅ cycloalkylthio,C₃ -C₅ cycloalkylsulfinyl, C₃ -C₅ cycloalkylsulfonyl, SO₂ NH₂, SO₂NR_(d) R_(e), SO₂ NR₇ R₈, OSO₂ R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂ alkyl)₂,CN, CO₂ R₉ or C₁ -C₄ haloalkyl;

R₆ is C₁ -C₄ alkylthio, C₁ -C₄ alkylsulfinyl, C₁ -C₄ haloalkylthio, C₁-C₄ haloalkylsulfinyl, C₁ -C₄ haloalkylsulfonyl, C₃ -C₄ alkenylthio, C₃-C₄ alkenylsulfinyl, C₃ -C₄ alkenylsulfonyl, C₃ -C₄ alkynylthio, C₃ -C₄alkynylsulfinyl, C₃ -C₄ alkynylsulfonyl, C₃ -C₅ cycloalkylthio, C₃ -C₅cycloalkylsulfinyl, C₃ -C₅ cycloalkylsulfonyl, SO₂ NR_(d) R_(e), SO₂ NR₇R₈, OSO₂ R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂ alkyl)₂, CN, CO₂ R₉ or C₁ -C₄haloalkyl;

R₇ is H, C₂ -C₃ cyanoalkyl, C₃ -C₄ alkenyl or C₃ -C₄ alkynyl;

R'₇ is C₁ -C₄ alkyl;

R₈ is C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂-C₄ alkoxyalkyl or cyclopropyl; or

R₇ and R₈ may be taken together as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ --or --CH₂ CH₂ OCH₂ CH₂ --;

R₉ is CH₂ CH₂ R₁₀, CH₂ CF₃, C₃ -C₄ haloalkyl, C₃ -C₄ alkynyl, C₂ -C₄alkylthioalkyl, C₃ -C₅ cycloalkyl or C₄ -C₇ cycloalkylalkyl;

R'₉ is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, CH₂ CH₂ Cl, CH₂ CH₂ Br, CH₂ CH₂OCH₃ or CH₂ CH₂ OC₂ H₅ ;

R₁₀ is OH, F, CN, OSO₂ (C₁ -C₃ alkyl) or OSO₂ (C₁ -C₃ haloalkyl);

R₁₁ is C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, C₃ -C₄ alkenyl or C₃ -C₄ alkynyl;

W₁ is O or S;

W₂ is O or S;

A is ##STR28## X is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₂ -C₄ haloalkoxy,C₁ -C₄ haloalkyl, C₂ -C₄ haloalkylthio, C₁ -C₄ alkylthio, halogen, C₂-C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino or di(C₁-C₃ alkyl)amino;

Y is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₂ -C₄ haloalkoxy, C₂ -C₄haloalkylthio, C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino, C₃ -C₄alkenyloxy, C₃ -C₄ alkynyloxy, C₂ -C₅ alkylthioalkyl, C₂ -C₅alkylsulfinylalkyl, C₂ -C₅ alkylsulfonylalkyl, C₁ -C₄ haloalkyl, C₂ -C₄alkynyl, C₃ -C₅ cycloalkyl, azido, ##STR29## N(OCH₃)CH₃ ; m is 2 or 3;

Q₁ and Q₂ are independently O or S;

R_(a) is H or C₁ -C₃ alkyl;

R_(b) and R_(c) are independently C₁ -C₃ alkyl;

R_(d) is H or C₁ -C₂ alkyl;

R_(e) is C₁ -C₂ alkoxy;

Z is CH, N, CCH₃, CC₂ H₅, CCl or CBr;

Y₁ is O or CH₂ ;

X₁ is CH₃, OCH₃, OC₂ H₅ or OCF₂ H;

X₂ is CH₃, C₂ H₅ or CH₂ CF₃ ;

Y₂ is OCH₃, OC₂ H₅, SCH₃, SC₂ H₅, CH₃ or CH₂ CH₃ ;

X₃ is CH₃ or OCH₃ ;

Y₃ is H or CH₃ ;

X₄ is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃ or Cl;

Y₄ is CH₃, OCH₃, OC₂ H₅ or Cl;

and their agriculturally suitable salts; provided that

1) when X is halogen, then Z is CH and Y is OCH₃, OC₂ H₅, NH₂, NHCH₃,N(CH₃)₂ or N(OCH₃)CH₃ ;

2) when W is S, then R is H, A is A-1, Z is CH or N, and Y is CH₃, OCH₃,OC₂ H₅, CH₂ OCH₃, C₂ H₅, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂OCH₃, CH(OCH₃)₂ or ##STR30## 3) when the total number of carbon atoms ofX and Y is greater than four, then the combined number of carbons of R₁,R₂, R₃, R₄, R₅ or R₆ is less than or equal to six;

4) when J is J-1 and R₂ is C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl,SO₂ NR_(d) R_(e), SO₂ NR'₇ R₈ or CO₂ R'₉, or when J is J-2 and R₃ is C₁-C₄ alkylsulfinyl, CF₃, SO₂ NR_(d) R_(e), SO₂ NR'₇ R₈ or CO₂ R'₉, then Yis other than C₂ -C₅ alkylthioalkyl, C₂ -C₅ alkylsulfinylalkyl, C₂ -C₅alkylsulfonylalkyl, ##STR31## 5) when J is J-2 or J-3 and R₃ or R₄ is C₁-C₄ alkylsulfinyl, then X and Y are other than NH₂ or NHCH₃ ;

6) when J is J-2 and R₃ is C₁ -C₄ alkylsulfinyl or SO₂ NR_(d) R_(e), orR₇ is H, then X and Y are other than C₂ -C₄ haloalkoxy;

7) when J is J-5, then R₇ is other than H and R₆ is other than SO₂NR_(d) R_(e) ;

8) when J is J-2 and R₃ is SO₂ NH₂ or SO₂ NR_(d) R_(e), or R₇ is H, thenX is other than iodine;

9) when J is J-2 and R₇ is H or R₃ is SO₂ NR_(d) R_(e), then Y is otherthan C₂ -C₄ alkynyl;

10) X₄ and Y₄ are not simultaneously Cl;

11) when J is J-1, J-2, J-3, J-4 and A is A-5, then R_(f) is other thanH;

12) when J is J-1 or J-2, then A is other than A-6;

13) when J is J-1 and A is A-7, then R₂ is other than C₁ -C₄alkylsulfonyl;

14) when R₂ or R₃ is CO₂ R'₉ or SO₂ NR'₇ R₈, then R₁ is R_(g) and whenR₂ or R₃ is other than CO₂ R'₉ or SO₂ NR'₇ R₈, then R₁ is R_(f) ; and

15) when J is J-2 and R₁ is adjacent to the sulfonylurea bridge, thenR_(g) is C₁ -C₃ haloalkyl, C₂ -C₃ alkyl, cyclopropyl, CN, W₂ R₁₁, amino,C₁ -C₃ alkylamino or C₁ -C₃ dialkylamino.

In the above definitions, the term "alkyl", used either alone or incompound words such as "alkylthio" or "haloalkyl", denotes straightchain or branched alkyl, e.g. methyl, ethyl, n-propyl, isopropyl or thedifferent butyl isomers.

Alkoxy denotes methoxy, ethoxy, n-propyloxy or isopropyloxy.

Alkenyl denotes straight chain or branched alkenes, e.g. 1-propenyl,2-propenyl, 3-propenyl and the different butenyl isomers.

Alkynyl denotes straight chain or branched alkynes, e.g. ethynyl,1-propynyl, 2-propynyl and the different butynyl isomers.

Alkylsulfonyl denotes methylsulfonyl, ethylsulfonyl and the differentpropylsulfonyl and butylsulfonyl isomers.

Cycloalkyl denotes cyclopropyl, cyclobutyl and cyclopentyl.

The term "halogen", either alone or in compound words such as"haloalkyl", denotes fluorine, chlorine, bromine or iodine. Further,when used in compound words such as "haloalkyl" said alkyl may bepartially halogenated or fully substituted with halogen atoms which maybe the same or different. Examples of haloalkyl include CH₂ CH₂ F, CF₂CF₃ and CH₂ CHFCl. Similarly, this definition applies to haloalkoxy andhaloalkylthio.

The total number of carbon atoms in a substituent group is indicated bythe C_(i) -C_(j) prefix where i and j are numbers from 1 to 5. Forexample, C₁ -C₃ alkylsulfonyl would designate methylsulfonyl throughpropylsulfonyl, C₂ alkoxyalkoxy would designate OCH₂ OCH₃, C₂ cyanoalkylwould designate CH₂ CN and C₃ cyanoalkyl would designate CH₂ CH₂ CN andCH(CN)CH₃.

PREFERRED COMPOUNDS

Preferred for reasons of increased ease of synthesis and/or greaterherbicidal efficacy are:

1. Compounds of Formula I where

X is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, Cl, F, Br, I, CH₂ F, CF₃, OCH₂ CH₂ F,OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; and

Y is H, C₁ -C₂ alkyl, C₁ -C₂ alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃,N(OCH₃)CH₃, N(CH₃)₂, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂OCH₃, ##STR32## CH₂ SCH₃, cyclopropyl, C.tbd.CH or C.tbd.CCH₃ ; R_(a) isH or CH₃ ; and

Z is CH or N.

2. Compounds of Preferred 1 where

W is O;

R_(f) is H, CH₃, C₁ haloalkyl, halogen or OCH₃ ;

R_(g) is C₁ -C₂ haloalkyl, ethyl, W₂ R₁₁, CH₂ OCH₃, CH₂ SCH₃, CH₂ CN, C₁-C₂ alkylamino or N(CH₃)₂ ;

R₂ is C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl, SO₂ NH₂, SO₂ NR_(d)R_(e), SO₂ NR₇ R₈, SO₂ NR'₇ R₈, OSO₂ R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂alkyl)₂, CN, CO₂ R₉, CO₂ R'₉, CHF₂, CF₂ H, CH₂ Cl, CCl₂ H or C₂ -C₄haloalkyl;

R₃ is C₁ -C₄ alkylsulfinyl, SO₂ NH₂, SO₂ NR_(d) R_(e), SO₂ R₇ R₈, SO₂NR'₇ R₈, OSO₂ R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂ alkyl)₂, CN, CO₂ R₉, CO₂R'₉ or C₁ -C₄ haloalkyl;

R₄ is C₁ -C₄ alkylsulfinyl, SO₂ NH₂, SO₂ N(OCH₃)CH₃, SO₂ NR₇ R₈, OSO₂R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂ alkyl)₂, CN, CO₂ R₉ or C₁ -C₄ haloalkyl;

R₅ is C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl, SO₂ NH₂, SO₂N(OCH₃)CH₃, SO₂ NR₇ R₈, OSO₂ R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂ alkyl)₂, CN,CO₂ R₉ or C₁ -C₄ haloalkyl;

R₆ is C₁ -C₄ alkylthio, C₁ -C₄ alkylsulfinyl, C₁ -C₄ haloalkylthio, C₁-C₄ haloalkylsulfinyl, C₁ -C₄ haloalkylsulfonyl, C₃ -C₄ alkenylthio, C₃-C₄ alkenylsulfinyl, C₃ -C₄ alkenylsulfonyl, C₃ -C₄ alkynylthio, C₃ -C₄alkynylsulfinyl, C₃ -C₄ alkynylsulfonyl, SO₂ N (OCH₃)CH₃, SO₂ NR₇ R₈,OSO₂ R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂ alkyl)₂, CN, CO₂ R₉ or C₁ -C₄haloalkyl;

R₇ is H, C₂ -C₃ cyanoalkyl, C₃ -C₄ alkenyl or C₃ -C₄ alkynyl;

R₈ is C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂-C₄ alkoxyalkyl or cyclopropyl; and

R₁₁ is C₁ -C₃ alkyl, C₁ -C₂ haloalkyl, allyl or propargyl.

3. Compounds of Preferred 2 where J is J-1.

4. Compounds of Preferred 2 where J is J-2.

5. Compounds of Preferred 2 where J is J-3.

6. Compounds of Preferred 2 where J is J-4.

7. Compounds of Preferred 2 where J is J-5.

8. Compounds of Preferred 3 where

R₇ is H, C₂ -C₃ cyanoalkyl, allyl or propargyl;

R'₇ is C₁ -C₃ alkyl;

R₈ is C₁ -C₃ alkyl, allyl, propargyl or cyclopropyl;

R₉ is CH₂ CH₂ R₁₀, CH₂ CH₂ SCH₃, propargyl or cyclopropylmethyl;

R'₉ is C₁ -C₃ alkyl, allyl, CH₂ CH₂ OCH₃ or CH₂ CH₂ Cl; and

R₁₀ is OH, CN or OSO₂ CH₃.

9. Compounds of Preferred 8 where

A is A-1;

X is CH₃, OCH₃, OCH₂ CH₃, Cl or OCH₂ CF₃ ; and

Y is CH₃, OCH₃, CH₂ CH₃, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

10. Compounds of Preferred 9 where Z is CH.

11. Compounds of Preferred 9 where Z is N.

12. Compounds of Preferred 4 where

R₇ is H, C₂ -C₃ cyanoalkyl, allyl or propargyl; and

R₈ is C₁ -C₃ alkyl, allyl, propargyl or cyclopropyl.

13. Compounds of Preferred 12 where

A is A-1;

X is CH₃, OCH₃, OCH₂ CH₃, Cl or OCH₂ CF₃ ; and

Y is CH₃, OCH₃, CH₂ CH₃, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

14. Compounds of Preferred 13 where Z is CH.

15. Compounds of Preferred 13 where Z is N.

16. Compounds of Preferred 5 where

R₇ is H, C₂ -C₃ cyanoalkyl, allyl or propargyl; and

R₈ is C₁ -C₃ alkyl, allyl, propargyl or cyclopropyl.

17. Compounds of Preferred 16 where

A is A-1;

X is CH₃, OCH₃, OCH₂ CH₃, Cl or OCH₂ CF₃ ; and

Y is CH₃, OCH₃, CH₂ CH₃, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

18. Compounds of Preferred 17 where Z is CH.

19. Compounds of Preferred 17 where Z is N.

20. Compounds of Preferred 6 where

R₇ is H, C₂ -C₃ cyanoalkyl, allyl or propargyl; and

R₈ is C₁ -C₃ alkyl, allyl, propargyl or cyclopropyl.

21. Compounds of preferred 20 where

A is A-1;

X is CH₃, OCH₃, OCH₂ CH₃, Cl or OCH₂ CF₃ ; and

Y is CH₃, OCH₃, CH₂ CH₃, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

22. Compounds of Preferred 21 where Z is CH.

23. Compounds of Preferred 21 where Z is N.

24. Compounds of Preferred 7 where

R₆ is C₁ -C₂ alkylthio, C₁ -C₂ alkylsulfinyl, C₁ -C₂ haloalkylthio, C₁-C₂ haloalkylsulfinyl, C₁ -C₂ haloalkylsulfonyl, SO₂ N(OCH₃)CH₃ or SO₂NR₇ R₈ ;

R₇ is H, C₂ -C₃ cyanoalkyl, allyl or propargyl;

R₈ is C₁ -C₃ alkyl, allyl, propargyl or cyclopropyl.

25. Compounds of Preferred 24 where

A is A-1;

X is CH₃, OCH₃, OCH₂ CH₃, Cl or OCH₂ CF₃ ; and

Y is CH₃, OCH₃, CH₂ CH₃, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

26. Compounds of Preferred 25 where Z is CH.

27. Compounds of Preferred 25 where Z is N.

28. Compounds of Preferred 1 where

J is J-1;

A is A-1;

Z is CH;

W is O;

R₂ is C₁ -C₄ alkylsulfinyl or C₁ -C₄ alkylsulfonyl; and

R_(f) is H, C₁ -C₂ alkyl, C₁ haloalkyl, C₁ -C₂ alkoxy or C₁ -C₂thioalkyl.

29. Compounds of Preferred 28 where

R_(f) is H;

R₂ is C₁ -C₄ alkylsulfonyl;

X is OCH₃ ; and

Y is OCH₃.

Specifically Preferred for reasons of greatest ease of synthesis and/orgreatest herbicidal efficacy are:

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-3-(1-propylsulfonyl)-2-pyridinesulfonamide;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-3-(1-propylsulfinyl)-2-pyridinesulfonamide;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-3-(ethylsulfonyl)-2-pyridinesulfonamide;

N2-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-N3-ethyl-2,3-pyridinedisulfonamide;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-3-(methylsulfonyloxy)-2-pyridinesulfonamide;and

N2-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-N3-methyl-2,3-pyridinedisulfonamide.

This invention also pertains to novel compounds of the followingformulas ##STR33## wherein X_(a) is Cl, NH₂, HNC(CH₃)₃ and ##STR34##which are useful as intermediates to herbicidal sulfonylureas.Specifically preferred are:

3-ethylsulfonyl-2-pyridinesulfonamide andN3-methyl-2,3-pyridinedisulfonamide.

DETAILED DESCRIPTION OF THE INVENTION Synthesis

Compounds of Formula I can be synthesized either by one or more of themethods described in U.S. Pat. No. 4,456,469, or by the reaction ofsulfonamides II with the phenyl ester of the appropriate carbamic acidIII in the presence of an equimolar quantity of a tertiary amine basesuch as 1,8-diazabicyclo[5.4.0]undec-7-ene (DBU) as shown in Equation 1.##STR35## wherein J, R, and A are as previously defined.

The reaction shown in Equation 1 is best carried out at 25° C. in asolvent such as dioxane or acetonitrile for 1-2 hours under an inertatmosphere as described in European Patent Application No. 70,804(published Jan. 26, 1983). The desired products of Formula I can beconveniently isolated by acidifying the reaction solution with aqueoushydrochloric acid. Alternatively, the aqueous layer can be extractedwith a solvent such as methylene chloride or ethyl acetate. Drying andevaporation of the solvent affords the desired products. The phenylcarbamates can be synthesized by treatment of the correspondingheterocyclic amines of Formula A-NHR with diphenyl carbonate or phenylchloroformate in the presence of a base such as sodium hydride,pyridine, or potassium carbonate with a catalytic amount of4-dimethylaminopyridine. The mixture is stirred at temperatures between25° and 65° C. in a suitable solvent such as tetrahydrofuran for 12-36hours.

The required sulfonamides of Formula II can be synthesized by either oneof the methods shown below in Equations 2 and 3.

Equation 2 depicts the reaction of sulfonyl chlorides of Formula IV withammonia to give sulfonamides of Formula II. ##STR36## wherein J is aspreviously defined.

The amination of Equation 2 is conveniently effected by adding at leasttwo molar equivalents of either anhydrous ammonia or concentratedammonium hydroxide to a solution of the sulfonyl chloride IV in asuitable solvent such as diethyl ether, tetrahydrofuran or methylenechloride at temperatures between -30° and 25° C. The desiredsulfonamides of Formula II are isolated either by filtration, in whichcase the by-product ammonium chloride is removed by washing with water,or extraction into a suitable organic solvent such as methylene chlorideor ethyl acetate. Drying and evaporation of the solvent then affords theproducts II which are usually sufficiently pure to be carried directlyon to the next step.

Sulfonamides of Formula II can also be prepared as shown in Equation 3by treatment of the corresponding N-t-butylsulfonamides VI with anappropriate acid such as trifluoroacetic (TFA), polyphosphoric (PPA), orp-toluenesulfonic acid (p-TSA). ##STR37## wherein J is as previouslydefined.

The reaction of Equation 3 is conveniently carried out by stirring asolution of the compound of Formula VI in excess trifluoroacetic acid(approximately 0.3M) at about 25° C. for 1-72 hours. The desiredsulfonamides of Formula II are then isolated by removal of the volatilesin vacuo and crystallization from a suitable solvent such as diethylether, 1-chlorobutane, or ethyl acetate. Alternatively, theN-t-butylsulfonamides of Formula VI can be treated with a catalyticamount of p-toluenesulfonic acid monohydrate in a solvent such astoluene or xylenes at reflux temperature for 1-6 hours. The desiredproducts are then isolated in a manner analogous to the one describedabove. For use of polyphosphoric acid in the deprotection ofN-t-butylsulfonamides, see J. G. Lombardino, J. Org. Chem., 36, 1843(1971); for use of trifluoroacetic acid, see J. D. Catt and W. L.Matier, J. Org. Chem., 38, 1974 (1973).

Sulfonamides of Formula VI can be prepared by the reaction of sulfonylchlorides of Formula IV with excess t-butyl amine as shown in Equation4. ##STR38## wherein J is as previously defined.

Sulfonyl chlorides of Formula IV can be prepared according to theprocedures described in U.S. Pat. No. 4,456,469. Alternatively, theprocedures of South African Patent Application 84/8844 may be utilizedwhich describe the conversion of mercapto or arylmethylthio compounds tosulfonyl chlorides via treatment with hypochlorite solution.

Sulfonyl chlorides of Formula IVa may also be prepared via metallationof 2-fluoropyridine derivatives with lithium diisopropyl amide (LDA)according to the procedure of T. Gungot, F. Marsais and G. Queguiner, J.Organomet. Chem., 1981, 215, 139-150, followed by treatment with sulfurdioxide and N-chlorosuccinimide (NCS) as shown in Equation 5. ##STR39##wherein R₁ is as previously defined.

Sulfonyl chlorides of Formula IVb can be prepared from compounds ofFormula VII as shown in Equation 6 and described in U.S. Pat. No.4,420,325. ##STR40## wherein J is as previously defined; and

[X] is a suitable halogenating reagent which would be obvious to oneskilled in the art.

The sulfides of Formula VIII can be prepared by the reaction of a halopyridine compound of Formula IX with an appropriate mercaptan in thepresence of a base as described in U.S. Pat. No. 4,456,469 and shown inEquation 7. ##STR41## wherein X' is F, Cl, or Br; and

R' is C₁ -C₄ alkyl or benzyl.

The sulfides of Formula VIIIa can be prepared by metallation of thepyridine compound of Formula X with two equivalents of a strong basesuch as n-butyllithium or lithium diisopropylamide (LDA) as described byP. Breant, F. Marsais, and G. Queguiner, Synthesis, 1983, 822-824,followed by treatment with the appropriate disulfide as shown inEquation 8. ##STR42## wherein R' is C₁ -C₄ alkyl, C₃ -C₅ cycloalkyl orbenzyl; and

R₁ is as previously defined.

In an analogous manner, sulfides of Formula VIIIb can be prepared asshown in Equation 9. ##STR43## wherein R' is C₁ -C₄ alkyl, C₃ -C₅cycloalkyl, or benzyl; and

R₁ is as previously defined.

Sulfides of Formula VIIIc can be prepared by the metallation of a2-fluoropyridine derivative as described previously and again followedby treatment with an appropriate disulfide as shown in Equation 10.##STR44## wherein R' is C₁ -C₄ alkyl, C₃ -C₅ cycloalkyl, or benzyl; and

R₁ is as previously defined.

The sulfones and Sulfoxides of General Formula XI can be prepared fromthe corresponding sulfides of Formula VIIId by any one of the numerousoxidation reagents [O] known in the art such as hydrogen peroxide orperacids, as shown in Equation 11. ##STR45## wherein R₁ is as previouslydefined;

R' is C₁ -C₄ alkyl or C₃ -C₅ cycloalkyl; and

n is 1 or 2.

The chloropyridine of Formula IXa can be prepared by diazotization of3-amino-2-chloropyridine followed by displacement with cuprous cyanideas shown in Equation 12. The diazonium group can also be replaced byother groups such as SO₂ Cl and N₃ by those skilled in the art viamethods known in the literature. ##STR46## wherein R₁ is as previouslydefined.

The sulfides of General Formula VIIIf can be prepared as shown inEquation 13. Alkylation of a 3-hydroxy-2-mercaptopyridine derivativewith alkyl halides utilizing a variety of bases such as potassiumcarbonate or potassium t-butoxide afforded the sulfides of Formula VIIIewhich were then treated with the appropriate sulfonyl chlorides in thepresence of an acid acceptor such as triethylamine to afford sulfides ofFormula VIIIf. ##STR47## wherein R' is C₁ -C₄ alkyl or benzyl;

X' is Cl, Br, or I; and

R₁ and R₈ are as previously defined.

The esters of Formula VIIIg, VIIIh, and VIIIj can be prepared by eitherof the two methods shown in Equation 14. The first method involvesmetallation of a 2-fluoropyridine derivative as previously described inEquation 5, followed by treatment with ethyl or methyl chloroformatewhich afforded esters of Formula XIII. Mercaptide displacement asdescribed in Equation 7 resulted in esters of Formula VIIIg. Acidcatalyzed transesterification using the appropriate alcohol as thesolvent afforded esters of Formula VIIIh.

The second method involves the alkylation of a 2-mercaptonicotinic acidderivative VIIIi with alkyl halides utilizing a variety of bases such aspotassium carbonate or potassium t-butoxide, followed by conversion tothe acid halides by any number of standard reagents such as thionylchloride, phosphorous trichloride or pentachloride, or oxalyl chloride.The acid chlorides were then treated with the appropriate alcohols inthe presence of an acid acceptor such as triethylamine, to afford estersof Formula VIIIh. Conversion of the sulfides VIIIh to the sulfonamidesVIIIj was carried out as previously described. ##STR48## wherein R₉ canalso be R'₉ ; and

X', R', R₁, R₉ and R'₉ are as previously defined.

The sulfonamides of General Formula XIIa can be prepared as shown inEquation 15. However, for the preparation of primary or unhinderedsecondary sulfonamides, a protective group is needed for a later stagein the synthetic sequence. A representative example is shown in Equation16 where a t-butyl protective group is utilized for the synthesis ofsulfonamide IIa. ##STR49## wherein [D] is R_(d) R_(e), R₇ R₈, R'₇ R₈, orH₂ ; and R₁, R_(d), R_(e), R₇, R₈ and R'₇ are as previously defined.##STR50## wherein R₁ is as previously defined.

The difluoro compounds of Formula XIVa in Equation 17 can be preparedusing the reactions previously described. Treatment with one equivalentof various R₁ nucleophiles (those that are available in the art) resultsin a mixture of products which can be separated. An example of the useof sodium methoxide as the reactive nucleophile is shown. IntermediatesXIVb and XIVc can be separated and further derivatized as previouslydescribed. ##STR51## wherein R₂ is as previously defined.

An alternative method to prepare esters of Formula XVd is shown inEquation 18. Mercaptide displacement of a 2,6-dihalopyridine can beachieved followed by conversion to the sulfonamide XVa as previouslydescribed. Treatment with two equivalents of a strong base such asn-butyllithium in a similar manner to that described by P. Breant, F.Marsails, and G. Queguiner, Synthesis, 1983, 822-824, followed bytreatment with carbon dioxide affords the acids of Formula XVb. Theacids can then be treated with various R₁ nucleophiles such asalkoxides, mercaptides or amines to afford the acids of Formula XVc(using sodium methoxide as an example) which can then be esterified withthe appropriate alcohols utilizing standard 1,3-dicyclohexylcarbodiimide(DCC) coupling conditions to afford esters of Formula XVd. ##STR52##wherein R₉ can also be R'₉ ;

X' is F or Cl; and

R', R₉ and R'₉ are as previously defined.

In an analogous manner, sulfonamides of General Formula XVIb can beprepared as shown in Equation 19. Treatment of XVa with strong basefollowed by an appropriate disulfide affords sulfides of Formula XVIa.Further elaboration utilizing chemistry previously described affordssulfonamides of Formula XVIb. ##STR53## wherein X' is F or Cl; and

R' and [D] are as previously defined.

A choice by one skilled in the art of the appropriate methods forpreparing compounds of Formula I must take into account the nature ofthe substituents R₁ through R₁₁, and R_(d) through R_(g), and theirchemical compatibility with the reaction conditions of Equations 1through 19.

The heterocyclic amines of Formula A-NHR in Equation 1 above can beprepared by methods known in the literature, or simple modificationsthereof, by those skilled in the art. For instance, EP-A No. 84,224(published Jul. 27, 1983) and W. Braker et al., J. Chem. Soc., 69, 3072(1947) describes methods for preparing aminopyridines and triazinessubstituted by acetal groups such as dialkoxymethyl or1,3-dioxolan-2-yl, among other groups. Also, for example, South Africanpatent application Nos. 82/5045 and 82/5671 describe methods forpreparing aminopyrimidines and triazines substituted by haloalkyl orhaloalkylthio groups such as OCH₂ CH₂ F, OCH₂ CF₃, SCF₂ H, or OCF₂ H,among other groups. South African patent application No. 83/7434(published Oct. 5, 1983) describes methods for the synthesis ofcyclopropylpyrimidines and triazines substituted by such groups asalkyl, haloalkyl, alkoxy, haloalkoxy, alkylamino, dialkylamino oralkoxyalkyl.

The 5,6-dihydrofuro[2.3-d]pyrimidine-2-amines, thecyclopenta[d]pyrimidine-2-amines (A is A-2) and the6,7-dihydro-5H-pyrano[2.3-d]pyrimidin-2-amines (A is A-3) can beprepared as described in EP-A No. 15,683. Thefuro[2.3-d]pyrimidin-2-amines (A is A-4) are described in EP-A No.46,677.

Compounds of Formula A-NHR where A is A-5 are described in EP-A-73,562.Compounds where A is A-6 are described in EP-A-94,260.

In addition, general methods for preparing aminopyrimidines andtriazines have been reviewed in the following publications:

The Chemistry of Heterocyclic Compounds", a series published byInterscience Publishers, Inc., New York and London;

"Pyrimidines", Vol. 16 of the same series by D. J. Brown;

"s-Triazines and Derivatives", Vol. 13 of the same series by E. M.Smolin and L. Rappoport; and

F. C. Schaefer, U.S. Pat. No. 3,154,547 and K. R. Huffman and F. C.Schaefer, J. Org. Chem., 28, 1812 (1963), which describes the synthesisof triazines.

Preparation in view of the above would be obvious to one skilled in theart. Agriculturally suitable salts of compounds of Formula I are alsouseful herbicides and can be prepared in a number of ways known to theart. For example, metal salts can be made by contacting compounds ofFormula I with a solution of an alkali or alkaline earth metal salthaving a sufficiently basic anion (e.g., hydroxide, alkoxide, carbonateor hydroxide). Quaternary amine salts can be made by similar techniques.

Salts of compounds of Formula I can also be prepared by exchange of onecation for another. Cationic exchange can be effected by direct contactof an aqueous solution of a salt of a compound of Formula I (e.g.,alkali or quaternary amine salt) with a solution containing the cationto be exchanged. This method is most effective when the desired saltcontaining the exchanged cation is insoluble in water and can beseparated by filtration.

Exchange may also be effected by passing an aqueous solution of a saltof a compound of Formula I (e.g., an alkali metal or quaternary aminesalt) through a column packed with a cation exchange resin containingthe cation to be exchanged for that of the original salt and the desiredproduct is eluted from the column. This method is particularly usefulwhen the desired salt is water-soluble, e.g., a potassium, sodium orcalcium salt.

Acid addition salts, useful in this invention, can be obtained byreacting a compound of Formula I with a suitable acid, e.g.,p-toluenesulfonic acid, trichloroacetic acid or the like.

The preparation of the compounds of this invention is furtherillustrated by the following specific examples. Temperatures arereported in degrees Celsius; abbreviations for nuclear magneticresonance (NMR) are: s=singlet, d=doublet, t=triplet, m=multiplat, andpeak positions are reported as parts per million downfield from internaltetramethylsilane. Infrared (IR) peak positions are given in reciprocalcentimeters (cm⁻¹).

EXAMPLE 1 Preparation of 2-Fluoro-3-(propylthio)pyridine

To a stirred solution of 59 ml (0.113 mol) of 1.9 molar lithiumdiisopropyl amide (in hexanes) in 150 mls dry tetrahydrofuran cooled to-70° under nitrogen was added dropwise a solution of 10.0 g of2-fluoropyridine (0.103 mol) in 30 mls dry tetrahydrofuran such that thetemperature was maintained below -65°. The solution was stirred at -70°for 4 hours and a solution 17 g of n-propyldisulfide (0.113 mol) in 45mls dry tetrahydrofuran was added dropwise while maintaining thetemperature below -65°. After stirring another hour at -70° the solutionwas poured into water and extracted with ether. The combined organicphases were washed with brine, dried over magnesium sulfate, andevaporated to afford 14.5 g (82%) of a red oil: NMR (CDCl₃, 200 MHz),1.0 (3H, m), 1.7 (2H, m), 2.9 (2H, m), 7.1 (1H, m), 7.7 (1H, m), 8.0(1H, m); IR (neat) 1585, 1560, 1410, 1245 cm⁻¹.

EXAMPLE 2 Preparation of 2-(Phenylmethylthio)-3-(propylthio)pyridine

To a stirred suspension of 0.62 g (0.013 mol) of 50% sodium hydride (inmineral oil), which had been washed with hexanes, in 20 mls drydimethylformamide cooled to -5° under nitrogen was added dropwise 1.6 g(0.013 mol) benzyl mercaptan such that the temperature was maintainedbelow 5°. The suspension was stirred at room temperature for 1 hour,cooled to 0°, and a solution of 2.0 g (0.012 mol) of the product fromExample 1 was added dropwise while maintaining the temperature between0° and 5°. After warming to room temperature, the solution was pouredinto water and extracted with ether. The combined organic layers werewashed with water and with brine, dried over magnesium sulfate, andevaporated to an oil which was purified by flash chromatography toafford 0.9 g (27%) oil: NMR (CDCl₃, 200 MHz), 1.02 (3H, t, J=7 Hz), 1.6(2H, m), 2.9 (2H, t, J=7 Hz), 4.45 (2H, s), 6.9-7.6 (7H, m), 8.3 (1H,m); IR (neat) 1560, 1370 cm⁻¹.

EXAMPLE 3 Preparation ofN-(1,1-Dimethylethyl)-3-(propylsulfinyl)-2-pyridinesulfonamide

To a vigorously stirred mixture of 0.5 g (0.0018 mol) of the productfrom Example 2 in 9 mls methylene chloride and 4 mls water cooled to 0°was added 0.7 mls (0.008 mol) concentrated hydrochloric acid followed bythe dropwise addition of 8.9 mls (0.006 mol) of a 5% sodium hypochloritesolution such that the temperature was maintained between 0° and 5°.After the mixture was stirred for an additional 30 minutes at 0° thereaction was poured into water and extracted with methylene chloride.The combined organic layers were washed with brine, dried over magnesiumsulfate, and filtered. The filtrate was stirred and cooled to -70° undernitrogen and 0.53 g (0.0072 mol) of t-butyl amine was added dropwise andthe mixture was allowed to warm to room temperature. The reaction waspoured into water and extracted with methylene chloride. The organiclayers were combined and washed with brine, dried over magnesiumsulfate, and evaporated to a mixture which was purified by flashchromatography to afford 0.4 g (69%) white solid: m.p. 138°-140°; NMR(CDCl₃, 200 MHz) 1.09 (3H, m), 1.7 (1H, m), 2.0 (1H, m), 2.8 (1H, m),3.3 (1 H, m), 5.2 (NH), 7.7 (1H, m), 8.6 (1H, m), 8.8 (1H, m); IR(nujol) 3400, 1375, 1325, 1160, 1065, 1015 cm⁻¹.

EXAMPLE 4 Preparation of 3-(Propylsulfonyl)-2-pyridinesulfonamide

To a stirred solution of 8.8 g (0.029 mol) of the product from Example 3in 400 mls methylene chloride cooled to -5°, under nitrogen, was added6.6 g (0.038 mol) of 3-chloroperbenzoic acid and stirred at roomtemperature for 20 hours. The reaction mixture was poured into water andextracted with methylene chloride. The organic layers were combined andwashed with saturated sodium bisulfite and brine, dried over magnesiumsulfate, and evaporated to a solid mixture which was washed with hexanesto afford a white solid. The solid was dissolved and stirred in 150 mlstrifluoroacetic acid for 72 hours. The solution was evaporated andtriturated with ether to afford 5.3 g (46%) white solid: m.p. 153°-157°;NMR (CDCl₃, 200 MHz) 1.06 (3H, t, J=7 Hz), 1.8 (2H, m), 3.7 (2H, m) 5.8(NH₂), 7.8 (1H, m), 8.6 (1H, m), 8.95 (1H, m); IR (nujol) 3390, 3180,1360, 1310, 1175, 1150 cm⁻¹.

EXAMPLE 5 Preparation ofN-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-3-(propylsulfonyl)-2-pyridinesulfonamide

To a stirred suspension of 0.4 g (0.0015 mol) of the product fromExample 4 and 0.63 g (0.0023 mol) of phenyl(4,6-dimethoxypyrimidin-2-yl)carbamate in 4 mls acetonitrile was added0.35 g (0.0023 mol) of 1,8-diazabicyclo[5.4.0]undec-7-ene and stirredfor 30 minutes. The solution was diluted with water and acidified with 1normal hydrochloric acid. The resulting precipitate was collected andwashed with water and ether to afford 0.45 g (67%) white solid: m.p.168°-170°; NMR (CDCl₃, 200 MHz), 1.07 (3H, t, J=7 Hz), 1.85 (2H, m), 3.7(2H, m), 3.97 (6H, s), 5.8 (1H, s), 7.26 (NH), 7.8 (1H, m), 8.6 (1H, m),8.9 (1H, m), 12.9 (NH); IR (nujol) 3320, 1740, 1610, 1580, 1375, 1195,1170 cm⁻¹.

EXAMPLE 6 Preparation of 3-ethylthio-2-fluoropyridine

Using the procedure of Example 1, 40.0 g of 2-fluoropyridine (0.412 mol)was converted to 46.5 g (72%) of the title compound as an oil:NMR(CDCl₃, 200 MHz) 1.3 (3H, t, J=7 Hz), 2.95 (2H, q, J=7 Hz), 7.1 (1H,m), 7.7 (1H, m), 8.0 (1H, m); 1R (neat) 1585, 1565, 1410, 1230 cm⁻¹.

EXAMPLE 7 Preparation of 3-ethylthio-2-(phenylmethylthio)pyridine

Using the procedure of Example 2, 25.0 g (0.160 mol) of the product fromExample 6 was converted to 44.8 g (100%) of the title compound as ayellow liquid: NMR (CDCl₃, 200 MHz) 1.28 (3H, t, J=7 Hz), 2.9 (2H, q,J=7 Hz), 4.45 (2H, s), 7.0-7.6 (7H, m), 8.35 (1H, m); 1R (neat) 1610,1405 cm⁻¹.

EXAMPLE 8 Preparation ofN-(1,1-Dimethylethyl)-3-ethylsulfinyl-2-pyridinesulfonamide

Using the procedure of Example 3, 35.0 g (0.134 mol) of the product fromExample 7 was converted to 21.2 g (56%) of the title compound: m.p.129°-131°; NMR (CDCl₃, 200 MHz) 1.23 (9H, s), 1.28 (3H, t, J=7 Hz), 2.9(1H, m), 3.3 (1H, m), 5.2 (NH), 7.7 (1H, m), 8.55 (1H, m), 8.75 (1H, m);1R (nujol) 3100, 1320, 1155 cm⁻¹.

EXAMPLE 9 Preparation ofN-(1,1-Dimethylethyl)-3-ethylsulfonyl-2-pyridinesulfonamide

Using the first half of the procedure of Example 4 (i.e., the3-chloroperbenzoic acid reaction), 9.0 g (0.033 mol) of the product fromExample 9 was converted to 10.1 g (100%) of the title compound: m.p.58°-63°; NMR (CDCl₃, 200 MHz) 1.2 (3H, t, J=7 Hz), 1.2 (9H, s), 3.7 (2H,q, J=7 Hz), 6.1 (NH), 7.7 (1H, m), 8.55 (1H, m), 8.95 (1H, m); 1R(nujol) 3300, 1560, 1350, 1300, 1170, 1140 cm⁻¹.

EXAMPLE 10 Preparation of 3-ethylsulfonyl-2-pyridinesulfonamide

Using the second half of the procedure of Example 4 (i.e., thetrifluoroacetic acid reaction), 9.0 g (0.029 mol) of t-he product fromExample 9 was converted to 4.2 g (58%) of the title compound: m.p.211°-212.5°; NMR (DMSO-d₆, 200 MHz) 1.15 (3H, t, J=7 Hz), 3.4 (NH₂), 3.7(2H, q, J=7 Hz), 7.9 (1H, m), 8.5 (1H, m), 8.95 (1H, m); IR (nujol)3370, 3190, 1350, 1310, 1180 cm⁻¹.

EXAMPLE 11 Preparation ofN-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-3-ethylsulfonyl-2-pyridinesulfonamide

Using the procedure of Example 5, 0.60 g (0.0024 mol) of the productfrom Example 10 was converted to 0.70 g (70%) of the title compound:m.p. 160°-162°; NMR (CDCl₃, 200 MHz) 1.35 (3H, t, J=7 Hz), 3.7 (2H, q,J=7 Hz), 3.97 (6H, s), 5.8 (1H, s), 7.3 (NH), 7.75 (1H, m), 8.6 (1H, m),8.9 (1H, m), 12.95 (NH); IR (nujol) 3260, 1740, 1610, 1360, 1195, 1175cm⁻¹.

EXAMPLE 12 Preparation of 2,6-Difluoro-3-pyridinecarboxylic acid, methylester

To a stirred solution of 91 ml (0.182 mol) of 2.0 molar lithiumdiisopropylamide (in hexanes) in 200 mL dry tetrahydrofuran cooled to-70° under nitrogen was added dropwise a solution of 20.0 g of2,6-difluoropyridine (0.174 mol) in 75 mL dry tetrahydrofuran such thatthe temperature was maintained below -60°. The solution was stirred at-70° for 3 hours and was then added via a cannula to a solution 21.7 g(0.230 mol) of methyl chloroformate in 100 mL dry tetrahydrofuran cooledto -70° under nitrogen. After stirring another hour at -70°, the mixturewas poured into water and extracted with ether. The combined organiclayers were washed with brine, dried over magnesium sulfate, andevaporated to a semisolid which was purified by flash chromatography toafford 13.0 g (43%) orange oil: NMR (CDCl₃, 200 MHz) 3.95 (3H, s), 6.9(1H, m), 8.5 (1H, m); IR (neat) 1745, 1730, 1610, 1415, 1290 cm⁻¹.

EXAMPLE 13 Preparation of 2-Fluoro-6-Methoxy-3-Pyridinecarboxylic Acid,Methyl Ester

To a stirred solution of 15.0 g (0.0867 mol) of the product from Example12 in 240 mL dry tetrahydrofuran cooled to -78° was added dropwise 22.7mL (0.0993 mol) of 25% sodium methoxide in methanol solution over 45minutes. After warming to -20°, the mixture was poured into ice water,acidified with 1 normal hydrochloric acid and extracted with ether. Thecombined organic layers were washed with brine, dried over magnesiumsulfate, and evaporated to a semisolid which was purified by flashchromatography to afford 3.2 g (17%) light yellow solid: m.p. 81°-82°;NMR (CDCl₃, 200 MHz) 3.9 (3H, s), 3.98 (3H, s), 6.67 (1H, d, J=9 Hz),8.25 (1H, m); IR (nujol) 1715, 1615, 1290 cm⁻¹.

EXAMPLE 14 Preparation of6-Methoxy-2-(Phenylmethylthio)-3-Pyridinecarboxylic Acid, Methyl Ester

To a stirred mixture of 0.8 g (0.0161 mol) of 50% sodium hydride (inmineral oil), which had been washed with hexanes, in 20 mL drydimethylformamide cooled to -5° under nitrogen was added dropwise 1.9 mL(0.0161 mol) benzyl mercaptan. The suspension was stirred at roomtemperature for 1 hour, cooled to 0°, and a solution of 3.2 g (0.0147mol) of the product of Example 13 in 20 mL dry dimethylformamide wasadded dropwise. After warming to room temperature, the solution waspoured into water and extracted with ether. The combined organic layerswere washed with water and with brine, dried over magnesium sulfate, andevaporated to an oil which was purified by flash chromatography toafford 3.0 g (64%) of a yellow solid: m.p. 67°-71°; NMR (CDCl₃, 200 MHz)3.88 (3H, s), 3.96 (3H, s), 4.46 (2H, s), 6.44 (1H, d, J=9Hz ), 7.2-7.5(5H, m), 8.1 (1H, d, J=9Hz ); IR (nujol) 1700, 1580, 1305, 1255 cm⁻¹.

EXAMPLE 15 Preparation of2-[1,1-Dimethylethyl)Aminosulfonyl]-6-Methoxy-3-Pyridinecarboxylic Acid,Methyl Ester

To a vigorously stirred mixture of 3.7 g (0.0129 mol) of the productfrom Example 14 in 79 mL methylene chloride and 41 mL water cooled to 0°was added 6.3 mL (0.0759 mol) concentrated-hydrochloric acid followed bythe dropwise addition of 79 mL (0.053 mol) of a 5% sodium hypochloritesolution such that the temperature was maintained below 5°. After themixture was stirred for an additional 30 minutes at 0° the reaction waspoured into water and extracted with methylene chloride. The combinedorganic layers were washed with brine, dried over magnesium sulfate, andfiltered. The filtrate was stirred and cooled to -70° under nitrogen,and 4.7 (0.0645 mol) of t-butyl amine was added dropwise. The reactionmixture was allowed to warm to -20°, poured into water, acidified with 1normal hydrochloric acid, and extracted with methylene chloride. Thecombined organic layers were washed with brine, dried over magnesiumsulfate, and evaporated to a semisolid which was purified by flashchromatography to afford 3.0 g (77%) yellow solid: m.p. 128°-130°; NMR(CDCl₃, 200 MHz) 1.27 (9H, s), 3.94 (3H, s), 4.05 (3H, s) 5.75 (NH), 6.9(1H, d, J=9 Hz), 7.95 (1H, d, J=9 HZ); IR (nujol) 3260, 1740, 1605,1325, 1125 cm⁻¹.

EXAMPLE 16 Preparation of2-(Aminosulfonyl)-6-Methoxy-3-Pyridine-Carboxylic Acid, Methyl Ester

A solution of 2.9 g (0.0096 mol) of the product from Example 15 wasstirred in 50 mL trifluoroacetic acid at room temperature for 20 hours.The solution was evaporated to afford 2.4 g (100%) white solid: m.p.142.5°-144.5°; NMR (CDCl, 200 MHz) 3.97 (3H, s), 4.1 (3H, s), 5.6 (NH₂),6.9 (1H, d, J=9Hz), 8.1 (1H, d, J=9Hz); 1R (nujol) 3305, 3205, 1715,1590, 1355, 1320, 1175 cm⁻¹.

EXAMPLE 17 Preparation of 2-[[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]aminosulfonyl]-6-Methoxy-3-Pyridine-carboxylic Acid,Methyl Ester

To a stirred suspension of 0.4 g (0.0016 mol) of the product fromExample 16 and 0.54 g (0.002 mol) of phenyl(4,6-dimethoxypyrimidin-2-yl)carbamate in 4 mL acetonitrile was added dropwise 0.30 g (0.002 mol) of1,8-diazobicyclo[5.4.0]undec-7-ene and stirred for 30 minutes. Thesolution was diluted with water and acidified with 1 normal hydrochloricacid. The resulting precipitate was collected and washed with water andwith ether to afford 0.57 g (84%) white solid: m.p. 194°-196°; NMR(CDCl₃, 200 MHz), 3.83 (3H, s), 3.95 (9H, s), 5.8 (1H, s), 6.95 (1H, d,J=9 Hz), 7.4 (NH), 8.1 (1H, d, J=9 Hz), 12.8 (NH); IR (nujol) 3140,1740, 1720, 1640, 1360, 1195, 1140 cm⁻¹.

EXAMPLE 18 Preparation ofN-(1,1-Dimethylethyl)-2-Fluoro-3-Pyridinesulfonamide

To a stirred solution of 396 mL (0.740 mol) of 1.9 molar lithiumdiisopropylamide (in hexanes) in 1.5 L dry tetrahydrofuran cooled to-70° under nitrogen was added dropwise a solution of 65 g (0.670 mol) of2-fluoropyridine in 150 mL dry tetrahydrofuran such that the temperaturewas maintained below -65°. The suspension was stirred at -70° foranother 3.5 hours and 86 g (1.34 mol) of sulfur dioxide was added whilemaintaining the temperature below -65°. After stirring another 15minutes at -70°, the reaction was allowed to warm to 0° and evaporatedto half the original volume and diluted with ether. The whiteprecipitate was collected under nitrogen, washed with ether, and dried.The solid was dissolved in 800 mL acetic acid and cooled to 10°-20°. Tothis stirred solution was added portionwise 99.4 g (0.740 mol) ofN-chlorosuccinimide while maintaining the temperature below 20°. Afterstirring another 30 minutes, the suspension was evaporated, diluted withwater and extracted with methylene chloride. The combined organic phaseswere washed with saturated aqueous sodium bicarbonate solution until nomore gas evolution, washed with brine, dried over magnesium sulfate, andfiltered. The filtrate was cooled to -70° under nitrogen and to thisstirred solution was added dropwise 199 g (2.7 mol) of t-butylamine. Thesuspension was poured into ice water, acidified with concentratedhydrochloric acid, and extracted with methylene chloride. The combinedorganic layers were washed with brine, dried over magnesium sulfate, andevaporated to an oil which was purified by flash chromatography toafford 29.1 g (19%) of a brown solid which was further washed with coldn-butylchloride to afford 22.4 g (14.5%) of a white solid: m.p. 95°-97°;NMR (CDCl₃, 200 MHz) 1.25 (9H, s), 4.9 (NH), 7.35 (1H, m), 8.3-8.5 (2H,m).

EXAMPLE 19 Preparation ofN-(1,1-Dimethylethyl)-2-Fluoro-N-Methyl-3-Pyridinesulfonamide

To a stirred suspension of 3.4 g (0.071 mol) of 50% sodium hydride (inmineral oil), which had been washed with hexanes, in 120 mL drydimethyldormamide cooled to 0° under nitrogen was added dropwise asolution of 15.0 g (0.065 mol) of the product from Example 18 in 120 mLdry dimethylformamide. After stirring at room temperature for 1 hour,the mixture was cooled to 0° and 12.2 g (0.086 mol) of methyl iodide wasadded dropwise. After warming to room temperature the reaction waspoured into ice water and extracted with ether. The combined organiclayers were washed with brine, dried over magnesium sulfate, andevaporated to 15.9 g (99%) oil; NMR (CDCl₃, 200 MHz), 1.32 (9H, s), 3.1(3H, s), 7.3 (1H, m), 8.3-8.4 (2H, m); 1R (neat) 1590, 1570, 1335, 1155cm⁻¹.

EXAMPLE 20 Preparation ofN-(1,1-Dimethylethyl)-N-Methyl-2-(Phenylmethylthio)-3-Pyridinesulfonamide

Using the same procedure as in Example 14, 15.9 g (0.065 mol) of theproduct from Example 19 was converted to 19.5 g (86%) yellow solid: m.p.92°-94°; NMR (CDCl₃), 200 MHz) 1.26 (9H, s), 3.1 (3H, s), 4.5 (2H, s),7.0-7.5 (6H, m), 8.2 (1H, m); IR (nujol) 1570, 1385, 1315, 1150, 1120cm⁻¹.

EXAMPLE 21 Preparation of N2,N3=Bis(1,1-Dimethylethyl)-N3-Methyl-2,3-Pyridinedisulfonamide

Using the same procedure as in Example 15, 19.5 g (0.056 mol) of theproduct from Example 20 was converted to a tan solid which was washedwith n-butylchloride to afford 13.1 g (66%) white solid: m.p.155°-156.5°; NMR (CDCl₃, 200 MHz) 1.23 (9H, s), 1.33 (9H, s), 3.1 (3H,s), 6.0 (NH), 1H, m), 8.5 (1H, m), 8.8 (1H, m); 1R (nujol) 3320, 1340,1325, 1160, 1120 cm⁻¹.

EXAMPLE 22 Preparation of N3-Methyl-2,3-Pyridinedisulfonamide

A stirred solution of 13.1 g (0.036 mol) of the product from Example 21in 150 mL trifluoroacetic acid was refluxed for 5 hours. After coolingto room temperature, the solution was evaporated to a solid which waswashed with ether to afford 9.6 g (100%) white solid: m.p. 220°-223°;NMR (DMSO-d₆, 200 MHz), 2.5 (3H, d), 6.9 (NH), 7.65 (NH₂), 7.85 (1H, m),8.45 (1H, m), 8.9 (1H, m); IR (nujol) 3380, 3320, 3180, 1355, 1170 cm⁻¹.

EXAMPLE 23 Preparation ofN2-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-N3-Methyl-2,3-Pyridinedisulfonamide

To a stirred suspension of 4.15 g (0.0165 mol) of the product fromExample 22 and 5.0 g (0.018 mol) of phenyl(4,6-dimethoxypyrimidin-2-yl)carbamate in 50 mL acetonitrile was addeddropwise 2.8 g (0.018 mol) of 1,8-diazabicyclo[5.4.0]undec-4-ene andstirred for 30 minutes. The solution was diluted with water andacidified with 1 normal hydrochloric acid. The resulting precipitate wascollected and washed with water and with ether to afford 6.4 g (82%)white solid: m.p. 147°-148.5°; NMR (CDCl₃, 200 MHz) 2.7 (3H, d, J=7 Hz),3.97 (6H, s), 5.8 (1H, s), 6.15 (1H, m), 7.3 (NH), 7.7 (1H, m), 8.55(1H, m), 8.8 (1H, m), 13.1 (NH); IR (nujol) 3310, 1740, 1610, 1340,1190, 1165 cm⁻¹.

By applying the procedures of Examples 1 through 23 and Equations 1through 19, the compounds in Tables I through X can be prepared by oneskilled in the art. ##STR54##

                                      TABLE I                                     __________________________________________________________________________    General Formula 1                                                             R.sub.1 R.sub.2      R   X      Y     Z   m.p.(°C.)                    __________________________________________________________________________    H       SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  170-174                             H       SOCH.sub.3   H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  138-140                             H       SOCH.sub.3   H   Cl     OCH.sub.3                                                                           CH  124-126                             H       SOCH.sub.3   H   CH.sub.3                                                                             CH.sub.3                                                                            CH    126-127.5                         H       SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SOCH.sub.3   H   OCH.sub.3                                                                            CH.sub.3                                                                            N   165-167                             H       SOCH.sub.3   H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SOCH.sub.3   CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N   133-137                             4-CH.sub.3                                                                            SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  170-172                             H       SO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  158-160                             H       SO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH  158-160                             H       SO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH  162-164                             H       SO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   180-184                             H       SO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N     154-156.5                         H       SO.sub.2 CH.sub.3                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  132-136                             H       SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  141-144                             H       SOCH.sub.2 CH.sub.3                                                                        H   Cl     OCH.sub.3                                                                           CH    105-107.5                         H       SOCH.sub.2 CH.sub.3                                                                        H   CH.sub. 3                                                                            CH.sub.3                                                                            CH    153-156.5                         H       SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   154-158                             H       SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N   172-174                             H       SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SOCH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  160-162                             H       SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  160-162                             H       SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH    163-164.5                         H       SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH  167-169                             H       SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   155-158                             H       SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N   165.5-168                           H       SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N   137-138                             4-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  178-180                             6-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  169.5-172                           6-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH    172-173.5                         6-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N   133-135                             6-OCH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  210-213                             6-F     SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  157-160                             6-F     SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH  176-177                             6-Cl    SO.sub.2 CH.sub. 2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  187-189                             6-Cl    SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH  171-174                             6-Cl    SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH  181-182                             6-SCH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH                                      5-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  159-160                             5-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH  176-177                             5-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   155-156                             5-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N   159-161                             H       SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  111-115                             H       SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  141-145                             H       SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   Cl     OCH.sub.3                                                                           CH  111-113                             H       SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   CH.sub.3                                                                             CH.sub.3                                                                            CH  173-175                             H       SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub. 3                                                                          N   186-189                             H       SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            N   164-166                             H       SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N   121-123                             H       SOCH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  168-170                             H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  157-159                             H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   Cl     OCH.sub.3                                                                           CH  165-167                             H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH  158-160                             H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   164-166                             H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N   165-168                             H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N   148-152                             H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  144-147                             H       SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH    143-145.5                         H       SOCH(CH.sub.3).sub.2                                                                       H   Cl     OCH.sub.3                                                                           CH  133-135                             H       SOCH(CH.sub.3).sub.2                                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH  150-153                             H       SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   155-159                             H       SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N   150-153                             H       SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SOCH(CH.sub.3).sub.2                                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  140-146                             H       SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            CH    159-160.5                         H       SO.sub.2 CH(CH.sub.3).sub.2                                                                H   Cl     OCH.sub.3                                                                           CH    164-165.5                         H       SO.sub.2 CH(CH.sub.3).sub.2                                                                H   CH.sub.3                                                                             CH.sub.3                                                                            CH  161-163                             H       SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   164-166                             H       SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            N   165-167                             H       SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 CH(CH.sub.3).sub.2                                                                CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N   145-149                             4-CH.sub.3                                                                            SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 CH(CH.sub.3).sub.2                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   Cl     OCH.sub.3                                                                           CH                                      H       SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  155-157                             H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  142-144                             H       SO.sub.2 CH.sub. 2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   Cl     OCH.sub.3                                                                           CH  151-153                             H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   CH.sub.3                                                                             CH.sub.3                                                                            CH  142-143                             H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   153.5-155                           H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            N   142.5-145.5                         H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               CH.sub.3                                                                          OCH.sub.3                                                                            OCH.sub.3                                                                           N   133-136                             4-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.3                                                                            OCH.sub. 3                                                                          CH                                      6-F     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       S-cyclopropyl                                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       S-cyclopropyl                                                                              H   Cl     OCH.sub.3                                                                           CH                                      H       S-cyclopropyl                                                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       S-cyclopropyl                                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       S-cyclopropyl                                                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       S-cyclopropyl                                                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO-cyclopropyl                                                                             H   Cl     OCH.sub.3                                                                           CH                                      H       SO-cyclopropyl                                                                             H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO-cyclopropyl                                                                             H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO-cyclopropyl                                                                             CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 -cyclopropyl                                                                      H   Cl     OCH.sub.3                                                                           CH                                      H       SO.sub.2 -cyclopropyl                                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 -cyclopropyl                                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub. 2 -cyclopropyl                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  169-171                             H       OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            CH.sub.3                                                                            CH    172-173.5                         H       OSO.sub.2 CH.sub.3                                                                         H   Cl     OCH.sub.3                                                                           CH  171-173                             H       OSO.sub.2 CH.sub.3                                                                         H   CH.sub.3                                                                             CH.sub.3                                                                            CH  161.5-165                           H       OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            CH.sub.3                                                                            N   155-158                             H       OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       OSO.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH    162-163.5                         H       OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  160-162                             H       OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   Cl     OCH.sub.3                                                                           CH  139-143                             H       OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   CH.sub.3                                                                             CH.sub.3                                                                            CH  132-138                             H       OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   171.5-173                           H       OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            N   147-149                             H       OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       OSO.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH.sub. 2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  156-157                             H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  131-133                             H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   Cl     OCH.sub.3                                                                           CH  127-132                             H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH  152-153                             H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   154-155                             H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub. 3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   Cl     OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       OSO.sub.2 CH(CH.sub.3).sub.2                                                               CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    OSO.sub.2 CH(CH.sub.3).sub.2                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   Cl     OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub. 3                                                                          CH                                      6-OCH.sub.3                                                                           OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH   CH                                      6-F     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  140-142                             H       OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       OSO.sub.2 CF.sub.3                                                                         H   Cl     OCH.sub.3                                                                           CH  154-156                             H       OSO.sub.2 CF.sub.3                                                                         H   CH.sub.3                                                                             CH.sub.3                                                                            CH  157-160                             H       OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   164-166                             H       OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            CH.sub.3                                                                            N   157-159                             H       OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       OSO.sub.2 CF.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       OSO.sub.2 CCl.sub.3                                                                        H   Cl     OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CCl.sub.3                                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       OSO.sub.2 CCl.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   Cl     OCH.sub.3                                                                           CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   Cl     OCH.sub.3                                                                           CH                                      H       SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 OCH.sub.2 CF.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 OCH.sub.3                                                                         H   Cl     OCH.sub.3                                                                           CH                                      H       SO.sub.2 OCH.sub.3                                                                         H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 OCH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 OCH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   Cl     OCH.sub.3                                                                           CH                                      H       SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 OCH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 OCH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       N.sub.3      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       N.sub.3      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       N.sub.3      H   Cl     OCH.sub.3                                                                           CH                                      H       N.sub.3      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       N.sub.3      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       N.sub.3      H   OCH.sub.3                                                                            CH.sub. 3                                                                           N                                       H       N.sub.3      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       N.sub.3      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            N.sub.3      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           N.sub.3      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            N.sub.3      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           N.sub.3      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     N.sub.3      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    N.sub.3      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CN           H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CN           H   Cl     OCH.sub.3                                                                           CH                                      H       CN           H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CN           H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CN           H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CN           CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       P(O)(OCH.sub.3).sub.2                                                                      H   Cl     OCH.sub.3                                                                           CH                                      H       P(O)(OCH.sub.3).sub.2                                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       P(O)(OCH.sub.3).sub.2                                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  108-111                             H       P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   Cl     OCH.sub.3                                                                           CH                                      H       P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   CH.sub.3                                                                             CH.sub.3                                                                            CH  110-114                             H       P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    P(O)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       P(S)(OCH.sub.3).sub.2                                                                      H   Cl     OCH.sub.3                                                                           CH                                      H       P(S)(OCH.sub.3).sub.2                                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       P(S)(OCH.sub.3).sub.2                                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    P(S)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   Cl     OCH.sub.3                                                                           CH                                      H       P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    P(S)(OCH.sub.2 CH.sub.3).sub.2                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CH.sub.2 F   H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CH.sub.2 F   H   Cl     OCH.sub.3                                                                           CH                                      H       CH.sub.2 F   H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CH.sub.2 F   H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CH.sub.2 F   H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CH.sub.2 F   CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CF.sub.2 H   H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CF.sub.2 H   H   Cl     OCH.sub.3                                                                           CH                                      H       CF.sub.2 H   H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CF.sub.2 H   H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CF.sub.2 H   H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CF.sub.2 H   CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CH.sub.2 Cl  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CH.sub.2 Cl  H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CH.sub.2 Cl  H   Cl     OCH.sub.3                                                                           CH                                      H       CH.sub.2 Cl  H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CH.sub.2 Cl  H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CH.sub.2 Cl  H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CH.sub.2 Cl  H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CH.sub.2 Cl  CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CH.sub.2 Cl  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CH.sub.2 Cl  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CH.sub.2 Cl  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CH.sub.2 Cl  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CH.sub.2 Cl  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CH.sub.2 Cl  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CCl.sub.2 H  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CCl.sub.2 H  H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CCl.sub.2 H  H   Cl     OCH.sub.3                                                                           CH                                      H       CCl.sub.2 H  H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CCl.sub.2 H  H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CCl.sub.2 H  H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CCl.sub.2 H  H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CCl.sub.2 H  CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CCl.sub.2 H  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CCl.sub.2 H  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CCl.sub.2 H  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CCl.sub.2 H  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CCl.sub.2 H  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CCl.sub.2 H  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CH.sub.2 CH.sub.2 Cl                                                                       H   Cl     OCH.sub.3                                                                           CH                                      H       CH.sub.2 CH.sub.2 Cl                                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CH.sub.2 CH.sub.2 Cl                                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CH.sub.2 CH.sub.2 Cl                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CH.sub.2 CH.sub.2 Br                                                                       H   Cl     OCH.sub.3                                                                           CH                                      H       CH.sub.2 CH.sub.2 Br                                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CH.sub.2 CH.sub.2 Br                                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CH.sub.2 CH.sub.2 Br                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CHFCH.sub.3  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CRFCH.sub.3  H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CHFCH.sub.3  H   Cl     OCH.sub.3                                                                           CH                                      H       CHFCH.sub.3  H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CHFCH.sub.3  H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CHFCH.sub.3  H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CHFCH.sub.3  H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CHFCH.sub.3  CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CHFCH.sub.3  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CHFCH.sub.3  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CHFCH.sub.3  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CHFCH.sub.3  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CHFCH.sub.3  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CHFCH.sub.3  H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CHClCH.sub.3 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CHClCH.sub.3 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CHClCH.sub.3 H   Cl     OCH.sub.3                                                                           CH                                      H       CHClCH.sub.3 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CHClCH.sub. 3                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CHClCH.sub.3 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CHClCH.sub.3 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CHClCH.sub.3 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CHClCH.sub.3 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CHClCH.sub.3 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CHClCH.sub.3 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CHClCH.sub.3 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CHClCH.sub.3 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CHClCH.sub.3 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CF.sub.2 CF.sub.2 H                                                                        H   Cl     OCH.sub.3                                                                           CH                                      H       CF.sub.2 CF.sub.2 H                                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CF.sub.2 CF.sub.2 H                                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CF.sub.2 CF.sub.2 H                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.2 CH.sub.3                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.2 CH.sub.3                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-CH.sub.2 CH.sub.3                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-CH.sub.2 CH.sub.3                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-CH.sub.2 CH.sub.3                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-CH.sub.2 CH.sub.3                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-CH.sub.2 CH.sub.3                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-CH.sub.2 CH.sub.3                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 CH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            N                                       6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-OCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-OCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-OCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-OCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 N(CH.sub.3).sub.2                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.3).sub.2                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub. 3                                                                         N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.3).sub.2                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-NHCH.sub.3                                                                          SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-NHCH.sub.3                                                                          SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-NHCH.sub.3                                                                          SO.sub.2 N(CH.sub.3).sub.2                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-NHCH.sub.3                                                                          SO.sub.2 N(CH.sub.3).sub.2                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-NHCH.sub.3                                                                          SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-NHCH.sub.3                                                                          SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-NHCH.sub.3                                                                          SO.sub.2 N(CH.sub.3).sub.2                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-NHCH.sub.3                                                                          SO.sub.2 N(CH.sub.3).sub.2                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   Cl     OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   Cl     OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-SCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub. 2 CH.sub.3).sub.2                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   Cl     OCH.sub.3                                                                           CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 N(CH.sub.2 CH.sub.3).sub.2                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   Cl     OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-SCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-SCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 NHOCH.sub.3                                                                       H   Cl     OCH.sub.3                                                                           CH                                      6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 NHOCH.sub.3                                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-SCH.sub.2 CH.sub.3                                                                  SO.sub.2 NHOCH.sub.3                                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 NHOCH.sub.3                                                                       H   Cl     OCH.sub.3                                                                           CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 NHOCH.sub.3                                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-N(CH.sub.3).sub.2                                                                   SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-N(CH.sub.3).sub.2                                                                   SO.sub.2 NHOCH.sub.3                                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   Cl     OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-OCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCH.sub.3                                                                           SO.sub.2 NHOCH.sub.3                                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   Cl     OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   Cl     OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-SCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-SCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH    147-148.5                         H       SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.3                                                                        H   Cl     OCH.sub.3                                                                           CH  155-157                             H       SO.sub.2 NHCH.sub.3                                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH  150-152                             H       SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N   153.5-155                           H       SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHCH.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH    163-165.5                         H       SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   Cl     OCH.sub.3                                                                           CH  158.5-161                           H       SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   CH.sub.3                                                                             CH.sub.3                                                                            CH    118-121.5                         H       SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   162-164                             H       SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            N   158-160                             H       SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N     122-125.5                         4-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  138.5-141                           H       SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  117-120                             H       SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   Cl     OCH.sub.3                                                                           CH  125-129                             H       SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 CH.sub. 2 CH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   132-135                             H       SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  164-166                             H       SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                H       SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   Cl     OCH.sub.3                                                                           CH  153.5-156                           H       SO.sub. 2 NHCH(CH.sub.3).sub.2                                                             H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   149-152                             H       SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   149-151                             H       SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHCH(CH.sub.3).sub.2                                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N   141-143                             4-CH.sub.3                                                                            SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 NHcyclopropyl                                                                     H   Cl     OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHcyclopropyl                                                                     H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHcyclopropyl                                                                     CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHcyclopropyl                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   CL     OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   Cl     OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHCH.sub.2 C.tbd. CH                                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH   SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHCH.sub.2 C.tbd.CH                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   CL     OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 NHCH.sub. 2 OCH.sub.3                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHCH.sub.2 OCH.sub.3                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   Cl     OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHCH.sub.2 CF.sub.3                                                               CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub. 2 NHCH.sub.2 CF.sub.3                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH   SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 CN                                                                     H   CL     OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CN                                                                     H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHCH.sub.2 CN                                                                     CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   Cl     OCH.sub.3                                                                           CH                                      H       SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 -pyrrolidino                                                                      H   CL     OCH.sub.3                                                                           CH                                      H       SO.sub.2 -pyrrolidino                                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 -pyrrolidino                                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   Cl     OCH.sub.3                                                                           CH                                      H       SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  146-149                             H       SO.sub.2 -pyrrolidino                                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH  169-171                             6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH                                      6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.3                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  194-196                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  165-167                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH  173-175                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH  138.5-145                           6-OCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   173-176                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N   158-161                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  154-157                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  160-162                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH  130-132                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH  140-141                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   160-162                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N   152-153                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCF.sub. 3                                                                          CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCF.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-OCF.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH                                      6-OCF.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-OCF.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-OCF.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  158-162                             6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  168-170                             6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH  149-150                             6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH  150-152                             6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCF.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub. 2 CH.sub.3                                                                  NHCH.sub.3                                                                          N                                       6-OCF.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH                                      6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.3                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-SCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-SCH.sub.3                                                                           CO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH                                      6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  164-167                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  178-179                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH  147-150                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH  164-165                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   171-172                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N   132-134                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.3                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N   152-155                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.3                                                                          H   Cl     OCH.sub.3                                                                           CH                                      6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.3                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.3                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.3                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-CH.sub.2 CH.sub.3                                                                   CO.sub. 2 CH.sub.2 CH.sub.3                                                                H   Cl     OCH.sub.3                                                                           CH                                      6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-CH.sub.2 CH.sub.3                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  158-161                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  147-149                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH  124-127                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH  149-151                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   164-165                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N   131-132                             6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub. 3                                                                  NHCH.sub.3                                                                          N                                       6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  152-154                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  134-135                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH  153-160                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH  159-163                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   320-330                             6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  173-175                             6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  166-167                             6-OCH.sub.2 CF.sub.3                                                                  CO.sub. 2 CH.sub.2 CH.sub.3                                                                H   Cl     OCH.sub.3                                                                           CH  150-152                             6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH  142-144                             6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   138-141                             6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N   122-126                             6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCH.sub.2 CF.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCF.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCF.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-OCF.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-OCF.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-OCF.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-OCF.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCF.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCF.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-OCF.sub.2 H                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-SCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-SCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-SCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-SCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-SCH.sub.2 CH.sub.3                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  147-149                             6-N(CH.sub. 3).sub.2                                                                  CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  149-150                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH  150-151                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH  172-175                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   152-153                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N   148-150                             6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-N(CH.sub.3).sub.2                                                                   CO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH                                      6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       6-NHCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   Cl     OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   Cl     OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   Cl     OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CO.sub. 2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   Cl     OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CF.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CO.sub.2 CH.sub.2 CF.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  127-128                             H       CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH  142-144                             H       CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   Cl     OCH.sub.3                                                                           CH  154-156                             H       CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH  141-142                             H       CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   137-138                             H       CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub. 3                                                                           CH.sub.3                                                                            N   136-137                             H       CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CO.sub.2 CH.sub.2 C.tbd.CH                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CO.sub.2 CH.sub.2 C.tbd.CH                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   Cl     OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CO.sub.2 CH.sub. 2 CH.sub.2 CH.sub.2 Cl                                                    H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 Cl                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   Cl     OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                      H       CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                       H       CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                       4-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      4-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                            CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-OCH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-F     CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl    CO.sub.2 CH.sub.2 CH.sub.2 SCH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H       CO.sub.2 CH.sub.2 -cyclopropyl                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH  143-145                             H       CO.sub.2 CH.sub.2 -cyclopropyl                                                             H   Cl     OCH.sub.3                                                                           CH  124-128                             H       CO.sub.2 CH.sub.2 -cyclopropyl                                                             H   CH.sub.3                                                                             CH.sub. 3                                                                           CH  134-138                             H       CO.sub.2 CH.sub.2 -cyclopropyl                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           N   154-161                             __________________________________________________________________________

                                      TABLE II                                    __________________________________________________________________________    General Formula 2                                                             R.sub.1                                                                             R.sub.3      R   X      Y     Z   m.p. (°C.)                     __________________________________________________________________________    H     SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SOCH.sub.3   H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SOCH.sub.3   H   Cl     OCH.sub.3                                                                           CH                                        H     SOCH.sub.3   H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SOCH.sub.3   H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SOCH.sub.3   CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SOCH.sub.3   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SOCH.sub.2 CH.sub.3                                                                        H   Cl     OCH.sub.3                                                                           CH                                        H     SOCH.sub.2 CH.sub.3                                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SOCH.sub.2 CH.sub. 3                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SOCH.sub.2 CH.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SOCH.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   Cl     OCH.sub.3                                                                           CH                                        H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub. 3                                                                           OCH.sub.3                                                                           CH                                        4-Cl  SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SOCH.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   Cl     OCH.sub.3                                                                           CH                                        H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub. 3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SOCH(CH.sub.3).sub.2                                                                       H   Cl     OCH.sub.3                                                                           CH                                        H     SOCH(CH.sub.3).sub.2                                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SOCH(CE.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SOCH(CH.sub.3).sub.2                                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub. 3                                                                           OCH.sub.3                                                                           CH                                        6-Cl  SOCH(CH.sub.3).sub.2                                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     S-cyclopropyl                                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     S-cyclopropyl                                                                              H   Cl     OCH.sub.3                                                                           CH                                        H     S-cyclopropyl                                                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     S-cyclopropyl                                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     S-cyclopropyl                                                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     S-cyclopropyl                                                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  S-cyclopropyl                                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO-cyclopropyl                                                                             H   Cl     OCH.sub.3                                                                           CH                                        H     SO-cyclopropyl                                                                             H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO-cyclopropyl                                                                             H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO-cyclopropyl                                                                             CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO-cyclopropyl                                                                             H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 -cyclopropyl                                                                      H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 -cyclopropyl                                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 -cyclopropyl                                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 -cyclopropyl                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     OSO.sub.2 CH.sub.3                                                                         H   Cl     OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CH.sub.3                                                                         H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     OSO.sub.2 CH.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  OSO.sub.2 CH.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   Cl     OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   CH.sub. 3                                                                            CH.sub.3                                                                            CH                                        H     OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     OSO.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  OSO.sub.2 CH.sub.2 CH.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     OSO.sub.2 CF.sub.3                                                                         H   Cl     OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CF.sub.3                                                                         H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     OSO.sub.2 CF.sub.3                                                                         CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   OSO.sub.2 CF.sub.3                                                                         H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  OSO.sub.2 CF.sub.3                                                                         H   OCO.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     OSO.sub.2 CCl.sub.3                                                                        H   Cl     OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CCl.sub.3                                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     OSO.sub.2 CCl.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  OSO.sub.2 CCl.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   Cl     OCH.sub.3                                                                           CH                                        H     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  OSO.sub.2 CH.sub. 2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H   OCO.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 OCH.sub.2 CF.sub.3                                                                CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 OCH.sub.2 CF.sub.3                                                                H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     P(O)(OCH.sub.3).sub.2                                                                      H   Cl     OCH.sub.3                                                                           CH                                        H     P(O)(OCH.sub.3).sub.2                                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     P(O)(OCH.sub.3).sub.2                                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         P(O)(OCH.sub.3).sub.2                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   P(O)(OCH.sub.3 ).sub.2                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  P(O)(OCH.sub.3).sub.2                                                                      H   OCO.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CN           H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     CN           H   Cl     OCH.sub.3                                                                           CH                                        H     CN           H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CN           H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     CN           H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     CN           CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CN           H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 F   H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     CH.sub.2 F   H   Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 F   H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 F   H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     CH.sub.2 F   H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     CH.sub.2 F   CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   CH.sub.2 F   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 F   H   OCO.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 H   H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     CF.sub.2 H   H   Cl     OCH.sub.3                                                                           CH                                        H     CF.sub.2 H   H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CF.sub.2 H   H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     CF.sub.2 H   H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     CF.sub.2 H   CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CF.sub.2 H   H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.3                                                                        H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.3                                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 NHCH.sub.3                                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 NHCH.sub.3                                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub. 2 NHCH.sub.2 CH.sub.3                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 NHCH.sub.2 CH.sub.3                                                               CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 NHCH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            CH.sub. 3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 NHCH(CH.sub.3).sub.2                                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 NHCH(CH.sub.3).sub.2                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 NH-cyclopropyl                                                                    H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 NH-cyclopropyl                                                                    H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 NH-cyclopropyl                                                                    CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 NH-cyclopropyl                                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            CH.sub. 3                                                                           N                                         H     SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 NHCH.sub.2 CH═CH.sub.2                                                        H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 NHCH.sub.2 CF.sub.3                                                               CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 NHCH.sub.2 CF.sub.3                                                               H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CN                                                                     H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CN                                                                     H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 NHCH.sub.2 CN                                                                     CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 NHCH.sub.2 CN                                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 N(CH.sub.2 CH═CH.sub. 2).sub.2                                                CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 N(CH.sub.2 CH═CH.sub.2).sub.2                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 -pyrrolidino                                                                      H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 -pyrrolidino                                                                      H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 -pyrrolidino                                                                      CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub. 3                                                                          CH                                        4-Cl  SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 -pyrrolidino                                                                      H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub. 3                                                    H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                     H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NH.sub.2                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     SO.sub.2 NH.sub.2                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     SO.sub.2 NH.sub.2                                                                          H   Cl     OCH.sub.3                                                                           CH                                        H     SO.sub.2 NH.sub.2                                                                          H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     SO.sub.2 NH.sub.2                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     SO.sub.2 NH.sub.2                                                                          H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     SO.sub.2 NH.sub.2                                                                          H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     SO.sub.2 NH.sub.2                                                                          CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          SO.sub.2 NH.sub.2                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  SO.sub.2 NH.sub.2                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          SO.sub.2 NH.sub.2                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         SO.sub.2 NH.sub.2                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   SO.sub.2 NH.sub.2                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  SO.sub.2 NH.sub.2                                                                          H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   Cl     OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CO.sub.2 CH.sub.2 CH.sub.2 OH                                                              H   OCO.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   Cl     OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub. 3                                                                          CH                                        6-F   CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CO.sub.2 CH.sub.2 CH.sub.2 CN                                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   Cl     OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                              H   OCO.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        H     CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   Cl     OCH.sub.3                                                                           CH                                        H     CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            CH.sub.3                                                                            N                                         H     CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.2 CH.sub.3                                                                   NHCH.sub.3                                                                          N                                         H     CO.sub.2 CH.sub.2 CF.sub.3                                                                 CH.sub.3                                                                          OCH.sub.3                                                                            CH.sub.3                                                                            N                                         4-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        4-Cl  CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-F   CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CO.sub.2 CH.sub.2 CF.sub.3                                                                 H   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        __________________________________________________________________________

                                      TABLE III                                   __________________________________________________________________________    General Formula 3                                                             R.sub.f                                                                            R.sub.4     R  X     Y    Z  m.p.(°C.)                            __________________________________________________________________________    H    SOCH.sub.3  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SOCH.sub.3  H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SOCH.sub.3  H  Cl    OCH.sub.3                                                                          CH                                             H    SOCH.sub.3  H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SOCH.sub.3  H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SOCH.sub.3  H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SOCH.sub.3  CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SOCH.sub.3  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SOCH.sub.3  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         SOCH.sub.3  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SOCH.sub.3  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SOCH.sub.3  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SOCH.sub.3  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SOCH.sub.2 CH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SOCH.sub.2 CH.sub.3                                                                       H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SOCH.sub.2 CH.sub.3                                                                       H  Cl    OCH.sub.3                                                                          CH                                             H    SOCH.sub.2 CH.sub.3                                                                       H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SOCH.sub.2 CH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SOCH.sub.2 CH.sub.3                                                                       H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SOCH.sub.2 CH.sub.3                                                                       CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SOCH.sub.2 CH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SOCH.sub.2 CH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         SOCH.sub.2 CH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SOCH.sub.2 CH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SOCH.sub.2 CH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SOCH.sub.2 CH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  Cl    OCH.sub.3                                                                          CH                                             H    SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SOCH.sub.2 CH.sub.2 CH.sub.3                                                              CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SOCH.sub.2 CH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  Cl    OCH.sub.3                                                                          CH                                             H    SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  OCH.sub.3                                                                           OCH.sub. 3                                                                         CH                                             6-CH.sub.3                                                                         SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SOCH(CH.sub.3).sub.2                                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SOCH(CH.sub.3).sub.2                                                                      H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SOCH(CH.sub.3).sub.2                                                                      H  Cl    OCH.sub.3                                                                          CH                                             H    SOCH(CH.sub.3).sub.2                                                                      H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SOCH(CH.sub.3).sub.2                                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SOCH(CH.sub.3).sub.2                                                                      H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SOCH(CH.sub.3).sub.2                                                                      CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SOCH(CH.sub.3).sub.2                                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SOCH(CH.sub.3).sub.2                                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         SOCH(CH.sub.3).sub.2                                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SOCH(CH.sub.3).sub.2                                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SOCH(CH.sub.3).sub.2                                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SOCH(CH.sub. 3).sub.2                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    S-cyclopropyl                                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    S-cyclopropyl                                                                             H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    S-cyclopropyl                                                                             H  Cl    OCH.sub.3                                                                          CH                                             H    S-cyclopropyl                                                                             H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    S-cyclopropyl                                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    S-cyclopropyl                                                                             H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    S-cyclopropyl                                                                             H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    S-cyclopropyl                                                                             CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl S-cyclopropyl                                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  S-cyclopropyl                                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         S-cyclopropyl                                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        S-cyclopropyl                                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  S-cyclopropyl                                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl S-cyclopropyl                                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO-cyclopropyl                                                                            H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO-cyclopropyl                                                                            H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SO-cyclopropyl                                                                            H  Cl    OCH.sub.3                                                                          CH                                             H    SO-cyclopropyl                                                                            H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SO-cyclopropyl                                                                            H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SO-cyclopropyl                                                                            H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SO-cyclopropyl                                                                            H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    SO-cyclopropyl                                                                            CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SO-cyclopropyl                                                                            H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SO-cyclopropyl                                                                            H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         SO-cyclopropyl                                                                            H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SO-cyclopropyl                                                                            H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SO-cyclopropyl                                                                            H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SO-cyclopropyl                                                                            H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SO.sub.2 -cyclopropyl                                                                     H  Cl    OCH.sub.3                                                                          CH                                             H    SO.sub.2 -cyclopropyl                                                                     H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    SO.sub.2 -cyclopropyl                                                                     CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SO.sub.2 -cyclopropyl                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CH.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CH.sub. 3                                                                       H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    OSO.sub.2 CH.sub.3                                                                        H  Cl    OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CH.sub.3                                                                        H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    OSO.sub.2 CH.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    OSO.sub.2 CH.sub.3                                                                        H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    OSO.sub.2 CH.sub.3                                                                        H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    OSO.sub.2 CH.sub.3                                                                        CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl OSO.sub.2 CH.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  OSO.sub.2 CH.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         OSO.sub.2 CH.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        OSO.sub.2 CH.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  OSO.sub.2 CH.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl OSO.sub.2 CH.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  Cl    OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    OSO.sub.2 CH.sub.2 CH.sub. 3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    OSO.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl OSO.sub.2 CH.sub.2 CH.sub.3                                                               H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  Cl    OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl OSO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    OSO.sub.2 CF.sub.3                                                                        H  Cl    OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CF.sub.3                                                                        H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    OSO.sub.2 CF.sub.3                                                                        CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl OSO.sub.2 CF.sub.3                                                                        H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    OSO.sub.2 CCl.sub.3                                                                       H  Cl    OCH.sub.3                                                                          CH                                             H    OSO.sub.2 CCl.sub.3                                                                       H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    OSO.sub.2 CCl.sub.3                                                                       CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub. 3                                                                         CH                                             2-F  OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl OSO.sub.2 CCl.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    N.sub.3     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    N.sub.3     H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    N.sub.3     H  Cl    OCH.sub.3                                                                          CH                                             H    N.sub.3     H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    N.sub.3     H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    N.sub.3     H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    N.sub.3     H  OCH.sub.2 CH.sub.3                                                                  NRCH.sub.3                                                                         N                                              H    N.sub.3     CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl N.sub.3     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  N.sub.3     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         N.sub.3     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        N.sub.3     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  N.sub.3     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl N.sub.3     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    P(O)(OCH.sub.3).sub.2                                                                     H  Cl    OCH.sub.3                                                                          CH                                             H    P(O)(OCH.sub.3).sub.2                                                                     H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    P(O)(OCH.sub.3).sub.2                                                                     CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl P(O)(OCH.sub.3).sub.2                                                                     H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CN          H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CN          H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    CN          H  Cl    OCH.sub.3                                                                          CH                                             H    CN          H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    CN          H  OCH.sub.3                                                                           OCH.sub.3                                                                          CN                                             H    CN          H  OCH.sub.3                                                                           CH.sub.3                                                                           CN                                             H    CN          H  OCH.sub.2 CH.sub. 3                                                                 NHCH.sub.3                                                                         CN                                             H    CN          CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           CN                                             2-Cl CN          H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  CN          H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         CN          H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        CN          H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  CN          H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl CN          H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CH.sub.2 F  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CH.sub.2 F  H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    CH.sub.2 F  H  Cl    OCH.sub.3                                                                          CH                                             H    CH.sub.2 F  H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    CH.sub.2 F  H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    CH.sub.2 F  H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    CH.sub.2 F  H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    CH.sub.2 F  CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl CH.sub.2 F  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  CH.sub.2 F  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         CH.sub.2 F  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        CH.sub.2 F  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  CH.sub.2 F  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl CH.sub.2 F  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CF.sub.2 H  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CF.sub.2 H  H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    CF.sub.2 H  H  Cl    OCH.sub.3                                                                          CH                                             H    CF.sub.2 H  H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    CF.sub.2 H  H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    CF.sub.2 H  H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    CF.sub.2 H  H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    CF.sub.2 H  CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl CF.sub.2 H  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  CF.sub.2 H  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         CF.sub.2 H  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        CF.sub.2 H  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  CF.sub.2 H  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl CF.sub.2 H  H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  Cl    OCH.sub.3                                                                          CH                                             H    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SO.sub.2 N(OCH.sub.3)CH.sub.3                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SO.sub.2 NHCH.sub.3                                                                       H  Cl    OCH.sub.3                                                                          CH                                             H    SO.sub.2 NHCH.sub.3                                                                       H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    SO.sub.2 NHCH.sub.3                                                                       CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SO.sub.2 NHCH.sub.3                                                                       H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  Cl    OCH.sub.3                                                                          CH                                             H    SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    SO.sub.2 NHCH.sub.2 CH.sub.3                                                              CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SO.sub.2 NHCH.sub.2 CH.sub.3                                                              H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  Cl    OCH.sub.3                                                                          CH                                             H    SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                    H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  Cl    OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             CH.sub. 3                                                                        OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl CO.sub.2 CH.sub.2 CH.sub.2 OH                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  Cl    OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             CH.sub.3                                                                         OCH.sub. 3                                                                          CH.sub.3                                                                           N                                              2-Cl CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl CO.sub.2 CH.sub.2 CH.sub.2 CN                                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  Cl    OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                              H    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                             H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CF.sub.3                                                                H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CF.sub.3                                                                H  OCH.sub.3                                                                           CH.sub.3                                                                           CH                                             H    CO.sub.2 CH.sub.2 CF.sub.3                                                                H  Cl    OCH.sub.3                                                                          CH                                             H    CO.sub.2 CH.sub.2 CF.sub.3                                                                H  CH.sub.3                                                                            CH.sub.3                                                                           CH                                             H    CO.sub.2 CH.sub.2 CF.sub.3                                                                H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    CO.sub.2 CH.sub. 2 CF.sub.3                                                               H  OCH.sub.3                                                                           CH.sub.3                                                                           N                                              H    CO.sub.2 CH.sub.2 CF.sub.3                                                                H  OCH.sub.3                                                                           OCH.sub.3                                                                          N                                              H    CO.sub.2 CH.sub.2 CF.sub.3                                                                CH.sub.3                                                                         OCH.sub.3                                                                           CH.sub.3                                                                           N                                              2-Cl CO.sub.2 CH.sub.2 CF.sub.3                                                                H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             2-F  CO.sub.2 CH.sub.2 CF.sub.3                                                                H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-CH.sub.3                                                                         CO.sub.2 CH.sub.2 CF.sub.3                                                                H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-OCH.sub.3                                                                        CO.sub.2 CH.sub.2 CF.sub.3                                                                H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-F  CO.sub.2 CH.sub.2 CF.sub.3                                                                H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             6-Cl CO.sub.2 CH.sub.2 CF.sub.3                                                                H  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                             __________________________________________________________________________

                                      TABLE IV                                    __________________________________________________________________________    General Formula 4                                                             R.sub.f                                                                              R.sub.5       R    X       Y      Z    m.p. (°C.)               __________________________________________________________________________    H      SOCH.sub.3    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SOCH.sub.3    H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SOCH.sub.3    H    Cl      OCH.sub.3                                                                            CH                                   H      SOCH.sub.3    H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SOCH.sub.3    H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SOCH.sub.3    H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SOCH.sub.3    H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SOCH.sub.3    CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SOCH.sub.3    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SOCH.sub.3    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SOCH.sub.3    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SOCH.sub.3    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SOCH.sub.3    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SOCH.sub.3    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.3                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.3                                                                           H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SO.sub.2 CH.sub.3                                                                           H    Cl      OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.3                                                                           H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SO.sub.2 CH.sub.3                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SO.sub.2 CH.sub.3                                                                           H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SO.sub.2 CH.sub.3                                                                           H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SO.sub.2 CH.sub.3                                                                           CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SO.sub.2 CH.sub.3                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO.sub.2 CH.sub.3                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2 CH.sub.3                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SO.sub.2 CH.sub.3                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SO.sub.2 CH.sub.3                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SO.sub.2 CH.sub.3                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SOCH.sub.2 CH.sub.3                                                                         H    Cl      OCH.sub.3                                                                            CH                                   H      SOCH.sub.2 CH.sub.3                                                                         H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub. 2 CH.sub.3                                                                   NHCH.sub.3                                                                           N                                    H      SOCH.sub.2 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SOCH.sub.2 CH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    Cl      OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SO.sub.2 CH.sub.2 CH.sub.3                                                                  CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SO.sub.2 CH.sub.2 CH.sub.3                                                                  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    Cl      OCH.sub.3                                                                            CH                                   H      SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SOCH.sub.2 CH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SOCH.sub.2 CH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    Cl      OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.3                                                                             OCH.sub. 3                                                                           CH                                   5-OCH.sub.3                                                                          SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    Cl      OCH.sub.3                                                                            CH                                   H      SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub. 3                                                                            N                                    5-CH.sub.3                                                                           SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    Cl      OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SOCH(CH.sub.3).sub.2                                                                        H    Cl      OCH.sub.3                                                                            CH                                   H      SOCH(CH.sub.3).sub.2                                                                        H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SOCH(CH.sub.3).sub.2                                                                        CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SOCH(CH.sub.3).sub.2                                                                        H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    Cl      OCH.sub.3                                                                            CH                                   H      SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SO.sub.2 CH(CH.sub.3).sub.2                                                                 CH.sub. 3                                                                          OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SO.sub.2 CH(CH.sub.3).sub.2                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      S-cyclopropyl H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      S-cyclopropyl H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      S-cyclopropyl H    Cl      OCH.sub.3                                                                            CH                                   H      S-cyclopropyl H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      S-cyclopropyl H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      S-cyclopropyl H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      S-cyclopropyl H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      S-cyclopropyl CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           S-cyclopropyl H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          S-cyclopropyl H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           S-cyclopropyl H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          S-cyclopropyl H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    S-cyclopropyl H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   S-cyclopropyl H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO-cyclopropyl                                                                              H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO-cyclopropyl                                                                              H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SO-cyclopropyl                                                                              H    Cl      OCH.sub.3                                                                            CH                                   H      SO-cyclopropyl                                                                              H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SO-cyclopropyl                                                                              H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SO-cyclopropyl                                                                              H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SO-cyclopropyl                                                                              H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SO-cyclopropyl                                                                              CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SO-cyclopropyl                                                                              H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO-cyclopropyl                                                                              H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO-cyclopropyl                                                                              H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SO-cyclopropyl                                                                              H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SO-cyclopropyl                                                                              H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SO-cyclopropyl                                                                              H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SO.sub.2 -cyclopropyl                                                                       H    Cl      OCH.sub.3                                                                            CH                                   H      SO.sub.2 -cyclopropyl                                                                       H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SO.sub.2 -cyclopropyl                                                                       CH.sub. 3                                                                          OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SO.sub.2 -cyclopropyl                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      OSO.sub.2 CH.sub.3                                                                          H    Cl      OCH.sub.3                                                                            CH                                   H      OSO.sub.2 CH.sub.3                                                                          H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      OSO.sub.2 CH.sub.3                                                                          CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   OSO.sub.2 CH.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      OSO.sub.2 CF.sub.3                                                                          H    Cl      OCH.sub.3                                                                            CH                                   H      OSO.sub.2 CF.sub.3                                                                          H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      OSO.sub.2 CF.sub.3                                                                          CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   OSO.sub.2 CF.sub.3                                                                          H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.3                                                                             OCH.sub. 3                                                                           CH                                   H      OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    Cl      OCH.sub.3                                                                            CH                                   H      OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      OSO.sub.2 CH.sub.2 CH.sub.3                                                                 CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   OSO.sub.2 CH.sub.2 CH.sub.3                                                                 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      N.sub.3       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      N.sub.3       H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      N.sub.3       H    Cl      OCH.sub.3                                                                            CH                                   H      N.sub.3       H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      N.sub.3       H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      N.sub.3       H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      N.sub.3       H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      N.sub.3       CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           N.sub.3       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          N.sub.3       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           N.sub.3       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          N.sub.3       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    N.sub.3       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   N.sub.3       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CN            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CN            H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      CN            H    Cl      OCH.sub.3                                                                            CH                                   H      CN            H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      CN            H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      CN            H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      CN            H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      CN            CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           CN            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          CN            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           CN            H    OCH.sub.3                                                                             OCH.sub. 3                                                                           CH                                   6-OCH.sub.3                                                                          CN            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    CN            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   CN            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CH.sub.2 F    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CH.sub.2 F    H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      CH.sub.2 F    H    Cl      OCH.sub.3                                                                            CH                                   H      CH.sub.2 F    H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      CH.sub.2 F    H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      CH.sub.2 F    H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      CH.sub.2 F    H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      CH.sub.2 F    CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           CH.sub.2 F    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          CH.sub.2 F    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           CH.sub.2 F    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          CH.sub.2 F    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    CH.sub.2 F    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   CH.sub.2 F    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CF.sub.2 H    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CF.sub.2 H    H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      CF.sub.2 H    H    Cl      OCH.sub. 3                                                                           CH                                   H      CF.sub.2 H    H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      CF.sub.2 H    H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    R      CF.sub.2 H    H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      CF.sub.2 H    H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      CF.sub.2 H    CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           CF.sub.2 H    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          CF.sub.2 H    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           CF.sub.2 H    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          CF.sub.2 H    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    CF.sub.2 H    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   CF.sub.2 H    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    Cl      OCH.sub.3                                                                            CH                                   H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.2 CH.sub. 3                                                                   NHCH.sub.3                                                                           N                                    H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SO.sub.2 N(OCH.sub.3)CH.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 NHCH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 NHCH.sub.3                                                                         H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SO.sub.2 NHCH.sub.3                                                                         H    Cl      OCH.sub.3                                                                            CH                                   H      SO.sub.2 NHCH.sub.3                                                                         H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SO.sub.2 NHCH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SO.sub.2 NHCH.sub.3                                                                         H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SO.sub.2 NHCH.sub.3                                                                         H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SO.sub.2 NHCH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO.sub.2 NHCH.sub. 3                                                                        H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2 NHCH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SO.sub.2 NHCH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SO.sub.2 NHCH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SO.sub.2 NHCH.sub.3                                                                         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    Cl      OCH.sub.3                                                                            CH                                   H      SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      SO.sub.2 NHCH.sub.2 CH.sub.3                                                                CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   SO.sub.2 NHCH.sub.2 CH.sub.3                                                                H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    Cl      OCH.sub.3                                                                            CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   CO.sub.2 CH.sub.2 CH.sub.2 OH                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    Cl      OCH.sub.3                                                                            CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.3                                                                             OCH.sub. 3                                                                           CH                                   6-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   CO.sub.2 CH.sub.2 CH.sub.2 CN                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    Cl      OCH.sub.3                                                                            CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                   H      CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                    H      CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                    H      CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                    H      CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                    5-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-F    CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   6-Cl   CO.sub.2 CH.sub.2 CH.sub.2 OSO.sub.2 CH.sub.3                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                   __________________________________________________________________________

                                      TABLE V                                     __________________________________________________________________________    General Formula 5                                                             R.sub.f                                                                              R.sub.6    R    X       Y      Z    m.p. (°C.)                  __________________________________________________________________________    H      SCH.sub.3  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      SCH.sub.3  H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      SCH.sub.3  H    Cl      OCH.sub.3                                                                            CH                                      H      SCH.sub.3  H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      SCH.sub.3  H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      SCH.sub.3  H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      SCH.sub.3  H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      SCH.sub.3  CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           SCH.sub.3  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub.3                                                                          SCH.sub.3  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           SCH.sub.3  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          SCH.sub.3  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-F    SCH.sub.3  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   SCH.sub.3  H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      SOCH.sub.3 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      SOCH.sub.3 H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      SOCH.sub.3 H    Cl      OCH.sub.3                                                                            CH                                      H      SOCH.sub.3 H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      SOCH.sub.3 H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      SOCH.sub.3 H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      SOCH.sub.3 H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      SOCH.sub.3 CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           SOCH.sub.3 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub.3                                                                          SOCH.sub.3 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           SOCH.sub.3 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          SOCH.sub.3 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-F    SOCH.sub.3 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   SOCH.sub.3 H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      SO-cyclopropyl                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      SO-cyclopropyl                                                                           H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      SO-cyclopropyl                                                                           H    Cl      OCH.sub.3                                                                            CH                                      H      SO-cyclopropyl                                                                           H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      SO-cyclopropyl                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      SO-cyclopropyl                                                                           H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      SO-cyclopropyl                                                                           H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      SO-cyclopropyl                                                                           CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           SO-cyclopropyl                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub.3                                                                          SO-cyclopropyl                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           SO-cyclopropyl                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          SO-cyclopropyl                                                                           H    OCH.sub.3                                                                             OCH.sub. 3                                                                           CH                                      6-F    SO-cyclopropyl                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   SO-cyclopropyl                                                                           H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      SO.sub.2 -cyclopropyl                                                                    H    Cl      OCH.sub.3                                                                            CH                                      H      SO.sub.2 -cyclopropyl                                                                    H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      SO.sub.2 -cyclopropyl                                                                    CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub.3                                                                          SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-F    SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   SO.sub.2 -cyclopropyl                                                                    H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      OSO.sub.2 CH.sub.3                                                                       H    Cl      OCH.sub.3                                                                            CH                                      H      OSO.sub.2 CH.sub. 3                                                                      H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      OSO.sub.2 CH.sub.3                                                                       CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub.3                                                                          OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-F    OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   OSO.sub.2 CH.sub.3                                                                       H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      CN         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      CN         H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      CN         H    Cl      OCH.sub.3                                                                            CH                                      H      CN         H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      CN         H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      CN         H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      CN         H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      CN         CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           CN         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub. 3                                                                         CN         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           CN         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          CN         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-F    CN         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   CN         H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      CH.sub.2 F H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      CH.sub.2 F H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      CH.sub.2 F H    Cl      OCH.sub.3                                                                            CH                                      H      CH.sub.2 F H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      CH.sub.2 F H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      CH.sub.2 F H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      CH.sub.2 F H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      CH.sub.2 F CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           CH.sub.2 F H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub.3                                                                          CH.sub.2 F H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           CH.sub.2 F H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          CH.sub.2 F H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-F    CH.sub.2 F H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   CH.sub.2 F H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    Cl      OCH.sub.3                                                                            CH                                      H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub.3                                                                          SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-F    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    Cl      OCH.sub.3                                                                            CH                                      H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-F    CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    Cl      OCH.sub.3                                                                            CH                                      H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-F    CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      H      CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.3                                                                             CH.sub.3                                                                             CH                                      H      CO.sub.2 CH.sub.2 CF.sub.3                                                               H    Cl      OCH.sub.3                                                                            CH                                      H      CO.sub.2 CH.sub.2 CF.sub.3                                                               H    CH.sub.3                                                                              CH.sub.3                                                                             CH                                      H      CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            N                                       H      CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.3                                                                             CH.sub.3                                                                             N                                       H      CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                           N                                       H      CO.sub.2 CH.sub.2 CF.sub.3                                                               CH.sub.3                                                                           OCH.sub.3                                                                             CH.sub.3                                                                             N                                       4-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      4-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-OCH.sub.3                                                                          CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-F    CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      6-Cl   CO.sub.2 CH.sub.2 CF.sub.3                                                               H    OCH.sub.3                                                                             OCH.sub.3                                                                            CH                                      __________________________________________________________________________

                                      TABLE VI                                    __________________________________________________________________________    General Formula 6                                                             R.sub.f                                                                             R.sub.6  R   X     Y     Z  m.p.(°C.)                            __________________________________________________________________________    H     SCH.sub.3                                                                              H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     SCH.sub.3                                                                              H   OCH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     SCH.sub.3                                                                              H   Cl    OCH.sub.3                                                                           CH                                             H     SCH.sub.3                                                                              H   CH.sub.3                                                                            CH.sub.3                                                                            CH                                             H     SCH.sub.3                                                                              H   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     SCH.sub.3                                                                              H   OCH.sub.3                                                                           CH.sub.3                                                                            N                                              H     SCH.sub.3                                                                              H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                          N                                              H     SCH.sub.3                                                                              CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                            N                                              4-CH.sub.3                                                                          SCH.sub.3                                                                              H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             4-Cl  SCH.sub.3                                                                              H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                          SCH.sub.3                                                                              H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-OCH.sub.3                                                                         SCH.sub.3                                                                              H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-F   SCH.sub.3                                                                              H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-Cl  SCH.sub.3                                                                              H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     SOCH.sub.3                                                                             H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     SOCH.sub.3                                                                             H   OCH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     SOCH.sub.3                                                                             H   Cl    OCH.sub.3                                                                           CH                                             H     SOCH.sub.3                                                                             H   CH.sub.3                                                                            CH.sub.3                                                                            CH                                             H     SOCH.sub.3                                                                             H   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     SOCH.sub.3                                                                             H   OCH.sub.3                                                                           CH.sub.3                                                                            N                                              H     SOCH.sub.3                                                                             H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                          N                                              H     SOCH     CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                            N                                              4-CH.sub.3                                                                          SOCH.sub.3                                                                             H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             4-Cl  SOCH.sub.3                                                                             H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                          SOCH.sub.3                                                                             H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-OCH.sub.3                                                                         SOCH.sub.3                                                                             H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-F   SOCH.sub.3                                                                             H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-Cl  SOCH.sub.3                                                                             H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     SO-cyclopropyl                                                                         H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     SO-cyclopropyl                                                                         H   OCH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     SO-cyclopropyl                                                                         H   Cl    OCH.sub.3                                                                           CH                                             H     SO-cyclopropyl                                                                         H   CH.sub.3                                                                            CH.sub.3                                                                            CH                                             H     SO-cyclopropyl                                                                         H   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     SO-cyclopropyl                                                                         H   OCH.sub.3                                                                           CH.sub.3                                                                            N                                              H     SO-cyclopropyl                                                                         H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                          N                                              H     SO-cyclopropyl                                                                         CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                            N                                              4-CH.sub.3                                                                          SO-cyclopropyl                                                                         H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             4-Cl  SO-cyclopropyl                                                                         H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                          SO-cyclopropyl                                                                         H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-OCH.sub.3                                                                         SO-cyclopropyl                                                                         H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-F   SO-cyclopropyl                                                                         H   OCH.sub. 3                                                                          OCH.sub.3                                                                           CH                                             6-Cl  SO-cyclopropyl                                                                         H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     SO.sub.2 -cyclopropyl                                                                  H   Cl    OCH.sub.3                                                                           CH                                             H     SO.sub.2 -cyclopropyl                                                                  H   CH.sub.3                                                                            CH.sub.3                                                                            CH                                             H     SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.3                                                                           CH.sub.3                                                                            N                                              H     SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                          N                                              H     SO.sub.2 -cyclopropyl                                                                  CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                            N                                              4-CH.sub.3                                                                          SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             4-Cl  SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                          SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-OCH.sub.3                                                                         SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-F   SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-Cl  SO.sub.2 -cyclopropyl                                                                  H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     OSO.sub.2 CH.sub.3                                                                     H   Cl    OCH.sub.3                                                                           CH                                             H     OSO.sub.2 CH.sub.3                                                                     H   CH.sub.3                                                                            CH.sub.3                                                                            CH                                             H     OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.3                                                                           CH.sub.3                                                                            N                                              H     OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                          N                                              H     OSO.sub.2 CH.sub.3                                                                     CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                            N                                              4-CH.sub.3                                                                          OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             4-Cl  OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                          OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-OCH.sub.3                                                                         OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-F   OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-Cl  OSO.sub.2 CH.sub.3                                                                     H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     CN       H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     CN       H   OCH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     CN       H   Cl    OCH.sub.3                                                                           CH                                             H     CN       H   CH.sub.3                                                                            CH.sub.3                                                                            CH                                             H     CN       H   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     CN       H   OCH.sub.3                                                                           CH.sub.3                                                                            N                                              H     CN       H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                          N                                              H     CN       CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                            N                                              4-CH.sub.3                                                                          CN       H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             4-Cl  CN       H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-CH.sub. 3                                                                         CN       H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-OCH.sub.3                                                                         CN       H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-F   CN       H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-Cl  CN       H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   Cl    OCH.sub.3                                                                           CH                                             H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   CH.sub.3                                                                            CH.sub.3                                                                            CH                                             H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                            N                                              H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                          N                                              H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                            N                                              4-CH.sub.3                                                                          SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             4-Cl  SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                          SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-OCH.sub.3                                                                         SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-F   SO.sub.2 N(OCH.sub.3)CH.sub. 3                                                         H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-Cl  SO.sub.2 N(OCH.sub.3)CH.sub.3                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   Cl    OCH.sub.3                                                                           CH                                             H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   CH.sub.3                                                                            CH.sub.3                                                                            CH                                             H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                            N                                              H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                          N                                              H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                            N                                              4-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             4-Cl  CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-F   CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-Cl  CO.sub.2 CH.sub.2 CH.sub.2 OH                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   Cl    OCH.sub.3                                                                           CH                                             H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   CH.sub.3                                                                            CH.sub.3                                                                            CH                                             H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                            N                                              H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                          N                                              H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                            N                                              4-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             4-Cl  CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                          CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-F   CO.sub.2 CH.sub.2 CH.sub. 2 CN                                                         H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             6-Cl  CO.sub.2 CH.sub.2 CH.sub.2 CN                                                          H   OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                             __________________________________________________________________________

                                      TABLE VII                                   __________________________________________________________________________    General Formula 7                                                             R.sub.1                                                                             R.sub.7    A  X      Y      m.p.(°C.)                            __________________________________________________________________________    H     SOCH.sub.3 A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.3 A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.3 A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.3 A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 CH.sub.3                                                                        A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 CH.sub.3                                                                        A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.3                                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.2 CH.sub.3                                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.2 CH.sub.3                                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.3                                                                      A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 CH.sub.2 CH.sub.3                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 CH.sub.2 CH.sub.3                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub. 3                                                     A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SOCH(CH.sub.3).sub.2                                                                     A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH(CH.sub.3).sub.2                                                                     A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH(CH.sub.3).sub.2                                                                     A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH(CH.sub.3).sub.2                                                                     A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 CH(CH.sub.3).sub.2                                                              A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 CH(CH.sub.3).sub.2                                                              A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 CH(CH.sub.3).sub.2                                                              A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 CH(CH.sub.3).sub.2                                                              A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                    A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                    A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                    A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.2 CH.sub.2 CH.sub. 3                                                   A-4                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                             A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                             A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                             A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                             A-4                                                                              X.sub.3 = OCH.sub.3                                       H     S-cyclopropyl                                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     S-cyclopropyl                                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     S-cyclopropyl                                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     S-cyclopropyl                                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 -cyclopropyl                                                                    A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 -cyclopropyl                                                                    A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 -cyclopropyl                                                                    A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 -cyclopropyl                                                                    A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.3                                                                       A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CH.sub.3                                                                       A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CH.sub.3                                                                       A-3                                                                              X.sub.1 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.3                                                                       A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.3                                                                       A-7                                                                              X.sub.4 = OCH.sub.3                                                                  Y.sub.4 = OCH.sub.3                                H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-3                                                                              X.sub.1 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CF.sub.3                                                                       A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CF.sub.3                                                                       A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CF.sub.3                                                                       A-3                                                                              X.sub.1 = OCH.sub.3                                       H     OSO.sub.2 CF.sub.3                                                                       A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CCl.sub.3                                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CCl.sub.3                                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CCl.sub.3                                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     OSO.sub.2 CCl.sub.3                                                                      A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CN         A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CN         A-3                                                                              X.sub.1 = CH.sub.3                                        H     CN         A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CN         A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CH.sub.2 F A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CH.sub.2 F A-3                                                                              X.sub.1 = CH.sub.3                                        H     CH.sub.2 F A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CH.sub.2 F A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CF.sub.2 H A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CF.sub.2 H A-3                                                                              X.sub.1 = CH.sub.3                                        H     CF.sub.2 H A-3                                                                              X.sub.1 =  OCH.sub.3                                      H     CF.sub.2 H A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.3                                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 NHCH.sub.3                                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 NHCH.sub.3                                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.3                                                                      A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                   A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                   A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 NECH.sub.2 CH.sub.2 OCH.sub.3                                                   A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.2 CH.sub.2 OCH.sub.3                                                   A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-3                                                                              X.sub.1  = OCH.sub.3                                      H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CF.sub.2                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CF.sub.2                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CF.sub.2                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-OCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-OCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        6-OCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-Y                                                                              X.sub.1 = OCH.sub.3                                       6-OCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       6-SCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-SCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        6-SCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-SCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       6-N(CH.sub.3).sub.2                                                                 SO.sub.2 N(CH.sub.3).sub.2                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-N(CH.sub.3).sub.2                                                                 SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        6-N(CH.sub.3).sub.2                                                                 SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-N(CH.sub.3).sub.2                                                                 SO.sub.2 N(CH.sub.3).sub.2                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       6-NHCH.sub.3                                                                        SO.sub.2 N(CH.sub.3).sub.2                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-NHCH.sub.3                                                                        SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 =  CH.sub.3                                       6-NHCH.sub.3                                                                        SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-NHCH.sub.3                                                                        SO.sub.2 N(CH.sub.3).sub.2                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       6-OCH.sub.3                                                                         CO.sub.2 CH.sub.3                                                                        A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-OCH.sub.3                                                                         CO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = CH.sub.3                                        6-OCH.sub.3                                                                         CO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = OCH.sub.3                                       6-OCH.sub.3                                                                         CO.sub.2 CH.sub.3                                                                        A-4                                                                              X.sub.3 = OCH.sub.3                                       6-SCH.sub.3                                                                         CO.sub.2 CH.sub.3                                                                        A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-SCH.sub.3                                                                         CO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = CH.sub.3                                        6-SCH.sub.3                                                                         CO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = OCH.sub.3                                       6-SCH.sub.3                                                                         CO.sub.2 CH.sub.3                                                                        A-4                                                                              X.sub.3 = OCH.sub.3                                       6-N(CH.sub.3).sub.2                                                                 CO.sub.2 CH.sub.3                                                                        A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-N(CH.sub.3).sub.2                                                                 CO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = CH.sub.3                                        6-N(CH.sub.3).sub.2                                                                 CO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.3 = OCH.sub.3                                       6-N(CH.sub.3).sub.2                                                                 CO.sub.2 CH.sub.3                                                                        A-4                                                                              X.sub.3 = OCH.sub.3                                       6-NHCH.sub.3                                                                        SO.sub.2 N(CH.sub.3).sub.2                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-NHCH.sub.3                                                                        SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        6-NHCH.sub.3                                                                        SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-NHCH.sub.3                                                                        SO.sub.2 N(CH.sub.3).sub.2                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       6-OCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-OCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        6-OCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-OCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       6-SCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-SCH.sub.3                                                                         SO.sub. 2 N(CH.sub.3).sub.2                                                              A-3                                                                              X.sub.1 = CH.sub.3                                        6-SCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-SCH.sub.3                                                                         SO.sub.2 N(CH.sub.3).sub.2                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       6-N(CH.sub.3).sub.2                                                                 SO.sub.2 N(CH.sub.3).sub.2                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-N(CH.sub.3).sub.2                                                                 SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        6-N(CH.sub.3).sub.2                                                                 SO.sub.2 N(CH.sub.3).sub.2                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-N(CH.sub.3).sub.2                                                                 SO.sub.2 N(CH.sub.3).sub.2                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       6-NHCH.sub.3                                                                        CO.sub.2 CH.sub.3                                                                        A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-NHCH.sub.3                                                                        CO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = CH.sub.3                                        6-NHCH.sub.3                                                                        CO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = OCH.sub.3                                       6-NHCH.sub.3                                                                        CO.sub.2 CH.sub.3                                                                        A-4                                                                              X.sub.3 = OCH.sub.3                                       6-OCH.sub.3                                                                         SO.sub.2 NHOCH.sub.3                                                                     A-2                                                                              X.sub.1 = CH.sub. 3                                                                  Y.sub.1 = CH                                       6-OCH.sub.3                                                                         SO.sub.2 NHOCH.sub.3                                                                     A-3                                                                              X.sub.1 = CH.sub.3                                        6-OCH.sub.3                                                                         SO.sub.2 NHOCH.sub.3                                                                     A-3                                                                              X.sub.1 = OCH.sub.3                                       6-OCH.sub.3                                                                         SO.sub.2 NHOCH.sub.3                                                                     A-4                                                                              X.sub.3 = OCH.sub.3                                       6-SCH.sub.3                                                                         SO.sub.2 NHOCH.sub.3                                                                     A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-SCH.sub.3                                                                         SO.sub.2 NHOCH.sub.3                                                                     A-3                                                                              X.sub.1 = CH.sub.3                                        6-SCH.sub.3                                                                         SO.sub.2 NHOCH.sub.3                                                                     A-3                                                                              X.sub.1 = OCH.sub.3                                       6-SCH.sub.3                                                                         SO.sub.2 NHOCH.sub.3                                                                     A-4                                                                              X.sub.3 = OCH.sub.3                                       6-N(CH.sub.3).sub.2                                                                 SO.sub.2 NHOCH.sub.3                                                                     A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-N(CH.sub.3).sub.2                                                                 SO.sub.2 NHOCH.sub.3                                                                     A-3                                                                              X.sub.1 = CH.sub.3                                        6-N(CH.sub.3).sub.2                                                                 SO.sub.2 NHOCH.sub.3                                                                     A-3                                                                              X.sub.1 = OCH.sub.3                                       6-N(CH.sub.3).sub.2                                                                 SO.sub.2 NHOCH.sub.3                                                                     A-4                                                                              X.sub.3 = OCH.sub.3                                       6-NHCH.sub.3                                                                        SO.sub.2 NHOCH.sub.3                                                                     A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1  = CH.sub.2                                6-NHCH.sub.3                                                                        SO.sub.2 NHOCH.sub.3                                                                     A-3                                                                              X.sub.1 = CH.sub.3                                        6-NHCH.sub.3                                                                        SO.sub.2 NHOCH.sub.3                                                                     A-3                                                                              X.sub.1 = OCH.sub.3                                       6-NHCH.sub.3                                                                        SO.sub.2 NHOCH.sub.3                                                                     A-4                                                                              X.sub.3 = OCH.sub.3                                       6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-4                                                                              X.sub.4 = OCH.sub.3                                       6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-2                                                                              X.sub.1  = CH.sub.3                                                                  Y.sub.1 = CH.sub.2                                 6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       6-OCH.sub.3                                                                         CO.sub.2 CH.sub.2 CH.sub.3                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       __________________________________________________________________________

                                      TABLE VIII                                  __________________________________________________________________________    General Formula 8                                                             R.sub.1                                                                             R.sub.3    A  X      X      m.p.(°C.)                            __________________________________________________________________________    H     SOCH.sub.3 A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.3 A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.3 A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.3 A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.3                                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.2 CH.sub.3                                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.2 CH.sub.3                                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.3                                                                      A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-4                                                                              X.sub.3 = OCH.sub.3                                       H     S-cyclopropyl                                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     S-cyclopropyl                                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     S-cyclopropyl                                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     S-cyclopropyl                                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 -cyclopropyl                                                                    A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 -cyclopropyl                                                                    A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 -cyclopropyl                                                                    A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 -cyclopropyl                                                                    A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.3                                                                       A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CH.sub.3                                                                       A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CH.sub.3                                                                       A-3                                                                              X.sub.1 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.3                                                                       A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-3                                                                              X.sub. 1 = CH.sub.3                                       H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-3                                                                              X.sub.1 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CF.sub.3                                                                       A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CF.sub.3                                                                       A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CF.sub.3                                                                       A-3                                                                              X.sub.1 = OCH.sub.3                                       H     OSO.sub.2 CF.sub.3                                                                       A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OCO.sub.2 CCl.sub.3                                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CCl.sub.3                                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CCl.sub.3                                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     OSO.sub.2 CCl.sub.3                                                                      A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CH.sub.2 F A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CH.sub.2 F A-3                                                                              X.sub.1 = CH.sub.3                                        H     CH.sub.2 F A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CH.sub.2 F A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.3                                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 NHCH.sub.3                                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 NHCH.sub.3                                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.3                                                                      A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CN.sub.2 CN                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub. 2 CN                                                           A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       __________________________________________________________________________

                                      TABLE IX                                    __________________________________________________________________________    General Pormula 9                                                             R.sub.f                                                                             R.sub.4    A  X      Y      m.p.(°C.)                            __________________________________________________________________________    H     SOCH.sub.3 A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.3 A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.3 A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.3 A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SOCH.sub.2 CN.sub.3                                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.2 CH.sub.3                                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.2 CH.sub.3                                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.3                                                                      A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-4                                                                              X.sub.3 = OCH.sub.3                                       H     S-cyclopropyl                                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     S-cyclopropyl                                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     S-cyclopropyl                                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     S-cyclopropyl                                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO-cyclopropyl                                                                           A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO-cyclopropyl                                                                           A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO-cyclopropyl                                                                           A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO-cyclopropyl                                                                           A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 -cyclopropyl                                                                    A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 -cyclopropyl                                                                    A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 -cyclopropyl                                                                    A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 -cyclopropyl                                                                    A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.3                                                                       A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CH.sub.3                                                                       A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CH.sub.3                                                                       A-3                                                                              X.sub.1 =  OCH.sub.3                                      H     OSO.sub.2 CH.sub.3                                                                       A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-3                                                                              X.sub.1 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.2 CH.sub.3                                                              A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CF.sub.3                                                                       A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CF.sub.3                                                                       A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CF.sub.3                                                                       A-3                                                                              X.sub.1 = OCH.sub.3                                       H     OSO.sub.2 CF.sub.3                                                                       A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CH.sub.2 F A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CH.sub.2 F A-3                                                                              X.sub.1 = CH.sub.3                                        H     CH.sub.2 F A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CH.sub.2 F A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CN         A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CN         A-3                                                                              X.sub.1 = CH.sub.3                                        H     CN         A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CN         A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.3                                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 NHCH.sub.3                                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 NHCH.sub.3                                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.3                                                                      A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CN.sub.2 OH                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       __________________________________________________________________________

                                      TABLE X                                     __________________________________________________________________________    General Formula 10                                                            R.sub.f                                                                             R.sub.5    A  X      Y      m.p.(°C.)                            __________________________________________________________________________    H     SOCH.sub.3 A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.3 A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.3 A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.3 A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.3                                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.2 CH.sub.3                                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.2 CH.sub.3                                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.3                                                                      A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-3                                                                              X.sub.1 = CH.sub.3                                        H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SOCH.sub.2 CH.sub.2 CH.sub.3                                                             A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 CH.sub.3                                                                        A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 CH.sub.3                                                                        A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 CH.sub.3                                                                        A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 CH.sub.2 CH.sub.3                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 CH.sub.2 CH.sub.3                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 CH.sub.2 CH.sub.3                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 CH.sub.2 CH.sub.2 CH.sub. 3                                                     A-4                                                                              X.sub.3 = OCH.sub.3                                       H     S-cyclopropyl                                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     S-cyclopropyl                                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     S-cyclopropyl                                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     S-cyclopropyl                                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO-cyclopropyl                                                                           A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO-cyclopropyl                                                                           A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO-cyclopropyl                                                                           A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO-cyclopropyl                                                                           A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 -cyclopropyl                                                                    A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 -cyclopropyl                                                                    A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 -cyclopropyl                                                                    A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 -cyclopropyl                                                                    A-4                                                                              X.sub.3 = OCH.sub.3                                       H     OSO.sub.2 CH.sub.3                                                                       A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     OSO.sub.2 CH.sub.3                                                                       A-3                                                                              X.sub.1 = CH.sub.3                                        H     OSO.sub.2 CH.sub.3                                                                       A-3                                                                              X.sub.1  = OCH.sub.3                                      H     OSO.sub.2 CH.sub.3                                                                       A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CH.sub.2 F A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CH.sub.2 F A-3                                                                              X.sub.1 = CH.sub.3                                        H     CH.sub.2 F A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CH.sub.2 F A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CN         A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CN         A-3                                                                              X.sub.1 = CH.sub.3                                        H     CN         A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CN         A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.3                                                                      A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub. 1 = CH.sub.2                                H     SO.sub.2 NHCH.sub.3                                                                      A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 NHCH.sub.3                                                                      A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.3                                                                      A-4                                                                              X.sub.3 = OCH.sub.3                                       H     SO.sub.2 NBCH.sub.2 CH.sub.3                                                             A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     SO.sub.2 NHCH.sub.2 CH.sub.3                                                             A-3                                                                              X.sub.1 = CH.sub.3                                        H     SO.sub.2 NHCH.sub.2 CH.sub.3                                                             A-3                                                                              X.sub.1 = OCH.sub.3                                       H     SO.sub.2 NHCH.sub.2 CH.sub.3                                                             A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 OH                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub. 1 = CH.sub.2                                H     CO.sub.2 CH.sub.2 CH.sub.2 CH                                                            A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CH.sub.2 CN                                                            A-4                                                                              X.sub.3 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-2                                                                              X.sub.1 = CH.sub.3                                                                   Y.sub.1 = CH.sub.2                                 H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-3                                                                              X.sub.1 = CH.sub.3                                        H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-3                                                                              X.sub.1 = OCH.sub.3                                       H     CO.sub.2 CH.sub.2 CF.sub.3                                                               A-4                                                                              X.sub.3 = OCH.sub.3                                       __________________________________________________________________________

Formulations

Useful formulations of the compounds of Formula I can be prepared inconventional ways. They include dusts, granules, pellets, solutions,suspensions, emulsions, wettable powders, emulsifiable concentrates andthe like. Many of these may be applied directly. Sprayable formulationscan be extended in suitable media and used at spray volumes of from afew liters to several hundred liters per hectare. High strengthcompositions are primarily used as intermediates for furtherformulation. The formulations, broadly, contain about 0.1% to 99% byweight of active ingredient(s) and at least one of (a) about 0.1% to 20%surfactant(s) and (b) about 1% to 99.9% solid or liquid inertdiluent(s). More specifically, they will contain these ingredients inthe following approximate proportions:

    ______________________________________                                                    Weight Percent*                                                               Active                                                                        Ingredient                                                                            Diluent(s)                                                                              Surfactant(s)                                   ______________________________________                                        Wettable Powders                                                                            20-90      0-74     1-10                                        Oil Suspensions,                                                                             3-50     40-95     0-15                                        Emulsions, Solutions,                                                         (including Emulsifiable                                                       Concentrates)                                                                 Aqueous Suspension                                                                          10-50     40-84     1-20                                        Dusts          1-25     70-99     0-5                                         Granules and Pellets                                                                        0.1-95      5-99.9  0-15                                        High Strength 90-99      0-10     0-2                                         Compositions                                                                  ______________________________________                                         *Active ingredient plus at least one of a Surfactant or a Diluent equals      100 weight percent.                                                      

Lower or higher levels of active ingredient can, of course, be presentdepending on the intended use and the physical properties of thecompound. Higher ratios of surfactant to active ingredient are sometimesdesirable, and are achieved by incorporation into the formulation or bytank mixing.

Typical solid diluents are described in Watkins, et al., "Handbook ofInsecticide Dust Diluents and Carriers", 2nd Ed Dotland Books, Caldwell,N.J., but other solids, either mined or manufactured, may be used. Themore absorptive diluents are preferred for wettable powders and thedenser ones for dusts. Typical liquid diluents and solvents aredescribed in Marsden, "Solvents Guide," 2nd Ed., Interscience, N.Y.,1950. Solubility under 0.1% is preferred for suspension concentrates;solution concentrates are preferably stable against phase separation at0° C. "McCutcheon's Detergents and Emulsifiers Annual", MC PublishingCorp., Ridgewood, N.J., as well as Sisely and Wood, "Encyclopedia ofSurface Active Agents", Chemical Publishing Co., Inc., New York, 1964,list surfactants and recommended uses. All formulations can containminor amounts of additives to reduce foaming, caking, corrosion,microbiological growth, etc.

The methods of making such compositions are well known. Solutions areprepared by simply mixing the ingredients. Fine solid compositions aremade by blending and, usually, grinding as in a hammer or fluid energymill. Suspensions are prepared by wet milling (see, for example,Littler, U.S. Pat. No. 3,060,084). Granules and pellets may be made byspraying the active material upon preformed granular carriers or byagglomeration techniques. See J. E. Browning, "Agglomeration", ChemicalEngineering, Dec. 4, 1967, pp. 147ff. and "Perry's Chemical Engineer'sHandbook", 5th Ed., McGraw-Hill, New York, 1963, pp. 8-57ff.

For further information regarding the art of formulation, see forexample:

H. M. Loux, U.S. Pat. No. 3,235,361, Feb. 15, 1966, Col. 6, line 16through Col. 7, line 19 and Examples 10 through 41;

R. W. Luckenbaugh, U.S. Pat. No. 3,309,192, Mar. 14, 1967, Col. 5, line43 through Col. 7, line 62 and Examples 8, 12, 15, 39, 41, 52, 53, 58,132, 138-140, 162-164, 166, 167 and 169-182;

H. Gysin and E. Knusli, U.S. Pat. No. 2,891,855, Jun. 23, 1959, Col. 3,line 66 through Col. 5, line 17 and Examples 1-4;

G. C. Klingman, "Weed Control as a Science", John Wiley and Sons, Inc.,New York, 1961, pp. 81-96; and

J. D. Fryer and S. A. Evans, "Weed Control Handbook", 5th Ed., BlackwellScientific Publications, Oxford, 1968, pp. 101-103.

In the following examples, all parts are by weight unless otherwiseindicated.

EXAMPLE 24 High Strength Concentrate

    ______________________________________                                        N2-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-                                                          99%                                               N3-methyl-2,3-pyridinedisulfonamide                                           trimethylnonyl polyethylene glycol ether                                                                   1%                                               ______________________________________                                    

The surfactant is sprayed upon the active ingredient in a blender andthe mixture sifted through a U. S. S. no. 40 sieve (0.42 mm openings)prior to packaging. The concentrate may be formulated further forpractical use.

EXAMPLE 25 Wettable Powder

    ______________________________________                                        2-[[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-                                                        65%                                                 aminosulfonyl]-3-pyridinecarboxylic acid,                                     methyl ester                                                                  dodecylphenol polyethylene glycol ether                                                                 2%                                                  sodium ligninsulfonate    4%                                                  sodium silicoaluminate    6%                                                  montmorillonite (calcined)                                                                              23%                                                 ______________________________________                                    

The ingredients are thoroughly blended. The liquid surfactant is addedby spraying upon the solid ingredients in the blender. After grinding ina hammer mill to produce particles essentially all below 100 microns,the material is reblended and sifted through a U.S.S. No. 50 sieve (0.3mm opening) and packaged.

EXAMPLE 26 Aqueous Suspension

    ______________________________________                                        N2-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-                                                        40.0%                                               N3-methyl-2,3-pyridinedisulfonamide                                           polyacrylic acid thickener                                                                              0.3%                                                dodecylphenol polyethylene glycol ether                                                                 0.5%                                                disodium phosphate        1%                                                  monosodium phosphate      0.5%                                                polyvinyl alcohol         1.0%                                                water                     56.7%                                               ______________________________________                                    

The ingredients are blended and ground together in a sand mill toproduce particles essentially all under 5 microns in size.

EXAMPLE 27 Oil Suspension

    ______________________________________                                        N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-3-(1-                                                     35%                                                propylsulfonyl)-2-pyridinesulfonamide                                         methyl ester                                                                  blend of polyalcohol carboxylic esters                                                                    6%                                                and oil soluble petroleum sulfonates                                          xylene                     59%                                                ______________________________________                                    

The ingredients are combined and ground together in a sand mill toproduce particles essentially all below 3 microns. The product can beused directly, extended with oils, or emulsified in water.

EXAMPLE 28 Oil Suspension

    ______________________________________                                        N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-                                                          25%                                                3-(1-methylsulfonyloxy)-2-pyridinesulfonamide                                 methyl ester                                                                  polyoxyethylene sorbitol hexaoleate                                                                       5%                                                highly aliphatic hydrocarbon oil                                                                         70%                                                ______________________________________                                    

The ingredients are ground together in a sand mill until the solidparticles have been reduced to under about 5 microns. The resultingthick suspension may be applied directly, but preferably after beingextended with oils or emulsified in water.

EXAMPLE 29 Aqueous Suspension

    ______________________________________                                        N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-                                                          25%                                                3-(1-ethylsulfonyl)-2-pyridinesulfonamide                                     methyl ester                                                                  hydrated attapulgite        3%                                                crude calcium ligninsulfonate                                                                            10%                                                sodium dihydrogen phosphate                                                                               0.5%                                              water                      61.5%                                              ______________________________________                                    

The ingredients are ground together in a ball or roller mill until thesolid particles have been reduced to diameters under 10 microns.

EXAMPLE 29 Wettable Powder

    ______________________________________                                        N2-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-                                                        40.0%                                               N3-methyl-2,3-pyridinedisulfonamide                                           dioctyl sodium sulfosuccinate                                                                           1.5%                                                sodium ligninsulfonate     3%                                                 low viscosity methyl cellulose                                                                          1.5%                                                attapulgite               54%                                                 ______________________________________                                    

The ingredients are thoroughly blended, passed through an air mill, toproduce an average particle size under 15 microns, reblended, and siftedthrough a U.S.S. No. 50 sieve (0.3 mm opening) before packaging.

All compounds of the invention may be formulated in the same manner.

EXAMPLE 30 Granule

    ______________________________________                                        wettable powder of Example 29                                                                       15%                                                     gypsum                69%                                                     potassium sulfate     16%                                                     ______________________________________                                    

The ingredients are blended in a rotating mixer and water sprayed on toaccomplish granulation. When most of the material has reached thedesired range of 1.0 to 0.42 cm (U.S.S.#18 to 40 sieves), the granulesare removed, dried, and screened. Oversized material is crushed toproduce additional material in the desired range. These granules contain% active ingredient.

EXAMPLE 31 Wettable Powder

    ______________________________________                                        N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl-                                                           50%                                                3-(ethylsulfonyl)-2-pyridinesulfonamide                                       methyl ester                                                                  sodium alkylnaphthalenesulfonate                                                                          2%                                                low viscosity methyl cellulose                                                                            2%                                                diatomaceous earth         46%                                                ______________________________________                                    

The ingredients are blended, coarsely hammermilled and the air milled toproduce particles of active essentially all below 10 microns indiameter. The product is reblended before packaging.

EXAMPLE 32 Extruded Pellet

    ______________________________________                                        N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl-                                                           25%                                                3-(ethylsulfonyl)-2-pyridinesulfonamide                                       anhydrous sodium sulfate   10%                                                crude calcium ligninsulfonate                                                                             5%                                                sodium alkylnaphthalenesulfonate                                                                          1%                                                calcium/magnesium bentonite                                                                              59%                                                ______________________________________                                    

The ingredients are blended, hammer-milled and then moistened with about12% water. The mixture is extruded as cylinders about 3 mm diameterwhich are cut to produce pellets about 3 mm long. These may be useddirectly after drying, or the dried pellets may be crushed to pass aU.S.S. No. 20 sieve (0.84 mm openings). The granules held on a U.S.S.No. 40 sieve (0.42 mm openings) may be packaged for use and the finesrecycled.

EXAMPLE 33 Wettable Powder

    ______________________________________                                        N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-                                                          80%                                                3-(1-ethylsulfonyl)-2-pyridinesulfonamide                                     sodium alkylnaphthalenesulfonate                                                                         2%                                                 sodium ligninsulfonate     2%                                                 synthetic amorphous silica 3%                                                 kaolinite                  13%                                                ______________________________________                                    

The ingredients are blended and then ground in a hammermill to produceparticles with an average particle size less than 25 microns indiameter. The material is reblended and sifted through a U.S.S. No. 50sieve (0.3 mm opening) before being packaged.

EXAMPLE 34 High Strength Concentrate

    ______________________________________                                        N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-                                                          98.5%                                              3-(1-ethylsulfonyl)-2-pyridinesulfonamide                                     silica aerogel             0.5%                                               synthetic amorphous fine silica                                                                          1.0%                                               ______________________________________                                    

The ingredients are blended and ground in a hammer mill to produce ahigh strength concentrate essentially all passing a U.S.S. No. 50 sieve(0.3 mm openings). This material may then be formulated in a variety ofways.

EXAMPLE 35 Wettable Powder

    ______________________________________                                        2-[[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-                                                        80%                                                 aminosulfonyl]-3-pyridinecarboxylic acid,                                     methyl ester                                                                  sodium alkylnaphthalenesulfonate                                                                        2%                                                  sodium ligninsulfonate    2%                                                  synthetic amorphous silica                                                                              3%                                                  kaolinite                 13%                                                 ______________________________________                                    

The ingredients are blended and then ground in a hammermill to produceparticles with an average particle size less than 25 microns indiameter. The material is reblended and sifted through a U.S.S. No. 50sieve (0.3 mm opening) before being packaged.

EXAMPLE 36 High Strength Concentrate

    ______________________________________                                        N2-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-                                                        98.5%                                               N3-methyl-2,3-pyridinedisulfonamide                                           silica aerogel            0.5%                                                synthetic amorphous fine silica                                                                         1.0%                                                ______________________________________                                    

The ingredients are blended and ground in a hammer mill to produce ahigh strength concentrate essentially all passing a U.S.S. No. 50 sieve(0.3 mm openings). This material may then be formulated in a variety ofways.

Utility

Test results indicate that the compounds of the present invention arehighly active preemergent and/or postemergent herbicides or plant growthregulants. Many of them have utility for broad-spectrum pre- and/orpostemergence weed control in areas where complete control of allvegetation is desired, such as around fuel storage tanks, industrialstorage areas, parking lots, drive-in theaters, around billboards,highway and railroad structures. Some of the compounds have utility forselective weed control in plantation crops, Solanaceae family crops suchas tomatoes, potatoes and peppers, other crops such as wheat, barley,corn, cotton or soybeans, and their fallow land. In particular, somecompounds of this invention control weeds in corn (maize) both pre- andpostemergence without significant crop damage. Some compounds of thisinvention also control weeds in potato (Solanum tuberosum) and tomato(Lycopersicon esculentum) without significant crop damage. Thesecompounds are particularly useful to control such problem weeds asfoxtail (Setaria spp.), fall panicum (Panicum dichotomiflorum),barnyardgrass (Echinochloa crusgalli), seedling johnsongrass (Sorghumhalepense) and shattercane (Sorghum bicolor). They can be usedpreemergence or postemergence and are most effective when appliedpostemergence to young weeds. They are also effective on certainbroadleaf weeds such as lambsquarters (Chenopodium album), pigweed(Amaranthus spp.) and velvetleaf (Abutlion theophrasti).

Alternatively, the subject compounds are useful to modify plant growthand as citrus abscission agents.

Rates of application for compounds of this invention are determined by anumber of factors, including their use as plant growth modifiers or asherbicides, crop species involved, types of weeds to be controlled,weather and climate, formulations selected, mode of application, amountof foliage present, etc. In general terms, the subject compounds shouldbe applied at levels of around 0.001 to 20 kg/ha, the lower rates beingsuggested for use on lighter soils and/or those having a low organicmatter content, for plant growth modification or for situations whereonly short-term persistence is required.

Compounds of this invention may be used in combination with any othercommercial herbicide, examples of which are those of the triazine,triazole, imidazolinone, uracil, urea, amide, diphenylether, cineole,carbamate and bipyridylium types. They are particularly useful incombination with the following herbicides.

    ______________________________________                                                  Chemical Name                                                       ______________________________________                                        Common Name                                                                   alachlor    2-chloro-2',6'-diethyl-N-(methoxymethyl)                          acetanilide                                                                   atrazine    2-chloro-4-(ethylamino)-6-(isopropyl-                                         amino)- .sub.-  s-triazine                                        butylate    s-ethyl-diisobutylthiocarbamate                                   cyanazine   2-[[4-chloro-6-(ethylamino)- .sub.-  s-triazin-2-                             yl]amino]-2-methylpropionitrile                                   dicamba     3,6-dichloro- -o-anisic acid                                      EPTC        S-ethyl dipropylthiocarbamate                                     linuron     3-(3,4-dichlorophenyl)-1-methoxy-1-                                           methylurea                                                        metolachlor 2-chloro-N-(2-ethyl-6-methylphenyl)-N-                                        (2-methoxy-1-methylethyl)acetamide                                metribuzin  4-amino-6-tert-butyl-3-(methylthio)-as-                                       triazine-5(4H)-one                                                tridiphane  2-(3,5-dichlorophenyl)-2-(2,2,2-tri-                                          chloroethyl)oxirane                                               2,4-D       (2,4-dichlorophenoxy)acetic acid                                  bromoxynil  3,5-dibromo-4-hydroxyphenylcyanide                                paraquat    1,1'-dimethyl-4,4-bipyridinium ion                                glyphosate  N-(phosphonomethyl)glycine                                        DCPA        dimethyl tetrachloroterephthalate                                 dalapon     2,2-dichloropropionic acid                                        dinoseb     2-(1-methylpropyl)-4,6-dinitrophenol                              diphenamid  N,N-dimethyl-2,2-diphenylacetamide                                pendimethalin                                                                             N-(1-ethylpropyl)-3,4-dimethyl-2,6-                                           dinitrobenamine                                                   oryzalin    3,5-dinitro-N,N-dipropylsulfanilamide                             trifluralin α,α,α-trifluoro-2,6-dinitro-N,N-                            dipropyl-p-toluidine                                              chloramben  3-amino-2,5-dichlorobenzoic acid                                  napropamide 2-(α-naphthoxy)-N,N-diethylpropion-                                     amide                                                             pebulate    S-propyl butylethylthiocarbamate                                  chlorpropham                                                                              isopropyl m-chlorocarbanilate                                     bensulide   S-(O,O-diisopropyl phosphorodithioate)                                        ester of N-(2-mercaptoethyl)benzene-                                          sulfonamide                                                       Trade Name                                                                    Harmony ®                                                                             3-[[(4-methoxy-6-methyl-1,3,5-triazin-                                        2-yl)aminocarbonyl]aminosulfonyl]-2-                                          thiophenecarboxylic acid, methyl ester                            Cinch ® 1-methyl-4-(1-methylethyl)-2-exo-[(2-                                         methylphenyl)-methoxy]-7-oxabicyclo-                                          [2.2.1]heptane                                                    --          2-ethoxy-N-[[4-(2,2,2-trifluoroethoxy)-                                       6-methoxy-1,3,5-triazin-2-yl]amino-                                           carbonyl]benzenesulfonamide                                       ______________________________________                                    

Herbicidal properties of the subject compounds were discovered in aseries of greenhouse tests. Test procedures and results follow.

    __________________________________________________________________________    Compounds                                                                      ##STR55##                                                                    Compound                                                                            R.sub.2    R   R.sub.1                                                                           X     Y    Z                                         __________________________________________________________________________     1    SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                         2    SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   H   CH.sub.3                                                                            OCH.sub.3                                                                          CH                                         3    SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   H   Cl    OCH.sub.3                                                                          CH                                         4    SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                         5    SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                          6    SO.sub.2 CH.sub.2 CH.sub.2 CH.sub.3                                                      H   H   CH.sub.3                                                                            OCH.sub.3                                                                          N                                          7    SO.sub. 2 CH.sub.2 CH.sub.2 CH.sub.3                                                     H   H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                          8    S(O)CH.sub.2 CH.sub.2 CH.sub.3                                                           H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                         9    S(O)CH.sub.2 CH.sub.2 CH.sub.3                                                           H   H   CH.sub.3                                                                            OCH.sub.3                                                                          CH                                        10    S(O)CH.sub.2 CH.sub.2 CH.sub.3                                                           H   H   Cl    OCH.sub.3                                                                          CH                                        11    S(O)CH.sub.2 CH.sub.2 CH.sub.3                                                           H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        12    S(O)CH.sub.2 CH.sub.2 CH.sub.3                                                           H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         13    S(O)CH.sub.2 CH.sub.2 CH.sub.3                                                           H   H   CH.sub.3                                                                            OCH.sub.3                                                                          N                                         14    S(O)CH.sub.2 CH.sub.2 CH.sub.3                                                           H   H   OCH.sub.2 CH.sub.3                                                                  NHCH.sub.3                                                                         N                                         15    S(O)CH.sub.2 CH.sub.3                                                                    H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        16    S(O)CH.sub.2 CH.sub.3                                                                    H   H   OCH.sub.3                                                                           CH.sub.3                                                                           CH                                        17    S(O)CH.sub.2 CH.sub.3                                                                    H   H   Cl    OCH.sub.3                                                                          CH                                        18    S(O)CH.sub.2 CH.sub.3                                                                    H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        19    S(O)CH.sub.2 CH.sub.3                                                                    H   H   OCH   OCH.sub.3                                                                          N                                         20    S(O)CH.sub.2 CH.sub.3                                                                    H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         21    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        22    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   H   OCH.sub.3                                                                           CH.sub.3                                                                           CH                                        23    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   H   Cl    OCH.sub.3                                                                          CH                                        24    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        25    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         26    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         27    SO.sub.2 CH.sub.2 CH.sub.3                                                               CH.sub.3                                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         28    S(O)CH.sub.3                                                                             H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        29    S(O)CH.sub.3                                                                             H   H   OCH.sub.3                                                                           CH.sub.3                                                                           CH                                        30    S(O)CH.sub.3                                                                             H   H   Cl    OCH.sub.3                                                                          CH                                        31    S(O)CH.sub.3                                                                             H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        32    S(O)CH.sub.3                                                                             H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         33    S(O)CH.sub.3                                                                             CH.sub.3                                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         34    SO.sub.2 CH.sub.3                                                                        H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        35    SO.sub.2 CH.sub.3                                                                        H   H   OCH.sub.3                                                                           CH.sub.3                                                                           CH                                        36    SO.sub.2 CH.sub.3                                                                        H   H   Cl    OCH.sub.3                                                                          CH                                        37    SO.sub.2 CH.sub.3                                                                        H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        38    SO.sub.2 CH.sub.3                                                                        H   H   OCH.sub. 3                                                                          OCH.sub.3                                                                          N                                         39    SO.sub.2 CH.sub.3                                                                        H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         40    S(O)CH(CH.sub.3).sub.2                                                                   H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        41    S(O)CH(CH.sub.3).sub.2                                                                   H   H   OCH.sub.3                                                                           CH.sub.3                                                                           CH                                        42    S(O)CH(CH.sub.3).sub.2                                                                   H   H   Cl    OCH.sub.3                                                                          CH                                        43    S(O)CH(CH.sub.3).sub.2                                                                   H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        44    S(O)CH(CH.sub.3).sub.2                                                                   H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         45    S(O)CH(CH.sub.3).sub.2                                                                   H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         46    SO.sub.2 CH(CH.sub.3).sub.2                                                              H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        47    SO.sub.2 CH(CH.sub.3).sub.2                                                              H   H   OCH.sub.3                                                                           CH.sub.3                                                                           CH                                        48    SO.sub.2 CH(CH.sub.3).sub.2                                                              H   H   Cl    OCH.sub.3                                                                          CH                                        49    SO.sub.2 CH(CH.sub.3).sub.2                                                              H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        50    SO.sub.2 CH(CH.sub.3).sub.2                                                              H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         51    SO.sub.2 CH(CH.sub.3).sub.2                                                              H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         52    SO.sub.2 CH(CH.sub.3).sub.2                                                              CH.sub.3                                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         53    SO.sub.2 (CH.sub.2).sub.3 CH.sub.3                                                       H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        54    SO.sub.2 (CH.sub.2).sub.3 CH.sub. 3                                                      H   H   OCH.sub.3                                                                           CH.sub.3                                                                           CH                                        55    SO.sub.2 (CH.sub.2).sub.3 CH.sub.3                                                       H   H   Cl    OCH.sub.3                                                                          CH                                        56    SO.sub.2 (CH.sub.2).sub.3 CH.sub.3                                                       H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        57    SO.sub.2 (CH.sub.2).sub.3 CH.sub.3                                                       H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         58    SO.sub.2 (CH.sub.2).sub.3 CH.sub.3                                                       H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         59    SO.sub.2 (CH.sub.2).sub.3 CH.sub.3                                                       CH.sub.3                                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         60    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   CH.sub.3                                                                          OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        61    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                           CH                                        62    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   CH.sub.3                                                                          CH.sub.3                                                                            CH.sub.3                                                                           CH                                        63    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   CH.sub.3                                                                          OCH.sub.3                                                                           CH.sub.3                                                                           N                                         64    SO.sub.2 CH.sub.2 CH.sub.3                                                               H   OCH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        65    OSO.sub.2 CH.sub.3                                                                       H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        66    OSO.sub.2 CH.sub.3                                                                       H   H   OCH.sub.3                                                                           CH.sub.3                                                                           CH                                        67    OSO.sub.2 CH.sub.3                                                                       H   H   Cl    OCH.sub.3                                                                          CH                                        68    OSO.sub. 2 CH.sub.3                                                                      H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        69    OSO.sub.2 CH.sub.3                                                                       H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         70    OSO.sub.2 C.sub.2 H.sub.5                                                                H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        71    OSO.sub.2 C.sub.2 H.sub.5                                                                H   H   CH.sub.3                                                                            OCH.sub.3                                                                          CH                                        72    OSO.sub.2 C.sub.2 H.sub.5                                                                H   H   Cl    OCH.sub.3                                                                          CH                                        73    OSO.sub.2 C.sub.2 H.sub.5                                                                H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        74    OSO.sub.2 C.sub.2 H.sub.5                                                                H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         75    OSO.sub.2 C.sub.2 H.sub.5                                                                H   H   CH.sub.3                                                                            OCH.sub.3                                                                          N                                         76    SO.sub.2 C.sub.2 H.sub.5                                                                 H   F   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        77    SO.sub.2 C.sub.2 H.sub.5                                                                 H   F   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        78    SO.sub.2 C.sub.2 H.sub.5                                                                 H   Cl  OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        79    SO.sub.2 C.sub.2 H.sub.5                                                                 H   Cl  Cl    OCH.sub.3                                                                          CH                                        80    SO.sub.2 C.sub.2 H.sub.5                                                                 H   Cl  CH.sub.3                                                                            CH.sub.3                                                                           CH                                        81    OSO.sub.2 CF.sub.3                                                                       H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        82    OSO.sub.2 CF.sub.3                                                                       H   H   Cl    OCH.sub.3                                                                          CH                                        83    OSO.sub.2 CF.sub.3                                                                       H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        84    OSO.sub.2 CF.sub.3                                                                       H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         85    OSO.sub.2 CF.sub.3                                                                       H   H   CH.sub.3                                                                            OCH.sub.3                                                                          N                                         86    CH.sub.2 Cl                                                                              H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        87    CH.sub.2 Cl                                                                              H   H   Cl    OCH.sub.3                                                                          CH                                        88    CH.sub.2 Cl                                                                              H   H   CH.sub.3                                                                            OCH.sub.3                                                                          N                                         89    P(O)(OCH.sub.2 CH.sub.3).sub.2                                                           H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        90    P(O)(OCH.sub.2 CH.sub.3).sub.2                                                           H   H   CH.sub.3                                                                            OCH.sub.3                                                                          CH                                        91    P(O)(OCH.sub.2 CH.sub.3).sub.2                                                           H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        92    SO.sub.2 NHCH.sub.3                                                                      H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        93    SO.sub.2 NHCH.sub.3                                                                      H   H   Cl    OCH.sub.3                                                                          CH                                        94    SO.sub.2 NHCH.sub.3                                                                      H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        95    SO.sub.2 NHCH.sub.3                                                                      H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         96    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        97    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        98    SO.sub.2 N(OCH.sub.3)CH.sub.3                                                            H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         99    SO.sub. 2 N(OCH.sub.2)CH.sub.3                                                           CH.sub.3                                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         100   SO.sub.2 NHCH.sub.2 CH.sub.3                                                             H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        101   SO.sub.2 NHCH.sub.2 CH.sub.3                                                             H   H   Cl    OCH.sub.3                                                                          CH                                        102   SO.sub.2 NHCH.sub.2 CH.sub.3                                                             H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        103   SO.sub.2 NHCH.sub.2 CH.sub.3                                                             H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         104   SO.sub.2 NHCH.sub.2 CH.sub.3                                                             H   H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         105   SO.sub.2 NHCH.sub.2 CH.sub.3                                                             CH.sub.3                                                                          H   OCH.sub.3                                                                           CH.sub.3                                                                           N                                         106   SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                    H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        107   SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                    H   H   CH.sub.3                                                                            OCH.sub.3                                                                          CH                                        108   SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                    H   H   Cl    OCH.sub.3                                                                          CH                                        109   SO.sub.2 NHCH.sub.2 CH.sub.2 CH.sub.3                                                    H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         110                                                                                  ##STR56## H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        111                                                                                  ##STR57## H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        112   CO.sub.2 CH.sub.2 cyclopropyl                                                            H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        113   CO.sub.2 CH.sub.2 cyclopropyl                                                            H   H   Cl    OCH.sub.3                                                                          CH                                        114   CO.sub.2 CH.sub.2 cyclopropyl                                                            H   H   CH.sub.3                                                                            CH.sub.3                                                                           CH                                        115   CO.sub.2 CH.sub.2 cyclopropyl                                                            H   H   OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         116   CO.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                          CH                                        117   CO.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                          CH                                        118   CO.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                         Cl    OCH.sub.3                                                                          CH                                        119   CO.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                         CH.sub.3                                                                            CH.sub.3                                                                           CH                                        120   CO.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                         OCH.sub.3                                                                           OCH.sub.3                                                                          N                                         121   CO.sub.2 CH.sub.3                                                                        H   OCH.sub.3                                                                         CH.sub.3                                                                            OCH.sub.3                                                                          N                                         __________________________________________________________________________

Test A

Seeds of large crabgrass (Digitaria sanguinalis), barnyardgrass(Echinochloa crus-galli), giant foxtail (Setaria faberi), wild oats(Avena fatua), cheatgrass (Bromus secalinus), velvetleaf (Abutliontheophrasti), cultivated morningglory (Ipomoea coccinea, variety ScarletO'Hara), cocklebur (Xanthium pensylvanicum), G522 sorghum (Sorghumvulgare, variety Funk G522), G4646 corn (Zea mays, variety Funk G4646),Williams soybeans (Glycine max, variety Williams), USH11 sugarbeet (Betavulgaris, variety Union Sugarbeet Co. USH11), Coker cotton (Gossypiumhirsutum, variety Coker 315), dry seeded rice (Oryza sativa, varietyCalifornia Rice Coop. M101), Era wheat (Triticum aestivum, variety Eraspring), Klages barley (Hordeum vulgare, variety Klages spring) andpurple nutsedge (Cyperus rotundus) tubers were planted and treatedpreemergence with the test chemicals dissolved in a non-phytotoxicsolvent. At the same time, these crop and weed species were treated witha soil/foliage application. At the time of treatment, the plants rangedin height from 2 to 18 cm. Treated plants and controls were maintainedin a greenhouse for sixteen days, after which all species were comparedto controls and visually rated for response to treatment. The ratings,summarized in Table A, are based on a numerical scale extending from0=no injury, to 10=complete kill. The accompanying descriptive symbolshave the following meanings:

C=chlorosis/necrosis;

B=burn;

D=defoliation;

E=emergence inhibition;

G=growth retardation;

H=formative effect;

U=unusual pigmentation;

X=axillary stimulation;

S=albinism; and

6Y=abscised buds or flowers.

"POSOL" and "PRSOL" in Table A denote post- and preemergence treatments,respectively.

    TABLE A      CMPD 1 CMPD 2 CMPD 3 CMPD 4 CMPD 5 CMPD 6 CMPD 7 CMPD 8 CMPD 9 RATE =     KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 9C 4C,9H 0 0 2G 0 0 0 0 0 0 0 0 0 4C,9H 2C,5G 3C,9G 9     H CULT MORNINGLRY 10C 10C 1H 0 9C 4C,8G 1H 0 0 0 0 0 0 0 10C 4C,9G 9C     5C,9G COCKLEBUR 10C 9C 1H 0 5C,9G 3C,8G 2H,5G 0 2G 0 0 0 0 0 10C 10C 10C     9C PURPLE NUTSEDGE 9C 4C,9G 0 0 3C,8G 2C 0 0 0 0 0 0 0 0 6C,9G 2C,9G     4C,8G 2C,5G LARGE CRABGRASS 2C,8G 5G 0 0 0 0 0 0 2G 0 0 0 0 0 2G 0 3G 0     BARNYARDGRASS 9C 9C 2H 0 3C,8H 3C,7H 1H 0 4C,8H 0 0 0 0 0 9C 4C,9H 3C,9H     3C,7H WILD OATS 4C,9G 9G 0 0 3C,8G 0 0 0 9G 0 0 0 0 0 9G 9G 3C,9G 8G ERA     WHEAT 9C 4C,9G 2G 0 6G 0 2G 0 9G 0 0 0 0 0 2C,9G 9G 9C 7G G4646 CORN 2H     0 0 0 0 0 0 0 3C,9G 0 0 0 0 0 4C,9G 3C,7H 3C,8H 1H WILLMS SOYBEANS 4C,9H     2C,4G 0 0 1C 0 0 0 0 0 0 0 0 0 4C,9G 2C,7H 4C,8H 3H RICE DRY SEEDED     6C,9G 9C 0 0 9C 5G 2G 0 8G 0 0 0 0 0 9C 9C 9C 5C,9G G522 SORGHUM 9C 9C     3G 0 9C 9C 2C,5G 2C,2G 3C,8H 0 0 0 0 0 9C 9C 5C,9G 4C,9G CHEAT GRASS 10C     9C 2G 0 5C,8G 7G 0 0 3C,8G 0 0 0 0 0 9C 4C,8G 4C,9G 3C,7G USH11 SUGARBEET      9C 9C 0 0 9C 3C,7H 0 0 3C,7G 0 0 0 0 0 10C 9C 9C 4C,8G VELVETLEAF 10C     5C,9G 0 0 7G 0 0 0 0 0 0 0 0 0 10C 4C,9H 9C 4C,9H GIANT FOXTAIL 9C 6C,9G     2G 0 2C,4G 2G 0 0 2C,5G 0 0 0 0 0 4C,9G 4C,8G 3C,5G 2G KLAGES BARLEY     5C,9G 2C,8G 0 0 2C,6G 0 0 0 3C,7G 0 0 0 0 0 9G 7G 2C,8G 4G       CMPD 10 CMPD 11 CMPD 12 CMPD 13 CMPD 14 CMPD 15 CMPD 16 CMPD 17 CMPD     18 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 3C,8H 2C,3G 3C,8H 2G 0 0 0 0 0 0 10C 3C,9H 3C,9H     3C,8H 4C,8H 0 3C,8H 2C CULT MORNINGLRY 4C,9H 3C,5H 3C,7H 2C,2H 0 0 1C,3G     0 0 0 10C 10C 6C,9G 6C,9H 5C,9G 2C,7H 4C,8H 3G COCKLEBUR 4C,9H 3C,7H     3C,9H 2C,3H 4C,8H 2H 3C,9G 3H 2C,5G 0 10C 10C 9C 4C,9H 4C,8H 1H 3C,8H     3C,5G PURPLE NUTSEDGE 2C,4G 0 0 0 0 0 0 0 0 0 4C,9G 9G 9G 6G 3C,5G 0 2G     2G LARGE CRABGRASS 0 0 0 0 0 0 0 0 0 0 9G 2C,5G 7G 2G 0 0 2G 0 BARNYARDGR     ASS 3C,6H 5H 5H 3H 2H 0 5H 0 7H 0 10C 10C 9C 3C,9H 5C,9H 3C,7H 3C,8H     3C,6H WILD OATS 2C,6G 0 2C,8G 5G 2G 0 0 0 7G 0 3C,9G 3C,9G 4C,9G 3C,8G     9G 4G 2C,9G 9G ERA WHEAT 4G 0 7G 5G 3G 0 6G 0 8G 2G 4C,9G 8G 9G 9G 7G 3G     9G 8G G4646 CORN 0 0 0 0 5H 0 3H 0 6H 0 3C,8H 2G 3G 2G 0 0 1H 0 WILLMS     SOYBEANS 1C,1H 0 0 0 0 0 0 0 0 0 9C 3C,8G 5C,9G 4C,9G 3C,6H 2G 3C,8G     3C,3H RICE DRY SEEDED 9G 5G 3C,5G 2C,5G 2G 0 2G 0 2C,5G 0 9C 9C 9C 9C     5C,9G 2G 5C,9G 5C,9G G522 SORGHUM 4C,9G 4C,9G 9C 3C,7H 2C,5G 0 8G 0     3C,8H 0 10C 9C 3C,9G 3C,9G 5C,9G 4C,9G 3C,9G 4C,9G CHEAT GRASS 8G 3G 5G     3G 3G 0 7G 0 2C,8G 0 10C 9C 10C 4C,9G 9G 9G 9C 9G USH11 SUGARBEET 3C,8H     6G 4C,8G 3C,3H 2H 0 3H 0 3H 0 9C 9C 9C 4C,9H 4C,8H 3C,6G 3C,7H 3C,5G     VELVETLEAF 2C,3G 0 3C,7H 2C,5G 0 0 0 0 0 0 10C 5C,9H 10C 5C,9H 4C,8H 5G     3C,7G 3C,6G GIANT FOXTAIL 1C 0 0 0 0 0 0 0 2G 0 10C 9C 9C 3C,9G 9C 3C,7G     3C,9G 3C,6G KLAGES BARLEY 0 0 3G 0 2G 0 0 0 2C,8G 4G 9C 3C,8G 2C,8G 6G     4G 0 2C,8G 6G       CMPD 19 CMPD 20 CMPD 21 CMPD 22 CMPD 23 CMPD 24 CMPD 25 CMPD 26 CMPD     27 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 0 0 0 0 10C 9C 2C,5G 0 10C 2C,6G 2G 0 0 0 0 0 5C,9G     4C,8G CULT MORNINGLRY 0 0 0 0 10C 10C 2C,7G 0 10C 4C,9G 2C,5H 0 0 0 2C     5C,9G 2C,7G COCKLEBUR 2H 0 2H 0 10C 10C 5G 0 10C 7H 4G 0 1H 0 0 0 10C     2C,8G PURPLE NUTSEDGE 0 0 0 0 10C 9G 0 0 3C,8G 7G 0 0 0 0 0 0 0 0 LARGE     CRABGRASS 0 0 0 0 5C,9G 8G 3G 0 7G 2G 2G 0 0 0 0 0 0 0 BARNYARDGRASS 0 0     2G 0 9C 9C 2C,5H 2G 9C 5C,9H 2C,5G 0 3G 0 0 0 3C,7G 4G WILD OATS 2G 0 0     0 3C,9G 3C,9G 0 0 8G 6G 2G 0 8G 0 0 0 3C,6G 0 ERA WHEAT 5G 0 3G 0 5C,9G     10C 0 0 8G 4G 6G 0 9G 0 3G 0 4C,9G 0 G4646 CORN 0 0 0 0 1C,4H 2G 0 0 0 0     0 0 3G 0 0 0 2H 0 WILLMS SOYBEANS 2C,2H 0 3C 0 9C 5C,9G 3C,4H 1C,1H     3C,8H 3C,4G 3C,5H 1H 2C,2H 0 0 0 4C,9G 3C,8G RICE DRY SEEDED 0 0 0 0 9C     9C 3G 0 10C 5C,9G 3G 0 4G 0 0 0 5G 2G G522 SORGHUM 0 0 3C,3G 0 9C 9C     3C,8G 3G 9C 9C 3C,7G 2G 2G 0 0 0 4C,9G 3C,8G CHEAT GRASS 0 0 0 0 9C 9C     5G 0 5C,9G 9G 3G 0 8G 0 2G 0 7G 3G USH11 SUGARBEET 1C 0 2H 0 10C 10C     2C,5G 2G 9C 5C,9G 3G 2G 2H 0 0 0 6C,9G 3C,6G VELVETLEAF 3G 0 0 0 10C 10C     2G 0 9C 8G 3C,7G 3H 0 0 2G 0 6C,9G 3C,7G GIANT FOXTAIL 2G 0 0 0 10C 10C     6G 0 10C 4C,9G 2C,7G 5G 0 0 2G 0 4C,8G 5G KLAGES BARLEY 2G 0 0 0 5C,9G     4C,9G 0 0 3C,9G 3G 0 0 7G 0 0 0 2G 0       CMPD 28 CMPD 29 CMPD 30 CMPD 31 CMPD 32 CMPD 33 CMPD 34 CMPD 35 CMPD     36 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 3C,9G 4C,9G 4C,8H 3G 0 0 1H 0 0 0 2C,4H 0 9C 4C,8G     0 0 6G 2G CULT MORNINGLRY 10C 5C,9H 4C,9G 3C,7H 3C,6G 0 0 0 0 0 2C 0     6C,9G 4C,9G 3G 0 5C,9H 3C,7H COCKLEBUR 10C 4C,9H 4C,9H 2C,6H 2H 0 0 0 0     0 1C 0 10C 4C,9H 2C,4G 0 4C,9H 4C,6H PURPLE NUTSEDGE 2C,9G 9G 2C,8G 5G 0     0 0 0 0 0 0 0 3C,9G 2C,9G 0 0 3G 0 LARGE CRABGRASS 4C,9G 2C,8G 3C,7G     2C,5G 2C,4G 0 2G 0 0 0 0 0 5C,9G 9G 0 0 2C,8G 5G BARNYARDGRASS 9C 9C 9C     4C,8H 4C,9H 3C,6H 3C,8H 2H 0 0 0 0 9C 4C,9G 2C,8H 0 9C 2C,8H WILD OATS     6C,9G 9G 4C,9G 2C,9G 9G 3G 2C,9G 4G 0 0 0 0 2C,9G 9G 8G 0 9G 3G ERA     WHEAT 6C,9G 9G 4C,9G 2C,9G 7G 4G 8G 4G 0 0 0 0 4C,9G 2C,9G 9G 0 9G 0     G4646 CORN 2U,9G 9G 2C,9G 2C,5H 2C,5G 0 2C,7H 1H 2G 0 0 0 4C,9G 2C,8G 0     0 0 0 WILLMS SOYBEANS 9C 9C 5C,9G 4C,8H 3C,3H 1C 3C,5H 1C,1H 0 0 2C,5H 0     9C 5C,9G 1C,5H 2C 4C,8G 2C,4H RICE DRY SEEDED 9C 9C 9C 5C,9G 8G 0 4C,9G     2C,2G 0 0 1C 0 5C,9G 4C,9G 7G 0 4C,9G 2C,6G G522 SORGHUM 9C 5C,9G 4C,9G     3C,7G 3C,8H 3C,3H 3C,8H 0 0 0 0 0 9C 6C,9G 2G 0 3C,9G 3C,9G CHEAT GRASS     9C 9C 5C,9G 4C,9G 3C,9G 7G 4C,9G 7G 0 0 0 0 9C 4C,9G 8G 4G 3C,9G 9G     USH11 SUGARBEET 9C 9C 5C,9G 2C,4G 3C,4H 2C 2C,2H 0 0 0 2C 0 4C,9H 2C,6H     2G 0 4C,8H 2C,7G VELVETLEAF 9C 4C,8H 4C,9H 3C,6H 5G 0 2C,5H 0 0 0 1C 0     10C 10C 5G 0 7G 0 GIANT FOXTAIL 9C 9C 5C,9G 3C,7G 4C,9G 2C,5G 2G 0 0 0 0     0 9C 9C 7G 0 4C,9G 3C,9G KLAGES BARLEY 5C,9G 4C,9G 4C,9G 3C,7G 2C,5G 3G     3C,7G 3G 0 0 0 0 4C,9G 3C,8G 4G 0 3C,8G 2C,7G       CMPD 37 CMPD 38 CMPD 39 CMPD 40 CMPD 41 CMPD 42 CMPD 43 CMPD 44 CMPD     45 RATE = KG/HA  0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 0 0 0 0 0 0 4C,9G 9H 3C,9G 3C,8H 3C,5H 0 2C,3G 0 0     0 0 0 CULT MORNINGLRY 0 0 0 0 0 0 10C 4C,8H 9C 3C,8H 3C,3H 0 3C,6G 1H 0     0 0 0 COCKLEBUR 0 0 0 0 0 0 10C 4C,9G 9C 3C,9G 3C,6H 2C,2H 3C,6G 1C,1H     2C,2H 1H 2C,2H 0 PURPLE NUTSEDGE 0 0 0 0 0 0 9G 8G 3G 0 0 0 0 0 0 0 0 0     LARGE CRABGRASS 0 0 0 0 0 0 3G 0 0 0 0 0 2G 0 0 0 0 0 BARNYARDGRASS 0 0     0 0 0 0 9C 3C,9H 4C,9G 4C,8H 3C,4G 0 3C,7G 1H 0 0 0 0 WILD OATS 0 0 0 0     0 0 3C,9G 8G 3C,9G 3C,8G 5G 0 9G 2G 0 0 0 0 ERA WHEAT 0 0 0 0 0 0 9G 8G     9G 9G 2G 0 9G 2G 0 0 0 0 G4646 CORN 0 0 0 0 0 0 4C,9H 2G 7G 0 0 0 0 0 0     0 0 0 WILLMS SOYBEANS 2H 0 0 0 0 0 4C,9G 4C,9G 4C,7G 3C,3H 0 0 1C 0 0 0     0 0 RICE DRY SEEDED 0 0 0 0 0 0 5C,9G 5C,9G 5C,9G 3C,7G 3G 0 4C,9G 0 0 0     0 0 G522 SORGHUM 0 0 0 0 0  0 4C,9G 4C,9G 4C,9G 4C,9G 3C,9G 0 4C,8H 4G 0     0 0 0 CHEAT GRASS 0 0 0 0 0 0 9C 6G 5C,9G 4C,8G 6G 0 3C,9G 8G 0 0 0 0     USH11 SUGARBEET 0 0 0 0 0 0 9C 9C 4C,8H 3C,7G 3C,6H 0 3C,6G 0 0 0 0 0     VELVETLEAF 0 0 0 0 4G 0 4C,9H 4C,7H 3C,8H 3C,6H 0 0 2C,2G 0 0 0 0 0     GIANT FOXTAIL 0 0 0 0 0 0 4C,9G 3C,7G 3C,7G 3G 0 0 3C,7G 4G 0 0 0 0     KLAGES BARLEY 0 0 0 0 0 0 8G 7G 8G 5G 0 0 7G 4G 0 0 0 0        CMPD 46 CMPD 47 CMPD 48 CMPD 49 CMPD 50 CMPD 51 CMPD 52 CMPD 53 CMPD     54 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 3C,8G 3C,7H 0 0 0 0 0 0 0 0 2G 0 3C,5H 3G 5G 0 0 0     CULT MORNINGLRY 10C 9C 2G 0 3C,8H 3C,6H 2H 0 0 0 2C,7H 0 2C,6H 2C,2H     3C,7G 3C,5H 0 0 COCKLEBUR 3C,9H 2C,8G 0 0 3C,8H 2C 0 0 0 0 2C,6H 0 1C,4G     0 3C,5G 3G 0 0 PURPLE NUTSEDGE 9G 2C,9G 0 0 5G 3G 0 0 0 -- 0 -- 0 0     3C,8G -- 0 0 LARGE CRABGRASS 6G 4G 0 0 0 0 2G 0 0 0 3G 0 2G 0 0 0 0 0     BARNYARDGRASS 9C 9C 2G 0 7H 4H 2G 0 2G 0 4G 0 4G 2G 3C,8H 4H 0 0 WILD     OATS 8G 2G 0 0 0 0 0 0 4G 0 2G 0 0 0 2C,9G 0 0 0 ERA WHEAT 8G 8G 0 0 0 0     0 0 7G 0 4G 0 0 0 7G 0 0 0 G4646 CORN 3G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0     0 WILLMS SOYBEANS 4C,9G 3C,7H 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 RICE DRY     SEEDED 9C 4C,9G 0 0 2C,7G 2G 0 0 2C 0 1C 0 2C,2G 0 9G 5G 0 0 G522     SORGHUM 4C,9G 4C,9G 4G 0 3C,9G 3C,7H 0 0 3G 0 3G 0 4H 0 3C,9H 7G 0 0     CHEAT GRASS 5C,8G 5G 4G 0 5G 3G 0 0 4G 0 2G 0 2G 0 9G 0 0 0 USH11     SUGARBEET 6C,8G 3C,7G 3H 0 2C,4G 1H 0 0 1H 0 0 0 2C,5G 0 3C,7G 4H 0 0     VELVETLEAF 4C,9H 2C,7H 0 0 -- 0 0 0 0 0 2G 0 6G 5G 2C,5G 0 0 0 GIANT     FOXTAIL 4C,9G 2C,8G 0 0 0 0 2C,7G 0 0 0 3G 0 5G 2G 2C,5G 3G 0 0 KLAGES     BARLEY 9C 7G 2G 0 4G 0 0 0 5G 0 3G 0 0 0 7G 0 0 0       CMPD 55 CMPD 56 CMPD 57 CMPD 58 CMPD 59 CMPD 60 CMPD 61 CMPD 62 CMPD     63 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 0 0 0 0 0 0 0 0 0 0 9C 3C,9G 4G 2G 2G 0 3C,8H 3C,6G     CULT MORNINGLRY 3H 0 0 0 0 0 0 0 0 0 10C 3C,9G 1H 0 0 0 3C,7G 3C,3H     COCKLEBUR 1H 0 0 0 0 0 0 0 0 0 10C 9C 2H 0 0 0 3C,7G 2C,2H PURPLE     NUTSEDGE 0 0 0 0 0 0 0 0 -- 0 4C,9G 8G 3G 0 0 0 2G -- LARGE CRABGRASS 0     0 0 0 0 0 0 0 0 0 4C,7G 2G 0 0 0 0 0 0 BARNYARDGRASS 0 0 0 0 0 0 0 0 0 0     10C 9C 0 0 0 0 3G 0 WILD OATS 0 0 0 0 0 0 0 0 0 0 5C,9G 7G 0 0 0 0 0 0     ERA WHEAT 0 0 0 0 0 0 0 0 0 0 9C 9G 0 0 0 0 0 0 G4646 CORN 0 0 0 0 0 0 0     0 0 0 3C,7H 0 1C,4H 0 0 0 0 0 WILLMS SOYBEANS 0 0 0 0 0 0 0 0 0 0 5C,9G     5C,9G 2C,8G 0 3H 0 3C,7G 2C,3H RICE DRY SEEDED 0 0 0 0 0 0 0 0 0 0 9C 9C     4G 0 2G 0 6G 0 G522 SORGHUM 0 0 0 0 0 0 0 0 0 0 9C 5C,9G 2G 0 0 0 7G 0     CHEAT GRASS 0 0 0 0 0 0 0 0 0 0 9C 4C,9G 0 0 0 0 0 0 USH11 SUGARBEET 2H     0 0 0 0 0 0 0 0 0 10C 4C,8G 5C,9G 3C,7G 3C,7H 0 3C,8H 3C,8G VELVETLEAF 0     0 0 0 0 0 0 0 0 0 10C 10C 3C,7G 3G 3G 0 3C,7G 3G GIANT FOXTAIL 0 0 0 0 0     0 0 0 0 0 4C,9G 7G 0 0 0 0 0 0 KLAGES BARLEY 0 0 0 0 0 0 0 0 0 0 5C,9G     6G 0 0 0 0 0 0       CMPD 64 CMPD 65 CMPD 66 CMPD 67 CMPD 68 CMPD 69 CMPD 70 CMPD 71 CMPD     72 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 5C,9G 9C 9C 9C 9C 4C,8G 10C 9C 9C 4C,9G 3C,5G 3C,4G 9     C 9C 9C 9C 9C 9C CULT MORNINGLRY 10C 10C 10C 10C 10C 10C 10C 4C,9G 10C     4C,9H 3C,6G 3G 10C 10C 9C 10C 10C 10C COCKLEBUR 10C 10C 9C 10C 10C 10C     10C 9C 10C 8G 3G 2G 10C 10C 10C 10C 10C 10C PURPLE NUTSEDGE 5C,9G 5C,9G     9C 5C,9G 5C,9G 3C,7G 5C,9G 3C,9G 5C,9G 3C,9G 5G 0 10C 9C 9C 9G -- 3C,9G     LARGE CRABGRASS 6G 4G 6C,9G 4C,9G 9C 3C,8G 5C,9G 8G 6C,9G 4C,8G 6G 4G     5C,9G 4G 8G 5G 2C,7G -- BARNYARDGRASS 9C 3C,9H 9C 9C 9C 9C 9C 9C 9C 9C     9C 2C,2H 9C 9C 9C 9C 9C 9C WILD OATS 8G 2C,3G 10C 9C 9C 5C,9G 6C,9G 9G     9C 9C 5C,9G 1C 5C,9G 9G 4C,9G 9G 9G 9G ERA WHEAT 7G 5G 6C,9G 6C,9G 9C 9G     9G 5G 4C,9G 5C,9G 5C,9G 8G 9G 7G 9G 8G 9G 5G G4646 CORN 3C,6G 3G 7U,9C     7U,9C 6U,9G 3U,9G 5U,9G 9H 2C,9G 3C,7G 4U,9G 9G 9C 9C 3C,9G 3C,8H 3C,9H     2C,7G WILLMS SOYBEANS 5C,9G 9C 9C 9C 9C 5C,9G 5C,9G 5C,9G 5C,9H 9C 4C,8H     2C,5G 9C 9C 9C 9C 9C 3C,8H RICE DRY SEEDED 9C 5C,9G 9C 9C 9C 9C 5C,9G 9C     9C 9C 9C 5C,9G 9C 9C 9C 3C,8G 9C 8G G522 SORGHUM 3C,9G 4C,9G 9C 9C 6C,9G     4C,9G 9C 9C 9C 6C,9G 3C,7G 3C,3G 9C 9C 9C 9G 9C 9C CHEAT GRASS 3C,8G     4C,9G 9C 9C 9C 9C 9C 9C 9C 6C,9G 5C,9G 9G 10C 5C,9G 9C 4C,9G 9C 9G USH11     SUGARBEET 9G 3C,8G 9C 9C 10C 10C 9C 9C 10C 9C 3C,5G 5H 9C 9C 10C 9C 10C     9C VELVETLEAF 9C 5C,9G 9C 9C 10C 9C 10C 3C,9G 10C 4C,9H 2H 3G 10C 10C 9C     9C 9C 8G GIANT FOXTAIL 7G 3G 9C 10C 9C 9C 6C,9G 8G 10C 5C,9G 3C,9G 2G     10C 9C 9C 3C,8G 4C,9G 2C,7G KLAGES BARLEY 7C,7G 2C,6G 9C 6C,9G 6C,9G     4C,9G 3C,8G 5G 6C,9G 5C,9G 5C,9G 3C,9G 3C,9G 6G 4C,9G 7G 2C,9G 4G       CMPD 73 CMPD 74 CMPD 75 CMPD 76 CMPD 77 CMPD 78 CMPD 79 CMPD 80 CMPD     81 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01        POSOL COKER COTTON 5C,9G 3C,8G 2C,5G 1C 3C,5G 2C,5G 0 0 0 0 0 0 0 0 0 0      4C,9G 0 CULT MORNINGLRY 10C 9C 3C,8H 2C,3H 3C,7H 1C,1H 0 0 0 0 0 0 0 0     0 0 4C,9G 3C,6G COCKLEBUR 10C 10C 3C,5H 1H 2C,6H 9C 2H 0 0 0 0 0 0 0 0 0     10C 10C PURPLE NUTSEDGE 4C,9G 4C,8G 5G 0 3G 0 0 0 -- 0 0 0 -- 0 0 0 --     5C,9G LARGE CRABGRASS 5C,9G 3C,7G 7G 2G 3C,7G 3G 0 0 0 0 0 0 1C,3G 0 0 0     3C,8G -- BARNYARDGRASS 10C 9C 9C 3C,7H 9C 9C 0 0 0 0 0 0 0 0 0 0 10C     3C,9H WILD OATS 5C,9G 3C,9G 5C,9G 4C,9G 9C 9C 0 0 0 0 0 0 0 0 0  0 2C,5G     0 ERA WHEAT 2C,9G 9G 9G 6G 2C,9G 2C,9G 0 0 0 0 0 0 0 0 0 0 2G 0 G4646     CORN 3C,9H 2C,5G 5C,9G 2C,9G 5C,9G 5C,9G 0 0 0 0 0 0 0 0 0 0 9C 9G     WILLMS SOYBEANS 9C 9C 4C,8H 5G 4C,9G 7H 0 0 0 0 0 0 0 0 0 0 3C,8G 4G     RICE DRY SEEDED 9C 9C 9C 9C 9C 9C 0 0 0 0 0 0 0 0 0 0 9C 5C,9G G522     SORGHUM 9C 9C 5C,9G 4C,9G 9C 5C,9G 0 0 0 0 0 0 0 0 0 0 9C 4C,9G CHEAT     GRASS 9C 5C,9G 4C,9G 9G 5C,9G 3C,9G 0 0 0 0 0 0 0 0 0 0 2C,6G 2G USH11     SUGARBEET 10C 9C 4C,9H 3C,6H 3C,6G 5C,9G 0 0 0 0 0 0 2C,6G 3G 0 0 10C 9C     VELVETLEAF 4C,9G 8G 3C,6H 0 0 7G 0 0 0 0 0 0 0 0 3G 0 10C 9C GIANT     FOXTAIL 9C 2C,9G 9C 3C,7G 9C 3C,8G 0 0 0 0 0 0 3G 0 0 0 9C 4C,8G KLAGES     BARLEY 3C,9G 7G 9C 9G 9C 9C 0 0 0 0 0 0 0 0 0 0 8G 7G       CMPD 82 CMPD 83 CMPD 84 CMPD 85 CMPD 86 CMPD 87 CMPD 88 CMPD 89  CMPD     90 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 2G 0 0 0 0 0 0 0 9C 4G 0 0 0 0 1H 0 0 0 CULT     MORNINGLRY 2G 0 2C,2G 0 3C,7G 0 3C,4H 0 4C,8G 3C,3G 0 0 0 0 3C,4G 0 0 0     COCKLEBUR 5C,9G 4C,9G 5C,9G 3C,8H 4C,9H 2H 4C,9H 2H 5C,9G 1C 0 0 0 0     3C,6G 2G 0 0 PURPLE NUTSEDGE 10C -- 5G 0 0 0 -- 0 10C 10C -- 0 0 0 0 0 0     0 LARGE CRABGRASS 5G 0 5G 0 3C,7G 0 5G -- 9C 3C,6G 0 0 0 0 0 0 0 0     BARNYARDGRASS 3C,8H 2C,5G 3C,8H 3G 4C,9G 3C,6G 9C 3C,8G 9C 3C,8H 0 0 0 0     4C,9H 2G 0 0 WILD OATS 2G 0 2C,6G 0 0 0 0 0 3C,5G 0 0 0 0 0 2C,5G 0 0 0     ERA WHEAT 2G 0 0 0 0 0 0 0 3C,5G 2G 0 0 0 0 3C,5G 0 0 0 G4646 CORN 3C,9H     3G 3C,7H 0 4C,9G 4C,8G 5C,9G 9G 4C,9G 3C,7G 2G 0 0 0 3C,8H 0 0 0 WILLMS     SOYBEANS 1H 0 0 0 3C,3H 0 3G 0 9C 4C,9G 0 0 0 0 3C,7G 1H 3H 0 RICE DRY     SEEDED 3C,8G 8G 9C 7G 5C,9G 8G 9C 3C,8G 9C 3C,8G 0 0 0 0 6G 0 0 0 G522     SORGHUM 5C,9H 2C,8G 4C,9G 2C,8G 5C,9G 3C,8G 5C,9G 3C,9G 3C,9G 3C,7G     2C,6G 0 0 0 3C,9H 2C,4G 0 0 CHEAT GRASS 2C,5G 0 4G 0 0 0 0 0 -- -- -- --     -- -- -- -- -- -- USH11 SUGARBEET 9C 2C,4H 3C,5H 4G 2H 0 3C,6G 2H 10C     10C 3G 0 0 0 10C 4G 3G 0 VELVETLEAF 5G 0 -- 0 -- 0 3C,7G 0 9C 10C 0 0 0     0 3C,6G 0 0 0 GIANT FOXTAIL 0 0 2C,5G 0 4C,9G 3C,8G 5C,9G 3C,7G 9C 2G 0     0 0 0 2C,5G 0 0 0 KLAGES BARLEY 4G 0 2C,5G 0 0 0 3G 0 2C,5G 0 0 0 0 0     3C,8G 0 0 0 DOWNY BROME       -- -- 5C,9G 5C,9G 0 0 0 0 4C,7G 0 0     0        CMPD 91 CMPD 92 CMPD 93 CMPD 94 CMPD 95 CMPD 96 CMPD 97 CMPD 98 C     MPD 99 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01     0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 0 0 10C 10C 6C,9G 4C,9G 2C,5G 2G 0 0 4C,8G 5G 0 0 0 0      4C,9G 3C,9H CULT MORNINGLRY 0 0 10C 10C 9C 4C,9G 1H 0 2C 0 10C 10C     2C,7G 0 2G 0 3C,8G 2C,5H COCKLEBUR 0 0 10C 10C 10C 3C,8H 2G 0 0 0 10C     4C,9H 2C 0 0 0 4C,9H 3C,8H PURPLE NUTSEDGE 0 0 9C 5C,9G 2C,9G 2C,6G 0 0     0 0 9G 2C,5G 5G 0 4G 0 0 0 LARGE CRABGRASS 0 0 8G 5G 5G 0 0 0 0 0 10C 9G     0 0 0 0 0 0 BARNYARDGRASS 0 0 9C 9C 3C,9H 3C,7H 1H 0 0 0 10C 9C 0 0 0 0     0 0 WILD OATS 0 0 5C,9G 3C,8G 5G 3G 0 0 0 0 3C,9G 9G 0 0 0 0 0 0 ERA     WHEAT 0 0 6C,9G 9G 8G 3G 0 0 0 0 3C,9G 9G 2G 0 0 0 0 0 G4646 CORN 0 0 6G     3G 3G 0 0 0 0 0 3C,9H 5G 0 0 0 0 2C,6G 0 WILLMS SOYBEANS 0 0 9C 9C 3C,7G     2C,6H 3C,4H 2H 0 0 5C,9H 6C,9G 2H 0 0 0 4C,8H 3C,6H RICE DRY SEEDED 0 0     9C 6C,9G 6C,9G 5C,9G 0 0 0 0 5C,9G 5C,9G 0 0 0 0 2G 0 G522 SORGHUM 0 0     9C 5C,9G 9C 9C 2G 0 0 0 9C 3C,9G 4G 0 0 0 3C,7H 6G CHEAT GRASS -- -- 9C     9C 2C,9G 8G 0 0 0 0 9C 9G 0 0 0 0 5G 0 USH11 SUGARBEET 0 0 9C 9C 9C 9C 0     0 0 0 10C 3C,7G 8G 4G 7G 0 10C 6H VELVETLEAF 0 0 10C 10C 4C,9H 5H 2C,7G     0 0 0 10C 9G 0 0 3G 0 9G 7G GIANT FOXTAIL 0 0 9C 9C 3C,8G 3C,6G 2G 0 0 0     10C 5C,9G 0 0 2C 0 0 0 KLAGES BARLEY 0 0 5C,9G 2C,8G 2C,5G 0 0 0 0 0     6C,9G 8G 0 0 0 0 0 0 DOWNY BROME 0 0 -- --       CMPD 100 CMPD 101 CMPD 102 CMPD 103 CMPD 104 CMPD 105 CMPD 106 CMPD     107 CMPD 108 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 5C,9G 5C,9G 5C,9G 3C,6H 3C,3H 0 0 0 0 0 3C,9H      3C,7H 3C,6G 2C,4G 0 0 2G 0 CULT MORNINGLRY 9C 9C 5C,9G 3C,8H 2C,3H 1H 0     0 0 0 2C,4H 2G 9C 3C,8H 0 0 2C,4G 0 COCKLEBUR 10C 9C 9G 2C,8H 2H 2G 3G 0     0 0 3C,9H 3C,9H 5C,9G 2C,8H 0 0 1C 0 PURPLE NUTSEDGE 4C,9G 2C,9G 9G 4G 0     -- 4G 0 -- 0 0 -- 2C,7G 2C,2G 0 0 0 0 LARGE CRABGRASS 3C,7G 3C,7G 2C,4G     0 4G 0 0 0 0 0 0 0 0 0 0 0 2G 0 BARNYARDGRASS 9C 9C 3C,9H 2C,6G 2H 0 0 0     0 0 0 0 9C 5C,9G 0 0 4G 0 WILD OATS 5C,9G 3C,9G 2C,7G 1C 2C,8G 0 0 0 0 0     0 0 9C 9C 0 0 3G 0 ERA WHEAT 9G 9G 2C,5G 3G 2C,8G 3G 0 0 0 0 0 0 9G 9G 0     0 2G 0 G4646 CORN 3C,9H 1C 0 0 0 0 0 0 0 0 0 0 2C,2G 2C 0 0 0 0 WILLMS     SOYBEANS 5C,9G 4C,9H 3C,7G 0 3C,4H 0 0 0 0 0 2C,6H 4H 3C,9G 0 0 0 0 0     RICE DRY SEEDED 9C 9C 4C,9G 2C,8G 4G 0 0 0 0 0 0 0 9C 3C,8H 0 0 0 0 G522     SORGHUM 9C 9C 5C,9G 4C,9G 0 0 0 0 0 0 0 0 5C,9G 4C,9G 0 0 2C,8G 0 CHEAT     GRASS 9C 9G 3C,9G 2C,9G 5G 0 0 0 0 0 0 0 9C 9G 0 0 5G 0 USH11 SUGARBEET     9C 9C 5C,9H 5C,9H 3C,5G 0 0 0 0 0 3C,9H 3C,8H 9C 6G 0 0 0 0 VELVETLEAF     9C 9C 3C,7H 1H 3C,5G 1H 0 0 0 0 3C,9G 5G 9C 2C,6G 8G 0 4G 0 GIANT     FOXTAIL 9C 5C,9G 3C,7G 2C 5G 0 0 0 0 0 0 0 9C 3C,8G 0 0 2G 0 KLAGES     BARLEY 5C,9G 4C,9G 2C,5G 3G 4G 0 0 0 0 0 0 0 2C,9G 2C,8G 0 0 3G 0       CMPD 109 CMPD 110 CMPD 111 CMPD 112 CMPD 113 CMPD 114 CMPD 115 CMPD     116 CMPD 117 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01       POSOL COKER COTTON 0 0 4C,9G 4C,8H 0 0 4C,8H 3C,8H 3C,9H 3C,7G 6G 0     2C,2G 0 10C 9C 5C,9G 9C CULT MORNINGLRY 1C 0 6C,9G 3C,8G 0 0 10C 10C 10C     3C,8G 0 0 1C 0 9C 9C 10C 10C COCKLEBUR 0 0 5C,9G 3C,9G 0 0 10C 10C 9C     4C,9G 3C,7G 7G 3C,8G 2H 10C 10C 10C 10C PURPLE NUTSEDGE 0 0 4G 3G 0 0 9C     5C,9G 9C 2C,8G 3G 0 0 0 10C 10C 10C 9C LARGE CRABGRASS 2G 0 9C 2G 0 0 0     0 0 0 0 0 0 0 3C,5G 2G 3C,9G 3G BARNYARDGRASS 0 0 9C 3C,8H 0 0 9C --     3C,9G 3C,7G 3C,3G 0 3C,9H 3C,7G 9C 9C 9C 5C,9G WILD OATS 0 0 2C,7G 4G 0     0 4C,9G 3G 0 0 3G 0 3C,7G 2G 5C,9G 2C,7G 3C,9G 9G ERA WHEAT 0 0 3C,9G 5G     0 0 3C,8G 3G 0 0 3G 0 3C,6G 2G 5C,9G 9G 2C,9G 9G G4646 CORN 0 0 3C,8H     2C,4G 0 0 5U,9C 3C,9G 3C,7H 3C,7H 3C,7G 2C,6G 5C,9G 2C,7H 7U,9C 5U,9C     4C,9G 9G WILLMS SOYBEANS 0 0 3C,7H 2H 0 0 9C 4C,9G 2H 0 3C,7G 2H 2H 0 9C     9C 9C 6C,9G RICE DRY SEEDED 0 0 3C,9G 4G 0 0 5C,9G 2C,8G 7G 2C,5G 2G 0     5C,9G 4C,9G 9C 9C 6C,9G 5C,9G G522 SORGHUM 0 0 9C 9G 0 0 3C,9G 3C,9H     3C,9G 3C,9G 3G 3G 3C,9G 3C,8G 5C,9G 9G 4C,9G 9G CHEAT GRASS 0 0 2C,8G 5G     0 0 -- -- -- -- -- -- -- -- 9C 9C 5C,9G 9G USH11 SUGARBEET 0 0 10C 9C 0     0 10C 9C 9C 3C,7H 5G 0 4C,9H 3C,7H 10C 9C 10C 10C VELVETLEAF 3G 0 5C,9G     3C,8G 0 0 10C 5C,9G 9C 2C,7G 3C,8G 2C,7G 0 0 10C 10C 10C 9C GIANT     FOXTAIL 2G 0 4C,9H 3C,7G 0 0 4C,9G 0 0 0 4G 0 3C,7G 2G 9C 4C,9G 10C     2C,9G KLAGES BARLEY 0 0 3C,8G 2C,5G 0 0 7G 3G 2G 0 3G 0 3G 3G 2C,9G 7G     5C,9G 9G DOWNY BROME -- -- -- -- -- -- 9C 9C 3C,9G 3G 2C,5G 2G 9C 2C,5G     -- --       CMPD 118 CMPD 119 CMPD 120 CMPD 121 RATE = KG/HA 0.05 0.01 0.05 0.01     0.05 0.01 0.05 0.01       POSOL COKER COTTON 9C 9C 9C 6C,9G 9C 3C,8H 5C,9G 4C,8G CULT MORNINGLRY     10C 10C 4C,8H 2C,6G 10C 4C,9G 10C 4C,9H COCKLEBUR 10C 10C 10C 10C 10C     5C,9G 10C 4C,9H PURPLE NUTSEDGE 10C -- 9C 9C 7G 0 6G 0 LARGE CRABGRASS     7G 6G 4C,9G 2C,7G 2C,7G 5G 3C,8G 2G BARNYARDGRASS 10C 5C,9H 10C 9C 9C     4C,8H 9C 9C WILD OATS 9G 7G 3C,9G 2C,9G 3C,9G 3C,9G 3C,9G 4C,9G ERA     WHEAT 2C,9G 8G 3C,9G 9G 7G 5G 4C,9G 9G G4646 CORN 5C,9G 2C,7H 6C,9G     3C,9G 9C 3C,9G 6U,9G 6U,9G WILLMS SOYBEANS 5C,9G 3C,8H 6C,9G 5C,9G 4C,9G     5C,9G 6C,9G 5C,9G RICE DRY SEEDED 5C,9G 4C,9G 9C 5C,9G 9C 5C,9G 9C 5C,9G     G522 SORGHUM 6C,9G 9H 5C,9G 4C,9G 9G 3C,8H 3C,9G 9G CHEAT GRASS 9G 7G     6C,9G 3C,9G 5C,9G 3C,9G 9C 9G USH11 SUGARBEET 10C 9C 10C 9C 10C 9C 10C     4C,8H VELVETLEAF 9C 9G 10C 10C 9G 4C,9H 10C 5C,9H GIANT FOXTAIL 4C,9G     3C,8G 10C 3C,9G 4C,9G 3C,6G 10C 4C,9G KLAGES BARLEY 9G 5G 6C,9G 3C,9G 6G     3G 4C,9G 4G       CMPD 1 CMPD 2 CMPD 3 CMPD 4 CMPD 5 CMPD 6 CMPD 7 CMPD 8 CMPD 9 RATE =     KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 8G 5G 0 0 2G 0 2G 0 0 0 0 0 0 0 4G 3G 1H 0 CULT     MORNINGLRY 9G 8H 0 0 5H 1H 1C 0 0 0 0 0 0 0 9G 8H 2C,8H 1C COCKLEBUR 9H     9H 0 0 3G 1C 0 0 0 0 0 0 0 0 8H 3C,5H -- -- PURPLE NUTSEDGE 10E 3C,7G 0     0 9G 8G 0 0 0 -- 0 0 10E 0 9G 3C,9G 3G 0 LARGE CRABGRASS 9G -- 9G 0 9G     5G 8G -- 2G -- -- -- -- -- 6G 2C 0 -- BARNYARDGRASS 9H 9H 0 0 3C,7G 2G     2G 0 2G 0 0 0 0 0 9H 3C,8H 3C,8H 2C WILD OATS 4C,8G 1C 0 0 0 4G 2G 0 0 0     0 0 0 0 3C,8H 6G 4C,9G 4G ERA WHEAT 10E 8G 0 0 0 0 0 0 0 0 0 0 0 0 8H 6G     4C,8G 0 G4646 CORN 5G 0 0 0 0 2G 2G 0 0 0 0 0 0 0 3C,7H 0 2G 0 WILLMS     SOYBEANS 3G 0 0 0 3G 0 5G 0 0 0 0 0 0 0 3G 5G 3G 1H RICE DRY SEEDED 10E     4C,9H 0 0 3C,8G 6G 2C,5G 0 0 0 0 0 0 0 10E 3C,9H 4C,9H 3G G522 SORGHUM     10E 10H 0 0 2C,9G 3C,8G 2C 0 0 0 0 0 0 0 5C,9H 3C,9H 5C,9H 3C,8H CHEAT     GRASS 9H 8G 0 0 7G 2G 5G 0 0 0 0 0 0 0 9H 9G 9G 5G USH11 SUGARBEET 9G 6G     6G 0 7G 4H 8G 4G 0 -- 0 0 0 0 4C,9G 3C,8G 4C,9G 8H VELVETLEAF 8H 3H 0 0     2G 0 0 0 0 0 0 0 0 0 8H 2C,2G 2C,3H 1C GIANT FOXTAIL 9H 3C,8G 0 0 2C 0     2G 0 2G 0 0 0 0 0 9H 7G 2C,3G 0 KLAGES BARLEY 8G 7G 0 0 6G 0 0 0 0 0 0 0     0 0 2C,9G 6G 4C,9G 0       CMPD 10 CMPD 11 CMPD 12 CMPD 13 CMPD 14 CMPD 15 CMPD 16 CMPD 17 CMPD     18 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 0 0 2G 0 5G 0 0 0 0 0 3C,9G 8G 5G 0 0 0 0 0 CULT     MORNINGLRY 3H 0 1H 0 0 0 0 0 0 0 9G 2C,9H 3C,7H 0 2C,3H 0 0 0 COCKLEBUR     0 0 4H 0 1H 0 0 0 0 0 8H 2H 1C,2G 0 0 0 -- 0 PURPLE NUTSEDGE 0 0 0 0 0 0     0 0 0 0 10E 9C 3G 0 8G 0 8G 0 LARGE CRABGRASS 0 0 0 0 0 0 0 0 0 0 9H 2G     2G 0 3G 0 0 0 BARNYARDGRASS 3G 0 2G 0 0 0 0 0 0 0 9H 4C,8H 3G 0 7G 0 2C     0 WILD OATS 2C,4G 0 7G 0 0 0 0 0 0 0 3C,7G 6G 2C,6G 6G 4G 0 7G 2G ERA     WHEAT 0 0 0 0 0 0 0 0 0 0 3C,9H 6G 7G 4G 2G 0 6G 2G G4646 CORN 0 0 2G 0     2G 0 0 0 0 0 4G 4G 3G 0 0 2G 0 0 WILLMS SOYBEANS 0 0 0 0 0 0 0 0 0 0 8H     3C,6H 3C,7H 0 2C,2H 0 0 0 RICE DRY SEEDED 5G 2G 2G 0 0 0 0 0 0 0 10H 10H     10H 2C,4G 9H 2G 8H 2G G522 SORGHUM 3C,8H 3C,7H 3C,5G 4G 0 0 0 0 0 0 10H     4C,9H 9H 4C,9H 9H 3C,8H 4C,9H 2C,7G CHEAT GRASS 7G 0 4G 0 0 0 0 0 0 0 9H     3C,9G 3C,8H 2C,7H 7G 0 7G 2G USH11 SUGARBEET 3C,3H 0 5H 0 3H 0 0 0 0 0     3C,9G 3C,9G 3C,8H 2C,3G 8G 5H 5H 0 VELVETLEAF 0 0 1H 0 0 0 0 0 0 0 3C,8G     3C,6H 2C,5G 0 3G 0 0 0 GIANT FOXTAIL 0 0 0 0 0 0 0 0 0 0 5C,9H 2C,8H 2C     0 2G 0 0 0 KLAGES BARLEY 0 0 2G 0 0 0 0 0 0 0 3C,8G 7G 2C,7G 2G 5G 0 3G     1C       CMPD 19 CMPD 20 CMPD 21 CMPD 22 CMPD 23 CMPD 24 CMPD 25 CMPD 26 CMPD     27 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01        PRSOL COKER COTTON 0 0 0 0 9G 8G 0 0 6G 3G 0 0 0 0 0 0 0 0 CULT     MORNINGLRY 0 0 0 0 9G 8G 2G 0 9G 2G 1C 0 1C,1H 0 0 0 0 0 COCKLEBUR 0 0     -- 0 9H 8G 0 0 8G 0 5G 0 -- 0 0 0 0 -- PURPLE NUTSEDGE 0 0 0 0 10E 5G 0     0 10E 7G 0 0 0 0 0 0 0 0 LARGE CRABGRASS 0 0 0 -- 9H 0 0 0 6G 0 0 0 0 --     0 -- 0 0 BARNYARDGRASS 2G 0 0 0 9H 9H 0 0 9H 3C,8H 0 0 0 0 0 0 0 0 WILD     OATS 0 0 0 0 3C,7H 6G 0 0 4G 0 0 0 0 0 0 0 0 0 ERA WHEAT 0 0 0 0 5C,9H     8H 0 0 5G 0 0 0 0 0 0 0 0 0 G4646 CORN 2G 0 0 0 1C,4G 2G 0 0 2G 0 0 0 0     0 0 0 0 0 WILLMS SOYBEANS 2G 0 0 0 9H 3C,6H 0 0 2G 0 0 0 0 0 0 0 0 0     RICE DRY SEEDED 0 0 0 0 10E 10H 0 0 10E 9H 0 0 0 0 0 0 0 0 G522 SORGHUM     0 0 0 0 10E 9H 3G 0 10E 10H 3G 0 2G 0 0 0 2C 0 CHEAT GRASS 2G 0 0 0 9H     9H 0 0 9H 7H 0 0 0 0 0 0 0 0 USH11 SUGARBEET 2H 0 0 0 9G 9G 3G -- 8G 3H     0 0 5G -- 0 0 3H 0 VELVETLEAF 0 0 0 0 7H 2G 2G 0 2G 0 0 0 2G 0 0 0 0 0     GIANT FOXTAIL 0 0 0 0 9H 9H 0 0 7H 3G 0 0 0 0 0 0 0 0 KLAGES BARLEY 0 0     0 0 9G 8G 0 0 4C,9G 2G 0 0 0 0 0 0 0 0       CMPD 28 CMPD 29 CMPD 30 CMPD 31 CMPD 32 CMPD 33 CMPD 34 CMPD 35  CMPD     36 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 8G 6G 5G 3G 0 0 2G 0 4G 0 0 0 8G 8G 4G -- 8G 4G     CULT MORNINGLRY 7H 7H 3G 0 3C,7G 2G 2G 0 2G 0 0 0 9G 8G 0 2C 7G 0     COCKLEBUR 1H -- 0 0 2C,3H 0 7G 0 0 0 -- 0 8H -- 0 0 2G 0 PURPLE NUTSEDGE     10E 3G 4G 0 0 0 0 0 0 0 0 0 10E 9G 0 0 9G 0 LARGE CRABGRASS 2C,8G 8G --     -- -- -- -- 0 0 0 0 0 4C,9H 10E 0 0 10E 8G BARNYARDGRASS 9H 2C,6G 2G 0 0     0 0 0 0 0 0 0 9H 3C,8H 0 0 9H 2G WILD OATS 3C,8G 2C,7G 3G 0 0 0 2G 0 5G     0 0 0 3C,8H 6G 0 0 0 4G ERA WHEAT 3C,9G 3C,8G 2G 0 0 0 4G 0 2G 0 0 0     4C,9H 8G 0 0 2G 3G G4646 CORN 2C,8G 3C,7G 2C,4G 0 2C 0 3G 0 0 0 0 0 9G     2C,4G 0 0 0 0 WILLMS SOYBEANS 3C,7H 3C,7H 3C,3H 2G 2C,2H 2H 4G 0 2G 0 0     0 9G 3C,6G 2G 2C 2C,4G 0 RICE DRY SEEDED 9H 9H 3C,6G 2C,3G 2G 2G 2G 0 0     0 0 0 10H 10H 3G 0 10E 2C,5G G522 SORGHUM 5C,9H 5C,9H 4C,5G 2G 2C 0 2G 0     0 0 0 0 9G 9G 2G 0 10E 3C,6H CHEAT GRASS 2C,8G 8G 3G 2G 0 0 0 0 2G 0 0 0     9H 6G 0 0 7G 2G USH11 SUGARBEET 4C,9G 1C 7G 5H 7G 2H 2H 0 2H 0 5H 3G 9G     7G 0 -- 7G 4G VELVETLEAF 7G 3G 2G 0 4G 0 0 0 0 0 3G 0 3C,8G 2C,8G 0 0     1C,3G 2C GIANT FOXTAIL 9H 7G 8G 0 5G 5G 2G 0 0 0 0 0 9H 9H 0 0 9H 4G     KLAGES BARLEY 2C,7G 8G 2C,6G 0 2C 0 0 0 0 0 0 0 3C,8G 8G 0 0 2G 0       CMPD 37 CMPD 38 CMPD 39 CMPD 40 CMPD 41 CMPD 42 CMPD 43 CMPD 44 CMPD     45 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 0 0 0 0 0 0 2C,5G 2G 0 0 0 0 0 0 0 0 0 0 CULT     MORNINGLRY 0 0 0 0 0 0 9H 7H 2C,7H 2C,5H 0 0 0 0 0 0 0 0 COCKLEBUR 0 0 0     0 0 0 8H 3H 2C,4H 3G 0 0 0 0 0 0 0 0 PURPLE NUTSEDGE 0 0 0 0 0 0 7G 7G 0     0 4G 0 0 0 0 0 0 0 LARGE CRABGRASS -- 0 0 -- -- -- 9G 4G 3G -- 4G -- 0 0     0 0 0 0 BARNYARDGRASS 0 0 0 0 0 0 5G 4G 7G 0 0 0 0 0 0 0 0 0 WILD OATS 0     0 0 0 0 0 3C,7G 3G 2C,6G 0 0 0 0 0 0 0 0 0 ERA WHEAT 0 0 0 0 0 0 8G 3G     2C,7G 0 0 0 0 0 0 0 0 0 G4646 CORN 0 0 0 0 0 0 3C,3G 3G 0 0 0 0 0 0 0 0     0 0 WILLMS SOYBEANS 0 0 0 0 0 0 3C,3H 2H 2C,2G 0 2G 0 0 0 0 0 0 0 RICE     DRY SEEDED 0 0 0 0 0 0 9H 5G 3C,5G 0 0 0 0 0 0 0 0 0 G522 SORGHUM 0 0 0     0 0 0 5C,9G 3C,7H 3C,5G 2C 3C,3G 0 0 0 0 0 0 0 CHEAT GRASS 0 0 0 0 0 0     8G 5G 7G 0 0 0 0 0 0 0 0 0 USH11 SUGARBEET 0 0 0 0 -- 0 3C,8G 6H 3C,5G     3G 0 0 0 0 0 0 0 0 VELVETLEAF 0 0 0 0 0 0 7H 1C 7G 0 0 0 0 0 0 0 0 0     GIANT FOXTAIL 0 0 -- -- 0 0 9H 0 9H 5G 3G 0 2G 0 0 0 0 0 KLAGES BARLEY 0     0 0 0 0 0 2C,8G 7G 7G 2G 3G 0 0 0 0 0 0 0       CMPD 46 CMPD 47 CMPD 48 CMPD 49 CMPD 50 CMPD 51 CMPD 52 CMPD 53 CMPD     54 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 3C,5H 2C,4G 0 0 1C 0 0 0 0 0 0 -- 2G 0 0 0 0 0 CULT     MORNINGLRY 9H 1C 0 0 0 0 0 0 0 0 1H 0 1H 1H 4H 0 0 0 COCKLEBUR 9H 0 0 0     1H -- 0 0 0 0 0 0 -- 0 2H 0 4G 0 PURPLE NUTSEDGE 10E 10E 4G 0 0 -- 0 0     -- 0 0 0 0 0 0 0 0 0 LARGE CRABGRASS 9H 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0     0 BARNYARDGRASS 2C,9H 3C,7H 0 0 0 0 0 0 0 0 0 0 2H 0 4G 0 0 0 WILD OATS     2C,4G 4G 0 0 0 0 0 0 0 0 0 0 0 0 6G 0 0 0 ERA WHEAT 9H 7G 0 0 0 0 0 0 0     0 0 0 0 0 5G 0 0 0 G4646 CORN 5G 0 0 0 2G 0 0 0 0 0 0 0 0 0 2G 0 0 0     WILLMS SOYBEANS 3C,9H 1C,2H 0 0 2G 0 0 0 0 0 0 0 0 0 0 0 0 0 RICE DRY     SEEDED 9H4C,8H 0 0 3C,9H 2C,3H 0 0 0 0 0 0 0 0 6G 0 0 0 G522 SORGHUM 9H     3C,9H 0 0 2C,8H 2C,4G 0 0 0 0 0 0 2G 0 2C,6G 0 0 0 CHEAT GRASS 9H 7G 0 0     2G 0 0 0 0 0 0 0 0 0 7G 0 0 0 USH11 SUGARBEET 4C,8G 3H 4H 0 2C,4H 2H 0 0     0 0 0 0 1H 0 6G 0 0 0 VELVETLEAF3C,8G 1C,4H 0 0 0 0 0 0 0 0 0 0 1H 0 0 0     2G 0 GIANT FOXTAIL 3C,9H 8G 0 0 3G 0 0 0 3G 0 0 0 2G 0 3G 0 0 0 KLAGES     BARLEY 2C,9H 2C,9H 0 0 5G 0 0 0 0 0 0 0 0 0 8G 0 0 0       CMPD 55 CMPD 56 CMPD 57 CMPD 58 CMPD 59 CMPD 60 CMPD 61 CMPD 62 CMPD     63 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 0 0 0 0 0 0 0 0 0 0 9G 2G 0 0 0 0 0 0 CULT MORNINGLR     Y 0 -- 0 0 0 0 0 0 0 0 9G 5G 1H 0 0 0 0 0 COCKLEBUR 0 0 3G 0 0 0 0 0 0 0     9H 3C,6G 0 0 0 0 0 -- PURPLE NUTSEDGE 0 0 0 0 0 0 0 -- 0 -- 10E 0 0 0 0     0 4G -- LARGE CRABGRASS 0 0 0 0 0 0 0 0 0 0 3C,7G 0 0 0 0 0 0 0 BARNYARDG     RASS 0 0 0 0 0 0 0 0 0 0 9H 3C,6G 0 0 0 0 0 0 WILD OATS 0 0 0 0 0 0 0 0     0 0 2C,8G 3C,7G 0 0 0 0 0 0 ERA WHEAT 0 0 0 0 0 0 0 0 0 0 9H 2C,9H 0 0 0     0 0 0 G4646 CORN 0 0 0 0 0 0 0 0 0 0 2C,4G 0 2C,2G 0 0 0 0 0 WILLMS     SOYBEANS 0 0 0 0 0 0 0 0 0 0 9H 3C,6G 2C,2H 0 0 0 0 0 RICE DRY SEEDED 0     0 0 0 0 0 0 0 0 0 10E 8H 0 0 0 0 2G 0 G522 SORGHUM 0 0 0 0 0 0 0 0 0 0     10H 3C,8H 0 0 0 0 0 0 CHEAT GRASS 0 0 0 0 0 0 0 0 0 0 9G 6G 0 0 0 0 0 0     USH11 SUGARBEET 0 0 0 0 0 0 0 0 0 0 9G 8G 4G 0 0 0 2H 0 VELVETLEAF 0 0     3G 0 0 0 0 0 0 0 4C,8G 0 3H 0 0 0 4G 1H GIANT FOXTAIL 0 0 0 0 0 0 0 0 0     0 3C,7G 3G 0 0 0 0 0 0 KLAGES BARLEY 0 0 0 0 0 0 0 0 0 0 9G 8G 0 0 0 0 0       CMPD 64 CMPD 65 CMPD 66 CMPD 67 CMPD 68 CMPD 69 CMPD 70 CMPD 71 CMPD     72 RATE = KG/HA 0.05 0.01 0.05 0.01  0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 9G 8G 9G 9G 8G 2G 8G 9G 9G 5G 7G 2G 9G 8G 2C,9G 3G     2C,7H 2C,6G CULT MORNINGLRY 9G 9G 9H 9H 9G 9G 9G 9H 9G 7G 6G 4G 9G 7G 9G     4G 2C,9G 9H COCKLEBUR 9H 9H 9H 9H 9G 8G 8G 4G 8H 4G 2H 4G 9H 3C,6H 8H     3C,6H 3C,9H 3H PURPLE NUTSEDGE 10E 5G 10E 9G 10E 4C,9G 10E 10E 10E 9G 0     0 10E 9G 10E 0 10E 10E LARGE CRABGRASS 3C,8G 3G 5C,9G 3C,8G 6C,9H 3C,6G     5C,9H 5C,9G 9C 3C,8G 3C,7G 0 4C,8G 5G 2C,8G 4G 2C,7G 2G BARNYARDGRASS 9H     3C,6G 9H 9H 9H 6G 9H 9H 9H 5G 5G 0 9H 8H 9H 9H 9H 8H WILD OATS 3C,7G     2C,4G 4C,8G 8G 3C,7G 2C,6G 4C,8G 3C,7G 4C,9G 3C,6G 2C,6G 6G 3C,7G 5G     4C,8G 2G 3C,8G 2G ERA WHEAT 3C,7G 0 4C,9G 9G 3C,9G 0 9H 3C,9G 9H 3C,7G     8G 6G 8H 4G 9H 0 8G 3G G4646 CORN 3C,9H 2C,4G 3C,9H 3C,9G 3C,9G 3C,9H 9H     3C,9H 3C,9G 3C,8G 3C,8G 5G 9H 9G 2C,9H 2C,4G 9G 3C,7H WILLMS SOYBEANS 9H     3C,8H 9H 9H 9H 7G 9H 3C,8G 9H 9H 8G 7G 9H 3C,7H 9H 3C,7H 3C,8H 3C,5G     RICE DRY SEEDED 10E 9H 10E 9H 10E 9H 10E 10E 10E 9H 8G 4G 10E 8G 10E     2C,5G 10E 9H G522 SORGHUM 9H 3C,8G 10H 3C,9H 9H 5G 10C 4C,9H 10E 3C,9H     6G 3G 9H 2C,9G 9H 9H 4C,9H 3C,9H CHEAT GRASS 8G 2G 9H 10E 9H 8G 10E 8G     10E 9H 8G 3G 4C,9G 5G 9H 2C,7G 9H 7G USH11 SUGARBEET 9G 9G 9G 3C,9G 8G     8G 9G 9G 5C,9G 7H 3H 4G 4C,9G 9G 3C,9G 3C,9G 4C,9G 3C,8H VELVETLEAF     4C,9G 3C,6G 9G 9G 7G 7G 4C,8G 5G 9G 2G 2G 0 5C,9G 5C,9G 3C,6G 2G 3C,7H     3G GIANT FOXTAIL 6G 0 9H 9H 10H 3C,9H 9H 6G 10H3C,8G 9H 3G 9H 3C,7G 9H     2C,7G 3C,8H 3G KLAGES BARLEY 9G 4G 5C,9G 3C,9G 5C,9H 3G 3C,9H 3C,9G     5C,9G 4C,9G 3C,9G 2G 9G 2C,4G 3C,7G 2C,4G 2C,9G 2G       CMPD 73 CMPD 74 CMPD 75 CMPD 76 CMPD 77 CMPD 78 CMPD 79 CMPD 80 CMPD     81 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 3C,7H 2C,2G 2G 0 0 0 0 0 0 0 0 0 0 0 0 0 8G 0 CULT     MORNINGLRY 9G 8H 0 0 0 0 0 0 0 0 0 0 0 0 0 0 9G 5G COCKLEBUR 3C,8H 3C,2H     0 0 0 0 0 0 0 0 0 0 0 -- 0 0 9H 3C,9H PURPLE NUTSEDGE 10E 3C,9G 0 0 0 0     0 0 0 0 0 0 0 0 0 0 10E 0 LARGE CRABGRASS 4C,9G 3C,5G 7G 0 9H 2G 0 0 0 0     0 0 0 0 0 0 5G 2G BARNYARDGRASS 9H 9H 3G 0 3C,5G 2G 0 0 0 0 0 0 0 0 0 0     9H 8H WILD OATS 3C,8H 3C,8H 6G 0 7G 2G 0 0 0 0 0 0 0 0 0 0 2G 0 ERA     WHEAT 3C,9H 2C,9H 7G 0 8G 3G 0 0 0 0 0 0 0 0 0 0 2G 0 G4646 CORN 3C,9H     3C,7H 3C,7G 2C,5G 9G 6G 0 0 0 0 0 0 0 0 0 0 5C,9H 7G WILLMS SOYBEANS     3C,9H 3C,5H 2G 0 0 0 0 0 0 0 0 0 0 0 0 0 5G 2C,2H RICE DRY SEEDED 10E 9H     7G 0 8G 7G 0 0 0 0 0 0 0 0 0 0 10E 9H G522 SORGHUM 9H 3C,9G 3C,8H 2C,6G     3C,9G 3C,8H 0 0 0 0 0 0 0 0 0 0 5C,9H 3C,9H CHEAT GRASS 3C,9H 9H 7G 0 8G     3G 0 0 0 0 0 0 0 0 0 0 5G 0 USH11 SUGARBEET 4C,9G 3C,7H 2H 0 0 2H 0 0 0     0 0 -- 0 -- 0 0 9G 8G VELVETLEAF 3C,8H 5G 0 0 4G 0 0 0 0 0 0 0 0 0 0 0     5H 3C,5G GIANT FOXTAIL 9H 3C,7H 7G 2G 3C,8H 3G 0 0 0 0 0 0 0 0 0 0 2C,9G     3C,8G KLAGES BARLEY 9G 3C,8H 3C,7G 0 9G 2G 0 0 0 0 0 0 0 0 0 0 2C,9G     3C,8G       CMPD 82 CMPD 83 CMPD 84 CMPD 85 CMPD 86 CMPD 87 CMPD 88 CMPD 89 CMPD     90 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 2G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 CULT MORNINGLRY      5G 0 0 0 0 0 0 0 2C,6G 0 0 0 0 0 0 0 0 0 COCKLEBUR 3C,3G 0 3C,8H 0 1C 0     0 0 3G 2G 0 0 0 0 1H 0 0 0 PURPLE NUTSEDGE 10E 0 0 0 0 0 0 0 5G 0 0 0 0     0 0 0 0 0 LARGE CRABGRASS 3G 0 0 0 -- 0 0 0 3C,7G 0 0 0 0 0 0 0 0 0     BARNYARDGRASS 7G 0 0 0 0 0 7G 0 9H 0 0 0 0 0 0 0 0 0 WILD OATS 0 0 0 0 0     0 0 0 0 0 0 0 0 0 0 0 0 0 ERA WHEAT 0 0 0 0 0 0 0 0 2G 0 0 0 0 0 0 0 0 0     G4646 CORN 6G 2G 3C,7G 0 3C,9G 2G 3C,9G 2G 3C,6G 0 0 0 0 0 0 0 0 0     WILLMS SOYBEANS 2C,3G 0 1H 0 2G 0 0 0 3C,5H 0 0 0 0 0 0 0 0 0 RICE DRY     SEEDED 10H 4C,9H 10H 7H 9H 4G 9H 4G 8G 0 0 0 0 0 0 0 0 0 G522 SORGHUM 9H     4C,9G 10H 5G 2C,9G 6G 9H 5G 9G 2C 0 0 0 0 0 0 0 0 CHEAT GRASS 3G 0 0 0 0     0 0 0 -- -- -- -- -- -- -- -- -- -- USH11 SUGARBEET 7G 5G 6G 2G 3G 2H 3G     2G 9G 5G 0 0 0 0 0 0 0 0 VELVETLEAF 3G 0 1H 0 0 0 2G 0 7G 5G 0 0 0 0 0 0     0 0 GIANT FOXTAIL 3G 0 3G 0 3G 0 7G 2G 5G 0 0 0 0 0 0 0 0 0 KLAGES     BARLEY 7G 2G 2C,7G 0 3G 0 2G 0 0 0 0 0 0 0 0 0 0 0 DOWNY BROME       --     -- 7G 0 0 0 0 0 0 0 0 0       CMPD 91 CMPD 92 CMPD 93 CMPD 94 CMPD 95 CMPD 96 CMPD 97 CMPD 98 CMPD     99 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 0 0 8G 8G 3G 1C 0 0 0 0 2C,8G 5G 0 0 0 0 2G 0 CULT     MORNINGLRY 0 0 9G 7G 2C,5H 1C 0 0 0 0 9G 0 0 0 0 0 2C 0 COCKLEBUR 0 0 --     5G 3C,8H 2H 0 0 0 -- 8H 2C,6H -- 0 0 0 2G 0 PURPLE NUTSEDGE 0 0 10E 9G     10E 10E 0 0 0 0 9G 8G 0 0 0 0 10E 0 LARGE CRABGRASS 0 0 3C,8G 2G 3C,5G 0     0 0 0 0 10E 3C,6G 0 0 0 0 0 0 BARNYARDGRASS 0 0 9H 3C,8H 3C,8H 2C,7G 0 0     0 0 4C,9H 4G 0 0 0 0 0 0 WILD OATS 0 0 2C,7G 5G 5G 0 0 0 0 0 7G 2G 0 0 0     0 0 0 ERA WHEAT 0 0 3C,9H 3C,8H 5G 0 0 0 0 0 9H 7G 0 0 0 0 0 0 G4646     CORN 0 0 2C,6G 3G 0 0 0 0 0 0 2C,7G 3G 0 0 0 0 0 0 WILLMS SOYBEANS 0 0     3C,9H 3C,7H 3G 2H 0 0 0 0 9H 8G 0 0 0 0 0 0 RICE DRY SEEDED 0 0 10E 10E     10E 9H 0 0 0 0 4C,9H 3C,8H 0 0 0 0 0 0 G522 SORGHUM 0 0 10H 6C,9H 7C,9H     9H 0 0 0 0 9H 9H 0 0 0 0 2C,3G 0 CHEAT GRASS -- -- 9G 9G 9H 6G 0 0 0 0     8G 2G 0 0 0 0 0 0 USH11 SUGARBEET 0 0 5C,9G 9G 4C,8H 6H 2G 0 0 0 5G 5G 0     0 0 0 8G 0 VELVETLEAF 0 0 3C,8G 4G 0 0 0 0 0 0 3C,8G 2G 0 0 0 0 3G 0     GIANT FOXTAIL 0 0 9H 2C,8G 3C,5G 0 0 0 0 0 9H 2C,9G 0 0 0 0 2G 0 KLAGES     BARLEY 0 0 8G 7G 7G 0 0 0 0 0 8G 2C,2G 0 0 0 0 0 0 DOWNY BROME 0 0 --     --   CMPD 100 CMPD 101 CMPD 102 CMPD 103 CMPD 104 CMPD 105 CMPD 106 CMPD     107 CMPD 108 RATE = KG/HA 0.05 0.01  0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 8H 2C,6G 5G 2C,3G 2G 0 0 0 0 0 0 0 2G 0 0 0 0 0     CULT MORNINGLRY 9G 9G 8G 7H 1C 0 0 0 0 0 0 0 1C 0 0 0 0 0 COCKLEBUR 9H     3C,7H -- 2C 1H 0 0 0 0 0 0 0 2G 0 0 0 0 0 PURPLE NUTSEDGE 10E 9G 10E 5G     0 0 -- 0 0 0 0 0 10E 0 0 0 0 0 LARGE CRABGRASS 6G 4G 2C,5G 2C 0 0 0 0 0     0 0 0 3G 0 0 0 0 0 BARNYARDGRASS 9H 5H 9H 6G 0 0 0 0 0 0 0 0 7H 0 0 0 0     0 WILD OATS 3C,8H 6G 5G 0 0 0 0 0 0 0 0 0 2C,3G 0 0 0 0 0 ERA WHEAT 9H     9H 7G 0 0 0 0 0 0 0 0 0 6G 0 0 0 0 0 G4646 CORN 2G 2G 2G 0 0 0 0 0 0 0 0     0 2C,4G 0 0 0 0 0 WILLMS SOYBEANS 3C,4H 3C,6H 4G 2H 2G 0 0 0 0 0 0 0 1C     0 0 0 0 0 RICE DRY SEEDED 10E 10E 9H 8H 0 0 0 0 0 0 0 0 8H 0 0 0 0 0     G522 SORGHUM 9H 9H 9H 4C,9H 0 0 0 0 0 0 0 0 2C,8H 0 0 0 0 0 CHEAT GRASS     8H 7H 8G 5G 0 0 0 0 0 0 0 0 4G 0 0 0 0 0 USH11 SUGARBEET 9G 9G 9G 5G 5G     0 0 0 0 0 3H 0 2G 0 0 0 0 0 VELVETLEAF 3C,8H 3C,5H 4G 0 2G 0 0 0 0 0 0     0 6G 0 0 0 0 0 GIANT FOXTAIL 9H 9H 3C,8H 5G 0 0 0 0 0 0 0 0 9H 0 0 0 0 0     KLAGES BARLEY 9G 8G 9G 7G 0 0 0 0 0 0 0 0 5G 0 0 0 0 0       CMPD 109 CMPD 110 CMPD 111 CMPD 112 CMPD 113 CMPD 114 CMPD 115 CMPD     116 CMPD 117 RATE = KG/HA 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05     0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01       PRSOL COKER COTTON 0 0 1H 0 0 0 7G 2G 8G 4G 0 0 0 0 9G 8G 9G 2C,6G     CULT MORNINGLRY 0 0 3G 0 0 0 9G 3C,4G 2C,2H 0 0 0 0 0 9G 9G 9G 9G     COCKLEBUR 0 0 2C 0 0 0 8H 8H 5H 1C 2G 0 2G 3G 9H 9H 8H 3C,7H PURPLE     NUTSEDGE 0 0 10E 0 0 0 10E 10E 9G 0 0 0 0 0 9G 9G 5C,9G 9G LARGE     CRABGRASS 0 0 7G 4G 0 0 0 0 0 0 0 0 7G 0 5G 2G 2C,7G 6G BARNYARDGRASS 0     0 3C,5G 3G 0 0 8H 7H 8H 0 0 0 0 0 9H 4H 9H 2C,5G WILD OATS 0 0 0 0 0 0     2G 0 0 0 0 0 0 0 7G 2G 2C,7G 2G ERA WHEAT 0 0 5G 0 0 0 3G 3G 2G 0 0 0 0     0 4C,9G 5G 3C,9H 7G G4646 CORN 0 0 3C,7G 2C,5G 0 0 9G 8G 2C,7G 0 0 0     2C,5G 0 3C,9G 3C,7G 9G 3C,8H WILLMS SOYBEANS 0 0 1H 0 0 0 3C,7G 1C,1H 1C     0 0 0 0 0 4C,8H 3C,8G 4C,9H 3C,6G RICE DRY SEEDED 0 0 6G 2G 0 0 9H 8H 8G     6G 0 0 7G 0 10E 3C,8G 10H 4C,8H G522 SORGHUM 0 0 10H 3C,3G 0 0 9H 7H 8G     8G 0 0 7G 0 9H 3C,7G 3C,9H 3C,9H CHEAT GRASS 0 0 4G 0 0 0 -- -- -- -- --     -- -- -- 4C,8G 7G 3C,8H 8G USH11 SUGARBEET 0 0 6G 4H 0 0 9G 2H 8G 4H 3G     0 3G 0 5C,9G 9G 4C,9G 3C,9G VELVETLEAF 3G 0 1H 0 0 0 7H 5H 3H 0 0 0 0 0     3C,9G 9G 4C,9G 4C,9G GIANT FOXTAIL 0 0 2C,8G 4G 0 0 4G 0 0 0 0 0 5G 0     3C,7H 2H 9H 3C,8H KLAGES BARLEY 0 0 3C,7G 2G 0 0 7G 2C,3G 2C,5G 0 0 0 7G     0 2C,9G 2C,6G 8G 6G DOWNY BROME -- -- -- -- -- -- 9H 7G 10C 3G 0 0 5G 0     -- --       CMPD 118 CMPD 119 CMPD 120 CMPD 121 RATE = KG/HA 0.05 0.01 0.05 0.01     0.05 0.01 0.05 0.01       PRSOL COKER COTTON 9G 9G 9G 8G 4C,8G 5G 9G 2C,6G CULT MORNINGLRY 9G 9G     8G 8G 9G 2C,5G 9G 9G COCKLEBUR 8H -- 10C 9H 8H 3C,6H 9H 9H PURPLE     NUTSEDGE 10E 7G 10E 10E 5G 2G 7G 7G LARGE CRABGRASS 7G 4G 3C,9H 9G 4C,9G     2C,4G 4C,8G 2C,5G BARNYARDGRASS 9H 2C,7H 9H 3C,8H 5C,9H 2G 4C,9H 3C,7H     WILD OATS 2G 0 3C,8G 6G 5G 0 4C,8G 2G ERA WHEAT 2C,8H 8G 5C,9H 8G 7G 0     3C,9H 4G G4646 CORN 9G 3C,8G 9G 3C,9H 2C,9G 2C,6G 9G 3C,7H WILLMS     SOYBEANS 2C,9H 3C,7H 9H 9H 9H 4C,8H 9H 4C,8H RICE DRY SEEDED 10H 9H 10E     10H 10H 3C,7H 10H 4C,8H G522 SORGHUM 9H 9H 5C,9H 4C,9H 4C,8H 3C,6H 3C,9H     5C,8H CHEAT GRASS 8G 8G 9H 8H 3C,8G 0 4C,8H 3C,8H USH11 SUGARBEET 4C,9G     4C,9G 5C,9G 7G 5C,9G 2C,4G 5C,9G 4C,9G VELVETLEAF 4C,9G 3C,7G 4C,9G     3C,9G 9C 2G 4C,8G 3C,3G GIANT FOXTAIL 8G 3C,7H 9H 8G 7G 0 9H 7G KLAGES     BARLEY 8G 8G 9G 9G 2C,8G 5G 9G 7G

It is noted that a few compounds such as compounds 6, 19, 20, 26, 32,37-39, 44, 49, 54-59, 76-78 and 88 show little or no herbicidal activityat the rate tested. It is thought they would show more herbicidalactivity at higher rates.

Test B Postemergence

Three round pans (25 cm diameter by 12.5 cm deep) were filled withSassafras sandy loam soil. One pan was planted with nutsedge (Cyperusrotundus) tubers, crabgrass (Digitaria sanguinalis), sicklepod (Cassiaobtusifolia), jimsonweed (Datura stramonium), velvetleaf (Abutilontheophrasti), chickweed (Stellaria media), lambsquarters (Chenopodiumalbum), rice (Oryza satira, variety California Rice Coop. M101) andteaweed (Sida spinosa). The second pot was planted with green foxtail(Setaria viridis), cocklebur (Xanthium pensylvanicum), morningglory(Ipomoea coccinea, variety Scarlet O'Hara), cotton (Gossypium hirsutum,variety Coker 315), johnsongrass (Sorghum halepense), barnyardgrass(Echinochloa crus-galli), corn (Zea mays, variety Funk G4646), soybeans(Glycine max, variety Williams) and giant foxtail (Setaria faberi). Thethird pot was planted with wheat (Triticum aestivum, variety Eraspring), barley (Hordeum vulgare, variety Klages spring), wild buckwheat(Polgonum convolvulus), cheatgrass (Bromus secalinus), sugarbeet (Betavulgaris, variety Union Sugarbeet Co. USH11), wild oats (Avena fatua),field violet (Viola arvensis), blackgrass (Alopecurus myosuroides), andrape (Brassica napus, variety Altex). The plants were grown forapproximately fourteen days, then sprayed postemergence with thechemicals dissolved in a non-phytotoxic solvent.

Preemergence

Three round pans (25 cm diameter by 12.5 cm deep) were filled withSassafras sandy loam soil. One pan was planted with nutsedge tubers,crabgrass, sicklepod, jimsonweed, velvetleaf, chickweed, lambsquarters,rice and teaweed. The second pot was planted with green foxtail,cocklebur, morningglory, cotton, johnsongrass, barnyardgrass, corn,soybean and giant foxtail. The third pot was planted with wheat, barley,wild buckwheat, cheatgrass, sugarbeet, wild oat, field violet,blackgrass and rape. The three pans were sprayed preemergence with thechemicals dissolved in a non-phytotoxic solvent.

Treated plants and controls were maintained in the greenhouse for 24days, then all treated plants were compared to controls and visuallyrated for plant response.

Response ratings are based on a scale of 0 to 100 where 0=no effect and100=complete control. A dash (--) response means no test.

Response ratings are contained in Table B.

                  TABLE B                                                         ______________________________________                                                   Cmpd 1                                                             RATE (g/ha)  1        4      16     62   250                                  ______________________________________                                        PREEMERGENCE                                                                  Barley       20       30     80     80   90                                   Barnyardgrass                                                                               0       20     100    95   95                                   Blackgrass    0       20     80     85   100                                  Cheatgrass   30       70     90     100  100                                  Chickweed    --       --     --     --   --                                   Cocklebur     0        0     30     85   90                                   Corn          0        0      0      0   10                                   Cotton        0       10     85     85   90                                   Crabgrass     0        0     40     50   75                                   Field violet --       --     --     --   --                                   Giant foxtail                                                                              20       20     80     85   90                                   Green foxtail                                                                              20       90     95     100  99                                   Jimsonweed   --        0     --     50   --                                   Johnsongrass 60       85     90     100  100                                  Lambsquarters                                                                               0        0     50     70   80                                   Morningglory  0        0     20     80   95                                   Nutsedge     20       30     80     90   95                                   Rape          0       50     80     90   95                                   Rice         20       85     90     95   100                                  Sicklepod    --        0     --     --   --                                   Soybean       0        0      0     10   30                                   Sugarbeet    20       60     70     80   90                                   Teaweed      --       --     30     80   80                                   Velvetleaf    0       20     30     40   70                                   Wheat         0       20     30     80   90                                   Wild buckwheat                                                                              0       50     70     80   90                                   Wild oat     10       20     30     60   70                                   ______________________________________                                                     Cmpd 21                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        PREEMERGENCE                                                                  Barley         30     50        80   90                                       Barnyardgrass  30     60        90   100                                      Blackgrass     60     70        80   90                                       Cheatgrass     30     70        100  100                                      Chickweed      --     --        --   --                                       Cocklebur       0     30        50   70                                       Corn            0      0         0    0                                       Cotton          0     30        50   80                                       Crabgrass      30     50        70   90                                       Field violet   30     50        70   90                                       Giant foxtail  30     70        90   100                                      Green foxtail  30     70        100  100                                      Jimsonweed     60     70        80   90                                       Johnsongrass   50     70        80   90                                       Lambsquarters  50     60        70   90                                       Morningglory    0     30        60   90                                       Nutsedge        0     30        80   100                                      Rape           70     90        100  100                                      Rice           60     100       100  100                                      Sicklepod      --     --        --   --                                       Soybean         0      0        30   90                                       Sugarbeet      30     60        90   100                                      Teaweed        30     50        70   90                                       Velvetleaf     30     50        70   90                                       Wheat           0     30        60   90                                       Wild buckwheat 70     80        90   90                                       Wild oat        0      0        30   80                                       ______________________________________                                                     Cmpd 46                                                          RATE (g/ha)    4      16        62   250                                      ______________________________________                                        PREEMERGENCE                                                                  Barley         20     40        60   80                                       Barnyardgrass  60     90        100  100                                      Blackgrass     50     70        80   90                                       Cheatgrass     60     70        80   90                                       Chickweed      30     50        70   90                                       Cocklebur       0     30        50   70                                       Corn            0      0         0   30                                       Cotton          0     30        40   60                                       Crabgrass       0     30        50   70                                       Field violet   --     --        --   --                                       Giant foxtail  50     80        90   100                                      Green foxtail  30     50        80   100                                      Jimsonweed      0     30        60   90                                       Johnsongrass   50     70        80   90                                       Lambsquarters  30     50        80   90                                       Morningglory   30     50        70   90                                       Nutsedge       30     60        90   100                                      Rape           50     70        90   100                                      Rice           80     90        100  100                                      Sicklepod      30     60        90   100                                      Soybean         0      0        70   --                                       Sugarbeet      70     90        100  --                                       Teaweed         0     30        50   80                                       Velvetleaf     30     60        90   100                                      Wheat          30     50        70   80                                       Wild buckwheat 30     50        70   90                                       Wild oat        0     30        40   60                                       ______________________________________                                                     Cmpd 60                                                          RATE (g/ha)    4      16        62   250                                      ______________________________________                                        PREEMERGENCE                                                                  Barley         20     30        30   90                                       Barnyardgrass  20     100       100  100                                      Blackgrass     70     80        100  100                                      Cheatgrass     30     70        100  100                                      Chickweed      60     100       100  100                                      Cocklebur       0     50        60   90                                       Corn            0     20        30   40                                       Cotton          0     50        90   90                                       Crabgrass      60     60        70   80                                       Field violet   --     --        --   --                                       Giant foxtail  --     --        --   --                                       Green foxtail   0     70        100  100                                      Jimsonweed      0     50        70   80                                       Johnsongrass   70     80        100  100                                      Lambsquarters  30     50        90   100                                      Morningglory   20     80        90   100                                      Nutsedge        0     80        90   100                                      Rape           80     90        90   100                                      Rice           90     90        100  100                                      Sicklepod      50     80        90   90                                       Soybean        30     60        90   100                                      Sugarbeet      80     90        90   90                                       Teaweed        50     70        90   90                                       Velvetleaf     30     40        80   100                                      Wheat          30     40        60   90                                       Wild buckwheat 50     70        80   90                                       Wild oat        0     30        50   70                                       ______________________________________                                                     Cmpd 64                                                          RATE (g/ha)    4      16        62   250                                      ______________________________________                                        PREEMERGENCE                                                                  Barley          0     30        60   90                                       Barnyardgrass  30     50        70   90                                       Blackgrass     30     70        80   90                                       Cheatgrass     50     70        80   90                                       Chickweed      30     50        70   90                                       Cocklebur      50     70        80   90                                       Corn            0     30        60   90                                       Cotton         30     50        70   90                                       Crabgrass       0     30        50   70                                       Field violet   --     --        --   --                                       Giant foxtail   0     50        70   90                                       Green foxtail  30     50        70   90                                       Jimsonweed     30     50        70   90                                       Johnsongrass   30     50        70   90                                       Lambsquarters  30     50        70   90                                       Morningglory   50     80        90   100                                      Nutsedge       80     90        100  100                                      Rape           80     100       100  100                                      Rice           50     70        100  100                                      Sicklepod      30     50        70   90                                       Soybean        30     60        80   90                                       Sugarbeet      80     90        100  100                                      Teaweed        30     50        70   90                                       Velvetleaf     50     70        90   100                                      Wheat          30     50        70   90                                       Wild buckwheat 70     80        90   95                                       Wild oat        0     30        50   70                                       ______________________________________                                                     Cmpd 65                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        PREEMERGENCE                                                                  Barley         20     40        80   100                                      Barnyardgrass   0     30        40   50                                       Blackgrass     40     50        90   100                                      Cheatgrass     70     80        100  100                                      Chickweed      70     90        100  100                                      Cocklebur       0     20        90   100                                      Corn            0      0        90   90                                       Cotton          0     20        80   100                                      Crabgrass      20     60        90   90                                       Field violet   --     --        --   --                                       Giant foxtail   0     20        100  100                                      Green foxtail   0     20        100  100                                      Jimsonweed      0     30        100  100                                      Johnsongrass    0     30        90   90                                       Lambsquarters  20     40        100  100                                      Morningglory    0     30        100  100                                      Nutsedge        0     30        90   90                                       Rape           70     100       100  100                                      Rice            0     20        100  100                                      Sicklepod       0     50        90   100                                      Soybean         0      0        30   50                                       Sugarbeet      70     90        100  100                                      Teaweed        20     50        100  100                                      Velvetleaf      0     20        80   90                                       Wheat           0     60        80   100                                      Wild buckwheat 80     100       100  100                                      Wild oat       20     40        80   100                                      ______________________________________                                                     Cmpd 66                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        PREEMERGENCE                                                                  Barley          0     30        60   90                                       Barnyardgrass   0      0        20   30                                       Blackgrass     30     50        90   100                                      Cheatgrass     60     70        100  100                                      Chickweed      70     80        90   100                                      Cocklebur       0      0        20   80                                       Corn            0      0        50   70                                       Cotton          0      0         0    0                                       Crabgrass      20     70        100  100                                      Field violet   --     --        --   --                                       Giant foxtail  20     40        70   90                                       Green foxtail   0     20        90   100                                      Jimsonweed     20     20        40   80                                       Johnsongrass    0      0        30   70                                       Lambsquarters   0      0        20   80                                       Morningglory    0     20        90   90                                       Nutsedge        0     20        40   80                                       Rape           40     60        90   100                                      Rice            0     20        60   100                                      Sicklepod      20     40        80   100                                      Soybean         0      0        30   80                                       Sugarbeet      40     60        100  100                                      Teaweed        20     30        90   90                                       Velvetleaf      0      0        40   60                                       Wheat           0     30        90   100                                      Wild buckwheat  0     40        100  100                                      Wild oat       20     30        40   90                                       ______________________________________                                                     Cmpd 67                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        PREEMERGENCE                                                                  Barley          0     20        70   100                                      Barnyardgrass   0     20        100  100                                      Blackgrass     30     50        80   90                                       Cheatgrass     30     70        80   100                                      Chickweed      30     70        80   90                                       Cocklebur       0     20        70   80                                       Corn            0     20        80   100                                      Cotton         --      0        20   90                                       Crabgrass      30     70        100  100                                      Field violet   --     --        --   --                                       Giant foxtail  20     40        100  100                                      Green foxtail   0     20        90   100                                      Jimsonweed      0     40        100  100                                      Johnsongrass    0     30        100  100                                      Lambsquarters   0     30        90   100                                      Morningglory    0     20        30   100                                      Nutsedge       20     60        100  100                                      Rape           30     70        100  100                                      Rice           20     50        100  100                                      Sicklepod       0     20        30   40                                       Soybean         0      0        40   80                                       Sugarbeet      60     70        100  100                                      Teaweed         0     20        70   80                                       Velvetleaf      0     30        70   100                                      Wheat           0     20        50   90                                       Wild buckwheat 60     90        100  100                                      Wild oat        0     20        30   40                                       ______________________________________                                                     Cmpd 68                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        PREEMERGENCE                                                                  Barley          0     40        80   90                                       Barnyardgrass  20     30        60   80                                       Blackgrass     30     50        80   90                                       Cheatgrass     30     40        100  100                                      Chickweed      40     60        70   80                                       Cocklebur       0     20        30   40                                       Corn            0      0         0   40                                       Cotton          0      0        20   40                                       Crabgrass       0     40        100  100                                      Field violet   --     --        --   --                                       Giant foxtail  20     40        90   100                                      Green foxtail   0     30        90   100                                      Jimsonweed      0     30        70   90                                       Johnsongrass   20     30        90   90                                       Lambsquarters   0     30        70   90                                       Morningglory    0     30        50   80                                       Nutsedge        0     30        100  100                                      Rape           30     70        100  100                                      Rice            0     30        100  100                                      Sicklepod       0     30        80   90                                       Soybean         0      0        30   70                                       Sugarbeet      30     40        100  100                                      Teaweed         0     30        80   80                                       Velvetleaf      0     30        80   90                                       Wheat           0     30        60   100                                      Wild buckwheat 40     70        90   90                                       Wild oat       40     50        80   100                                      ______________________________________                                                       Cmpd 92                                                        RATE (g/ha)      16     62                                                    ______________________________________                                        PREEMERGENCE                                                                  Barley           40     70                                                    Barnyardgrass    100    100                                                   Blackgrass       70     100                                                   Cheatgrass       70     90                                                    Chickweed        50     80                                                    Cocklebur        30     50                                                    Corn              0     40                                                    Cotton           50     90                                                    Crabgrass        60     70                                                    Field violet     --     --                                                    Giant foxtail    --     --                                                    Green foxtail    90     100                                                   Jimsonweed       70     90                                                    Johnsongrass     90     100                                                   Lambsquarters    90     100                                                   Morningglory     70     90                                                    Nutsedge         80     90                                                    Rape             90     100                                                   Rice             100    100                                                   Sicklepod        60     80                                                    Soybean          70     100                                                   Sugarbeet        80     90                                                    Teaweed          --     90                                                    Velvetleaf       50     60                                                    Wheat            40     70                                                    Wild buckwheat   80     80                                                    Wild oat         30     50                                                    ______________________________________                                                     Cmpd 93                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        PREEMERGENCE                                                                  Barley          0     20        40   60                                       Barnyardgrass   0     30        50   70                                       Blackgrass     30     50        70   100                                      Cheatgrass      0     30        50   70                                       Chickweed      --     --        --   --                                       Cocklebur       0      0        30   40                                       Corn            0      0         0    0                                       Cotton          0      0         0   20                                       Crabgrass       0     20        30   60                                       Field violet   20     30        60   80                                       Giant foxtail  30     50        70   80                                       Green foxtail   0      0        30   60                                       Jimsonweed      0     30        60   90                                       Johnsongrass   70     80        90   100                                      Lambsquarters   0     30        60   90                                       Morningglory    0     20        30   50                                       Nutsedge        0      0        30   70                                       Rape           50     70        80   90                                       Rice           30     50        90   100                                      Sicklepod       0     20        30   50                                       Soybean         0      0         0    0                                       Sugarbeet      30     50        80   90                                       Teaweed        30     50        70   90                                       Velvetleaf      0     30        50   70                                       Wheat           0      0        20   40                                       Wild buckwheat  0     30        50   70                                       Wild oat        0      0        30   50                                       ______________________________________                                                     Cmpd 96                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        PREEMERGENCE                                                                  Barley          0     20        30   80                                       Barnyardgrass   0     20        80   80                                       Blackgrass      0     50        50   70                                       Cheatgrass      0     30        50   80                                       Chickweed       0      0        40   40                                       Cocklebur       0     30        50   60                                       Corn            0      0         0    0                                       Cotton          0      0        40   70                                       Crabgrass       0      0        40   100                                      Field violet   --     --        --   --                                       Giant foxtail   0     20        90   100                                      Green foxtail   0     70        100  100                                      Jimsonweed      0     60        80   90                                       Johnsongrass    0     40        70   90                                       Lambsquarters   0     20        30   70                                       Morningglory    0      0        30   60                                       Nutsedge        0     20        40   60                                       Rape            0     70        70   90                                       Rice            0     50        90   90                                       Sicklepod       0      0        40   80                                       Soybean         0     20        50   60                                       Sugarbeet       0      0        60   80                                       Teaweed         0      0        30   30                                       Velvetleaf      0     30        30   40                                       Wheat           0      0        30   60                                       Wild buckwheat  0      0        50   90                                       Wild oat        0     30        40   40                                       ______________________________________                                                     Cmpd 100                                                         RATE (g/ha)    1      4         16   62                                       ______________________________________                                        PREEMERGENCE                                                                  Barley         30     50        70   90                                       Barnyardgrass  30     50        80   100                                      Blackgrass     50     60        70   90                                       Cheatgrass     50     70        80   90                                       Chickweed      30     50        70   90                                       Cocklebur        0    30        60   90                                       Corn            0      0         0    0                                       Cotton          0     30        50   60                                       Crabgrass       0     30        50   80                                       Field violet   --     --        --   --                                       Giant foxtail  70     90        100  100                                      Green foxtail  50     70        90   100                                      Jimsonweed      0     30        50   80                                       Johnsongrass   50     70        80   90                                       Lambsquarters  70     100       100  100                                      Morningglory    0     30        50   80                                       Nutsedge        0     30        60   90                                       Rape           70     100       100  100                                      Rice           30     60        80   90                                       Sicklepod      30     50        70   90                                       Soybean         0     30        40   60                                       Sugarbeet      70     90        100  100                                      Teaweed         0     30        50   70                                       Velvetleaf     30     60        90   95                                       Wheat           0     30        60   90                                       Wild buckwheat  0     30        60   90                                       Wild oat        0      0        30   50                                       ______________________________________                                                   Cmpd 106                                                           RATE (g/ha)  16           62     250                                          ______________________________________                                        PREEMERGENCE                                                                  Barley       50           80     90                                           Barnyardgrass                                                                              20           40     100                                          Blackgrass   80           100    100                                          Cheatgrass   70           100    100                                          Chickweed     0           10     20                                           Cocklebur     0           40     80                                           Corn          0            0     10                                           Cotton        0           10     20                                           Crabgrass    40           80     80                                           Field violet --           --     --                                           Giant foxtail                                                                              40           90     100                                          Green foxtail                                                                              40           90     100                                          Jimsonweed    0           --     20                                           Johnsongrass 70           90     100                                          Lambsquarters                                                                              80           90     100                                          Morningglory 20           40     50                                           Nutsedge     40           50     70                                           Rape         80           90     100                                          Rice         80           100    100                                          Sicklepod     0           20     60                                           Soybean       0            0     20                                           Sugarbeet    30           80     100                                          Teaweed      30           50     70                                           Velvetleaf    0           20     60                                           Wheat        20           40     60                                           Wild buckwheat                                                                             30           60     80                                           Wild oat     20           60     80                                           ______________________________________                                                   Cmpd 1                                                             RATE (g/ha)  0.25     1      4      16   62                                   ______________________________________                                        POSTEMERGENCE                                                                 Barley        0        0     30     80   90                                   Barnyardgrass                                                                              30       60     100    100  100                                  Blackgrass   50       50     70     85   100                                  Cheatgrass   20       30     65     85   95                                   Chickweed    --       --     --     --   --                                   Cocklebur     0       20     80     80   100                                  Corn          0        0      0      0   10                                   Cotton        0       20     30     80   85                                   Crabgrass    30       20     20     50   60                                   Field violet --         0     0     20   --                                   Giant foxtail                                                                               0       20     50     70   85                                   Green foxtail                                                                               0       20     30     75   85                                   Jimsonweed    0        0     10     20   30                                   Johnsongrass 60       80     100    100  100                                  Lambsquarters                                                                               0        0     20     20   50                                   Morningglory 10       30     50     85   90                                   Nutsedge      0       30     70     75   80                                   Rape         20       60     90     100  90                                   Rice         20       40     70     90   100                                  Sicklepod     0       50     80     70   100                                  Soybean       0        0     10     20   70                                   Sugarbeet    10        0     30     80   100                                  Teaweed       0       20     30     60   70                                   Velvetleaf    0       20     40     60   100                                  Wheat        10       10     60     100  100                                  Wild buckwheat                                                                              0       30     40     70   --                                   Wild oat      0        0     20     60   100                                  ______________________________________                                                   Cmpd 21                                                            RATE (g/ha)  0.25     1      4      16   62                                   ______________________________________                                        POSTEMERGENCE                                                                 Barley       20       20     60     70   70                                   Barnyardgrass                                                                              50       80     95     100  100                                  Blackgrass    0       50     80     90   90                                   Cheatgrass   20       30     50     90   100                                  Chickweed    --       --     --     --   --                                   Cocklebur      0       0     40     80   100                                  Corn          0        0      0      0    0                                   Cotton        0       30     60     80   100                                  Crabgrass     0        0      0     70   80                                   Field violet  0       30     40     80   80                                   Giant foxtail                                                                              40       70     100    100  100                                  Green foxtail                                                                              60       90     100    100  100                                  Jimsonweed    0        0     20     50   80                                   Johnsongrass 70       80     100    100  100                                  Lambsquarters                                                                               0       --      0     --   100                                  Morningglory  0       20     95     95   100                                  Nutsedge      0       30     40     70   100                                  Rape         50       80     100    100  100                                  Rice          0       40     90     100  100                                  Sicklepod     0       30     90     100  100                                  Soybean      40       50     80     90   90                                   Sugarbeet     0       20     40     70   80                                   Teaweed       0       --     --     --   80                                   Velvetleaf    0        0     50     90   100                                  Wheat        50       60     60     100  100                                  Wild buckwheat                                                                             20       20     50     60   80                                   Wild oat      0       20     70     80   100                                  ______________________________________                                                     Cmpd 46                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley         30     50        60   70                                       Barnyardgrass  50     70        80   90                                       Blackgrass     30     50        70   100                                      Cheatgrass     30     50        70   90                                       Chickweed      30     50        70   90                                       Cocklebur      30     40        50   60                                       Corn            0      0         0    0                                       Cotton          0     30        50   60                                       Crabgrass       0      0        30   50                                       Field violet   --     --        --   --                                       Giant foxtail  30     50        80   90                                       Green foxtail  30     50        70   80                                       Jimsonweed      0      0        30   60                                       Johnsongrass   30     60        90   100                                      Lambsquarters   0      0        30   50                                       Morningglory   30     50        70   80                                       Nutsedge        0     30        60   90                                       Rape           60     90        100  100                                      Rice           30     50        70   90                                       Sicklepod       0     30        60   90                                       Soybean         0     30        60   90                                       Sugarbeet      30     50        70   90                                       Teaweed         0     20        40   60                                       Velvetleaf     30     60        80   100                                      Wheat          30     50        80   100                                      Wild buckwheat 30     50        70   90                                       Wild oat        0      0        30   60                                       ______________________________________                                                     Cmpd 60                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley          0     40        60   90                                       Barnyardgrass  60     100       100  100                                      Blackgrass     60     100       100  100                                      Cheatgrass     40     60        80   100                                      Chickweed      30     60        90   100                                      Cocklebur      50     100       100  100                                      Corn           --     20        50   70                                       Cotton         20     30        90   100                                      Crabgrass       0      0        30   40                                       Field violet   --     --        --   --                                       Giant foxtail  20     20        80   90                                       Green foxtail  30     50        80   90                                       Jimsonweed     20     30        40   60                                       Johnsongrass   20     90        100  100                                      Lambsquarters   0     50        50   90                                       Morningglory   --     60        60   80                                       Nutsedge       20     30        80   90                                       Rape           80     100       100  100                                      Rice           60     60        90   100                                      Sicklepod      30     60        90   100                                      Soybean        60     80        90   100                                      Sugarbeet      --     60        80   100                                      Teaweed        20     30        40   60                                       Velvetleaf     70     80        100  100                                      Wheat           0     30        60   100                                      Wild buckwheat 70     70        80   90                                       Wild oat        0     40        60   80                                       ______________________________________                                                     Cmpd 64                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley          0     30        50   70                                       Barnyardgrass  30     50        80   100                                      Blackgrass     30     50        70   90                                       Cheatgrass      0     30        50   70                                       Chickweed      30     50        70   90                                       Cocklebur      70     80        90   100                                      Corn            0      0        20   60                                       Cotton         30     50        70   90                                       Crabgrass       0      0        30   50                                       Field violet   --     --        --   --                                       Giant foxtail   0     30        50   80                                       Green foxtail   0     30        50   70                                       Jimsonweed      0     30        60   90                                       Johnsongrass   30     50        70   90                                       Lambsquarters  60     70        80   90                                       Morningglory   50     70        90   100                                      Nutsedge       70     100       100  100                                      Rape           100    100       100  100                                      Rice           30     50        70   90                                       Sicklepod      50     70        100  100                                      Soybean        80     90        100  100                                      Sugarbeet      50     70        90   100                                      Teaweed        50     60        70   80                                       Velvetleaf     70     80        100  100                                      Wheat           0     30        50   70                                       Wild buckwheat 30     60        80   90                                       Wild oat        0      0        30   60                                       ______________________________________                                                     Cmpd 65                                                          RATE (g/ha)    0.25   1         4    16                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley         30     70        100  100                                      Barnyardgrass  60     100       100  100                                      Blackgrass     30     60        80   90                                       Cheatgrass     70     90        90   100                                      Chickweed      50     90        100  100                                      Cocklebur      50     80        100  100                                      Corn           90     100       100  100                                      Cotton          0     20        30   100                                      Crabgrass      30     60        90   100                                      Field violet   --     --        --   --                                       Giant foxtail  80     100       100  100                                      Green foxtail  70     100       100  100                                      Jimsonweed      0     20        80   100                                      Johnsongrass   60     100       100  100                                      Lambsquarters  80     100       100  100                                      Morningglory   40     90        100  100                                      Nutsedge       30     80        100  100                                      Rape           80     100       100  100                                      Rice           30     100       100  100                                      Sicklepod      50     90        100  100                                      Soybean        80     100       100  100                                      Sugarbeet      80     100       100  100                                      Teaweed         0     60        100  100                                      Velvetleaf     60     100       100  100                                      Wheat          80     90        100  100                                      Wild buckwheat 40     80        100  100                                      Wild oat       40     90        100  100                                      ______________________________________                                                     Cmpd 66                                                          RATE (g/ha)     0.25  1         4    16                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley         20     40        80   100                                      Barnyardgrass  30     80        100  100                                      Blackgrass     20     30        40   90                                       Cheatgrass     30     60        90   90                                       Chickweed      20     50        90   100                                      Cocklebur       0     30        90   100                                      Corn           30     50        90   100                                      Cotton          0      0        30   40                                       Crabgrass       0     40        60   100                                      Field violet   --     --        --   --                                       Giant foxtail  30     50        100  100                                      Green foxtail   0     50        90   100                                      Jimsonweed      0     60        90   100                                      Johnsongrass   40     60        80   100                                      Lambsquarters  50     60        90   100                                      Morningglory   20     40        90   100                                      Nutsedge        0     20        40   100                                      Rape           30     90        100  100                                      Rice           20     40        90   100                                      Sicklepod       0     30        90   100                                      Soybean        50     80        100  100                                      Sugarbeet      30     50        100  100                                      Teaweed         0     30        70   90                                       Velvetleaf     20     70        90   100                                      Wheat          40     80        90   100                                      Wild buckwheat  0     30        50   80                                       Wild oat       20     80        90   100                                      ______________________________________                                                     Cmpd 67                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley         20     40        80   90                                       Barnyardgrass  90     100       100  100                                      Blackgrass     40     80        90   90                                       Cheatgrass     40     80        90   100                                      Chickweed      40     60        90   100                                      Cocklebur      40     60        100  100                                      Corn           30     80        100  100                                      Cotton          0     40        80   100                                      Crabgrass      30     40        80   100                                      Field violet   --     --        --   --                                       Giant foxtail   0     30        100  100                                      Green foxtail  20     40        70   90                                       Jimsonweed     70     100       100  100                                      Johnsongrass   80     100       100  100                                      Lambsquarters  80     100       100  100                                      Morningglory   60     90        100  100                                      Nutsedge       30     80        90   100                                      Rape           80     100       100  100                                      Rice           30     80        100  100                                      Sicklepod      30     100       100  100                                      Soybean        60     90        100  100                                      Sugarbeet      80     100       100  100                                      Teaweed        30     70        90   100                                      Velvetleaf     50     80        90   100                                      Wheat           0     30        40   70                                       Wild buckwheat 30     60        80   100                                      Wild oat       20     30        80   90                                       ______________________________________                                                     Cmpd 68                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley         40     90        100  100                                      Barnyardgrass  60     100       100  100                                      Blackgrass     30     80        100  100                                      Cheatgrass     80     90        100  100                                      Chickweed      40     70        90   100                                      Cocklebur      40     80        100  100                                      Corn            0     20        90   100                                      Cotton          0     30        80   100                                      Crabgrass      30     70        90   100                                      Field violet   --     --        --   --                                       Giant foxtail  30     90        100  100                                      Green foxtail  40     80        100  100                                      Jimsonweed     70     100       100  100                                      Johnsongrass   70     90        100  100                                      Lambsquarters  70     90        100  100                                      Morningglory   30     80        100  100                                      Nutsedge       20     70        80   100                                      Rape           40     100       100  100                                      Rice           50     90        100  100                                      Sicklepod      30     90        100  100                                      Soybean        70     100       100  100                                      Sugarbeet      40     100       100  100                                      Teaweed        20     80        90   90                                       Velvetleaf     40     90        100  100                                      Wheat          60     90        100  100                                      Wild buckwheat 30     70        90   100                                      Wild oat       70     90        100  100                                      ______________________________________                                                       Cmpd 92                                                        RATE (g/ha)      4      16                                                    ______________________________________                                        POSTEMERGENCE                                                                 Barley           70     80                                                    Barnyardgrass    60     90                                                    Blackgrass       90     90                                                    Cheatgrass       90     100                                                   Chickweed        70     90                                                    Cocklebur        80     100                                                   Corn              0      0                                                    Cotton           90     90                                                    Crabgrass         0     60                                                    Field violet     --     --                                                    Giant foxtail    90     90                                                    Green foxtail    70     80                                                    Jimsonweed       50     50                                                    Johnsongrass     100    100                                                   Lambsquarters    80     90                                                    Morningglory     70     100                                                   Nutsedge          0     60                                                    Rape             100    100                                                   Rice             60     100                                                   Sicklepod        90     100                                                   Soybean          70     100                                                   Sugarbeet        100    100                                                   Teaweed          20     60                                                    Velvetleaf       70     70                                                    Wheat            90     90                                                    Wild buckwheat   70     80                                                    Wild oat         60     80                                                    ______________________________________                                                     Cmpd 93                                                          RATE (g/ha)    1      4         16   62                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley          0      0         0   10                                       Barnyardgrass  30     40        60   70                                       Blackgrass     50     50        70   80                                       Cheatgrass      0      0        30   70                                       Chickweed      --     --        --   --                                       Cocklebur      60     60        70   90                                       Corn            0      0         0   10                                       Cotton         --     40        50   70                                       Crabgrass       0      0         0   20                                       Field violet    0      0         0   30                                       Giant foxtail  --      0        20   60                                       Green foxtail  --     40        50   90                                       Jimsonweed     60     80        90   100                                      Johnsongrass   90     90        100  100                                      Lambsquarters  --     50        60   70                                       Morningglory   70     70        80   80                                       Nutsedge        0      0        30   40                                       Rape           100    100       100  100                                      Rice            0      0        60   80                                       Sicklepod       0      0        40   70                                       Soybean        --      0        10   50                                       Sugarbeet      --     30        80   100                                      Teaweed         0      0         0   50                                       Velvetleaf      0      0        20   70                                       Wheat           0      0        10   40                                       Wild buckwheat  0      0        30   30                                       Wild oat        0      0         0   50                                       ______________________________________                                                     Cmpd 96                                                          RATE (g/ha)    0.25   1         4    16                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley          0     20        40   90                                       Barnyardgrass  30     40        90   100                                      Blackgrass      0      0        70   80                                       Cheatgrass      0      0        70   70                                       Chickweed       0      0        40   60                                       Cocklebur        0     0        30   70                                       Corn            0      0        20   80                                       Cotton          0      0         0   20                                       Crabgrass       0      0        40   80                                       Field violet   --     --        --   --                                       Giant foxtail   0     --        40   100                                      Green foxtail   0     40        70   90                                       Jimsonweed      0     30        50   60                                       Johnsongrass    0     70        90   100                                      Lambsquarters   0      0         0   40                                       Morningglory    0      0        30   60                                       Nutsedge        0     20        30   60                                       Rape           20     30        90   100                                      Rice            0      0        50   90                                       Sicklepod       0      0        40   80                                       Soybean        30     40        90   90                                       Sugarbeet       0     20        30   60                                       Teaweed         0      0        20   70                                       Velvetleaf      0      0        20   60                                       Wheat          20     40        50   60                                       Wild buckwheat  0      0        --   80                                       Wild oat        0     30        50   70                                       ______________________________________                                                     Cmpd 100                                                         RATE (g/ha)    1      4         16   62                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley         50     70        100  100                                      Barnyardgrass  30     40        80   100                                      Blackgrass     70     90        100  100                                      Cheatgrass     70     80        100  100                                      Chickweed      50     70        90   100                                      Cocklebur      70     100       100  100                                      Corn           --      0        20   40                                       Cotton         50     80        90   90                                       Crabgrass       0      0        50   60                                       Field violet   --     --        --   --                                       Giant foxtail  40     50        90   100                                      Green foxtail  30     50        80   90                                       Jimsonweed      0      0        20   40                                       Johnsongrass   70     100       100  100                                      Lambsquarters  50     70        100  100                                      Morningglory   60     90        100  100                                      Nutsedge        0     30        60   100                                      Rape           100    100       100  100                                      Rice           50     90        100  100                                      Sicklepod      50     70        100  100                                      Soybean        80     80        100  100                                      Sugarbeet      90     100       100  100                                      Teaweed         0     30        50   70                                       Velvetleaf     30     80        90   100                                      Wheat          50     70        100  100                                      Wild buckwheat 30     60        90   100                                      Wild oat       40     70        100  100                                      ______________________________________                                                     Cmpd 106                                                         RATE (g/ha)    1      4         16   62                                       ______________________________________                                        POSTEMERGENCE                                                                 Barley          0     30        50   90                                       Barnyardgrass  30     60        90   100                                      Blackgrass     50     70        90   90                                       Cheatgrass      0     30        70   90                                       Chickweed       0      0        30   70                                       Cocklebur       0     50        70   100                                      Corn            0      0         0   20                                       Cotton          0      0        10   20                                       Crabgrass       0      0         0    0                                       Field violet   --     --        --   --                                       Giant foxtail   0     20        40   90                                       Green foxtail  20     40        80   90                                       Jimsonweed      0      0        20   40                                       Johnsongrass   50     50        70   90                                       Lambsquarters  40     60        80   90                                       Morningglory    0     50        90   90                                       Nutsedge        0      0        20   30                                       Rape           70     100       100  100                                      Rice            0     30        70   100                                      Sicklepod      --     20        --   50                                       Soybean         0     40        50   90                                       Sugarbeet      40     70        80   90                                       Teaweed         0      0        20   30                                       Velvetleaf      0     30        70   90                                       Wheat           0     40        80   100                                      Wild buckwheat  0      0        50   70                                       Wild oat        0     60        90   100                                      ______________________________________                                    

Test C Postemergence

Six round pots (17 cm diameter by 15 cm deep) were used to grow plantsto the treatment stage. Four were planted with seeds or tubers of fourspecies each and another with soybeans using Sassafras sandy loam as thegrowing media. The sixth pot was planted to corn using a Tama silt loam.During spraying, the soil of this pot was temporarily covered withperlite then later removed so any effects noted would be from foliaruptake only. A separate pot of corn (25.5 cm diameter by 19.5 cm deep)grown in Sassafras sandy loam was also included to determine foliar/soiltreatment effects on plant growth. Plants were grown 10 to 20 days andwere in the 2 to 5 leaf stage when sprayed postemergence with compoundsof the invention. Species included were as follows: G4646 corn [maize](Zea mays, variety Funk G4646), Williams soybeans (Glycine max, varietyWilliams), green foxtail (Setaria viridis), giant foxtail (Setariafaberi), fall panicum (Panicum dichotomiflorum), crabgrass (Digitariasanguinalis), barnyardgrass (Echinochloa crus-galli), johnsongrass(Sorghum halepense), G522 sorghum (Sorghum vulgare, variety Funk G522),nutsedge (Cyperus rotundus), velvetleaf (Abutlion theophrasti),cocklebur (Xanthium pensylvanicum), smartweed (Polygonum persicaria,lambsquarter (Chenopodium album), pigweed (Amaranthus retroflexus),ivyleaf morningglory (Ipomoea hederacea), jimsonweed (Daturastramonium), ragweed (Ambrosia artemisiifolia).

Preemergence

Plantings were made as above except all in Tama silt loam. Compoundswere sprayed preemergence the day after planting. All pots were thenwatered to simulate rainfall.

After treatment, all plantings were maintained in a greenhouse about 20days and then visually rated for plant response. Ratings are based on ascale of 0 to 100 where 0=no effect and 100=complete control. Responseratings are shown in Table C.

                  TABLE C                                                         ______________________________________                                        CMPD 1                                                                        RATE GM/HA  0004   0008   0016  0032 0064  0125                               ______________________________________                                        POST                                                                          SOIL TYPE   SAS    SAS    SAS   SAS  SAS   SAS                                G4646 CORN  0      0      0     0    25    40                                 WILLMS      0      20     35    50   65    85                                 SOYBEANS                                                                      GREEN       50     65     80    90   95    100                                FOXTAIL                                                                       GIANT FOXTAIL                                                                             40     65     70    90   95    100                                FALL PANICUM                                                                              70     90     95    100  100   100                                LARGE       0      0      0     30   70    80                                 CRABGRASS                                                                     BARNYARD-   90     100    100   100  100   100                                GRASS                                                                         JOHNSONGRASS                                                                              100    100    100   100  100   100                                G522 SORGHUM                                                                              100    100    100   100  100   100                                PURPLE      30     50     75    90   100   100                                NUTSEDGE                                                                      VELVETLEAF  20     45     75    85   95    100                                COCKLEBUR   50     85     100   100  100   100                                LADY        0      0      0     25   50    70                                 SMARTWEED                                                                     LAMBSQUARTER                                                                              0      0      0     0    35    50                                 REDROOT     70     85     100   100  100   100                                PIGWEED                                                                       IVY         50     85     100   100  100   100                                MORNINGLORY                                                                   JIMSONWEED  0      0      0     0    0     35                                 PERLITE CORN                                                                              0      0      0     0    20    30                                 ______________________________________                                        CMPD 21                                                                       RATE GM/HA  0002   0004   0008 0016 0032 0064 0125                            ______________________________________                                        POST                                                                          SOIL TYPE   SAS    SAS    SAS  SAS  SAS  SAS  SAS                             G4646 CORN  0      0      0    0    10   20   70                              WILLMS      95     98     100  100  100  100  100                             SOYBEANS                                                                      GREEN       80     90     90   100  100  100  100                             FOXTAIL                                                                       GIANT FOXTAIL                                                                             70     90     90   95   100  100  100                             FALL PANICUM                                                                              80     95     98   100  100  100  100                             LARGE       0      0      0    30   40   60   70                              CRABGRASS                                                                     BARNYARD-   100    100    100  100  100  100  100                             GRASS                                                                         JOHNSONGRASS                                                                              100    100    100  100  100  100  100                             G522 SORGHUM                                                                              100    100    100  100  100  100  100                             VELVETLEAF  40     60     60   60   90   100  100                             COCKLEBUR   40     40     40   90   100  100  100                             LADY        0      0      0    30   50   80   80                              SMARTWEED                                                                     LAMBSQUARTER                                                                              30     30     30   60   40   50   70                              REDROOT     90     100    100  100  100  100  100                             PIGWEED                                                                       IVY         0      0      0    20   30   40   70                              MORNINGLORY                                                                   JIMSONWEED  0      20     20   30   40   40   50                              PERLITE CORN                                                                              0      0      0    10   10   20   60                              ______________________________________                                        CMPD 46                                                                       RATE GM/HA  0002   0004   0008 0016 0032 0064 0125                            ______________________________________                                        POST                                                                          SOIL TYPE   SAS    SAS    SAS  SAS  SAS  SAS  SAS                             G4646 CORN  0      0      0    0    0    0    30                              WILLMS      25     45     75   90   100  100  100                             SOYBEANS                                                                      GREEN       0      30     60   75   85   90   100                             FOXTAIL                                                                       GIANT FOXTAIL                                                                             0      30     60   75   85   90   100                             TALL PANICUM                                                                              0      35     70   90   100  100  100                             LARGE       0      0      0    0    25   35   45                              CRABGRASS                                                                     BARNYARD-   45     90     100  100  100  100  100                             GRASS                                                                         JOHNSONGRASS                                                                              60     80     95   100  100  100  100                             G522 SORGHUM                                                                              75     90     100  100  100  100  100                             PURPLE      0      35     45   60   80   95   100                             NUTSEDGE                                                                      VELVETLEAF  0      0      35   70   70   85   95                              COCKLEBUR   0      30     40   60   75   95   95                              LADY        0      30     75   85   95   100  100                             SMARTWEED                                                                     LAMBSQUARTER                                                                              0      0      0    30   40   55   65                              REDROOT     35     70     100  100  100  100  100                             PIGWEED                                                                       IVY         0      0      20   40   60   70   80                              MORNINGLORY                                                                   JIMSONWEED  0      0      0    0    25   40   60                              PERLITE CORN                                                                              0      0      0    0    0    0    25                              ______________________________________                                        CMPD 60                                                                       RATE GM/HA  0002   0004   0008 0016 0032 0064 0125                            ______________________________________                                        POST                                                                          SOIL TYPE   SAS    SAS    SAS  SAS  SAS  SAS  SAS                             G4646 CORN  0      0      0    0    30   60   85                              WILLMS      100    100    100  100  100  100  100                             SOYBEANS                                                                      GREEN       20     35     45   65   75   85   95                              FOXTAIL                                                                       GIANT FOXTAIL                                                                             0      25     40   60   75   90   100                             TALL PANICUM                                                                              60     75     90   95   100  100  100                             LARGE       0      0      0    30   40   60   80                              CRABGRASS                                                                     BARNYARD-   80     95     100  100  100  100  100                             GRASS                                                                         JOHNSONGRASS                                                                              95     100    100  100  100  100  100                             G522 SORGHUM                                                                              100    100    100  100  100  100  100                             PURPLE      30     50     65   75   100  100  100                             NUTSEDGE                                                                      VELVETLEAF  20     35     55   85   100  100  100                             COCKLEBUR   35     40     60   70   85   100  100                             LADY        20     30     40   60   80   100  100                             SMARTWEED                                                                     LAMBSQUARTER                                                                              0      0      0    35   60   90   95                              REDROOT     60     75     100  100  100  100  100                             PIGWEED                                                                       IVY         0      0      20   40   65   80   95                              MORNINGLORY                                                                   JIMSONWEED  0      0      0    20   40   65   85                              PERLITE CORN                                                                              0      0      0    0    25   50   70                              ______________________________________                                        CMPD 160                                                                      RATE GM/HA  0016     0032     0064   0125                                     ______________________________________                                        PRE                                                                           SOIL TYPE   TAM      TAM      TAM    TAM                                      G4646 CORN  0        0        0      0                                        WILLMS      30       40       60     85                                       SOYBEANS                                                                      GREEN       20       25       35     60                                       FOXTAIL                                                                       GIANT FOXTAIL                                                                             20       20       30     40                                       FALL PANICUM                                                                              70       80       95     100                                      LARGE       0        0        20     --                                       CRABGRASS                                                                     BARNYARD-   65       70       90     100                                      GRASS                                                                         JOHNSONGRASS                                                                              70       90       100    100                                      G522 SORGHUM                                                                              75       100      100    100                                      PURPLE      35       60       80     --                                       NUTSEDGE                                                                      VELVETLEAF  0        0        0      --                                       COCKLEBUR   0        0        0      --                                       LADY        50       65       95     --                                       SMARTWEED                                                                     LAMBSQUARTER                                                                              25       40       60     --                                       REDROOT     50       60       90     --                                       PIGWEED                                                                       IVY         0        0        0      --                                       MORNINGLORY                                                                   JIMSONWEED  0        0        0      --                                       ______________________________________                                        CMPD 92                                                                       RATE GM/HA  0016     0032     0064   0125                                     ______________________________________                                        PRE                                                                           SOIL TYPE   TAM      TAM      TAM    TAM                                      G4646 CORN  0        0        0      0                                        WILLMS      0        25       50     80                                       SOYBEANS                                                                      GREEN       0        35       70     100                                      FOXTAIL                                                                       GIANT FOXTAIL                                                                             0        30       70     95                                       TALL PANICUM                                                                              20       45       85     95                                       LARGE       0        20       40     70                                       CRABGRASS                                                                     BARNYARD-   25       45       85     100                                      GRASS                                                                         JOHNSONGRASS                                                                              50       65       100    100                                      G522 SORGHUM                                                                              45       55       90     100                                      PURPLE      0        25       65     80                                       NUTSEDGE                                                                      VELVETLEAF  0        0        0      30                                       COCKLEBUR   0        0        0      20                                       LADY        30       60       95     100                                      SMARTWEED                                                                     LAMBSQUARTER                                                                              20       40       90     100                                      REDROOT     50       70       100    100                                      PIGWEED                                                                       IVY         0        0        0      25                                       MORNINGLORY                                                                   JIMSONWEED  0        0        0      35                                       ______________________________________                                        CMPD 92                                                                       RATE GM/HA  0002   0004   0008 0016 0032 0064 0125                            ______________________________________                                        POST                                                                          SOIL TYPE   SAS    SAS    SAS  SAS  SAS  SAS  SAS                             G4646 CORN  0      0      0    0    20   35   60                              WILLMS      65     85     100  100  100  100  100                             SOYBEANS                                                                      GREEN       40     60     80   90   95   100  100                             FOXTAIL                                                                       GIANT FOXTAIL                                                                             40     65     80   100  100  100  100                             TALL PANICUM                                                                              0      40     80   95   100  100  100                             LARGE       0      0      0    25   40   50   80                              CRABGRASS                                                                     BARNYARD-   0      30     50   70   100  100  100                             GRASS                                                                         JOHNSONGRASS                                                                              80     95     100  100  100  100  100                             G522 SORGHUM                                                                              85     95     100  100  100  100  100                             PURPLE      0      35     60   90   100  100  100                             NUTSEDGE                                                                      VELVETLEAF  0      25     40   65   85   95   100                             COCKLEBUR   35     50     90   100  100  100  100                             LADY        25     40     50   60   70   85   95                              SMARTWEED                                                                     LAMBSQUARTER                                                                              40     65     85   95   100  100  100                             REDROOT     75     95     100  100  100  100  100                             PIGWEED                                                                       IVY         0      30     55   70   85   95   100                             MORNINGLORY                                                                   JIMSONWEED  0      0      20   40   60   70   85                              PERLITE CORN                                                                              0      0      0    0    0    20   40                              ______________________________________                                        CMPD 96                                                                       RATE GM/HA  0016    0032    0064  0125  0250                                  ______________________________________                                        PRE                                                                           SOIL TYPE   TAM     TAM     TAM   TAM   TAM                                   G4646 CORN  0       0       0     0     0                                     WILLMS      0       0       0     20    45                                    SOYBEANS                                                                      GREEN       0       15      20    35    50                                    FOXTAIL                                                                       GIANT FOXTAIL                                                                             0       15      20    35    50                                    TALL PANICUM                                                                              0       0       0     0     15                                    LARGE       0       0       0     0     15                                    CRABGRASS                                                                     BARNYARD-   0       15      30    70    85                                    GRASS                                                                         JOHNSONGRASS                                                                              0       20      45    55    75                                    G522 SORGHUM                                                                              20      35      55    75    95                                    PURPLE      0       0       0     0     0                                     NUTSEDGE                                                                      VELVETLEAF  0       0       20    30    40                                    COCKLEBUR   0       10      20    35    50                                    LADY        15      35      50    60    75                                    SMARTWEED                                                                     LAMBSQUARTER                                                                              0       0       0     15    25                                    REDROOT     0       25      45    65    85                                    PIGWEEID                                                                      IVY         0       0       0     0     0                                     MORNINGLORY                                                                   JIMSONWEED  0       0       0     15    20                                    ______________________________________                                        CMPD 96                                                                       RATE GM/HA  0002   0004   0008  0016 0032  0064                               ______________________________________                                        POST                                                                          SOIL TYPE   SAS    SAS    SAS   SAS  SAS   SAS                                G4646 CORN  0      20     50    60   80    90                                 WILLMS      90     90     98    98   100   100                                SOYBEANS                                                                      GREEN       50     60     70    70   90    98                                 FOXTAIL                                                                       GIANT FOXTAIL                                                                             40     50     60    70   98    100                                LARGE       0      0      0     20   40    50                                 CRABGRASS                                                                     BARNYARD-   70     98     100   100  100   100                                GRASS                                                                         JOHNSONGRASS                                                                              60     98     100   100  100   100                                G522 SORGHUM                                                                              80     90     98    100  100   100                                PURPLE      0      0      0     0    30    70                                 NUTSEDGE                                                                      VELVETLEAF  0      0      30    50   60    90                                 COCKLEBUR   30     70     80    90   100   100                                LADY        20     30     30    50   70    98                                 SMARTWEED                                                                     LAMBSQUARTER                                                                              0      0      30    30   30    30                                 REDROOT     0      0      40    40   80    90                                 PIGWEED                                                                       IVY         0      30     30    30   40    50                                 MORNINGLORY                                                                   JIMSONWEED  40     60     60    60   100   100                                PERLITE CORN                                                                              20     20     30    60   60    90                                 ______________________________________                                        CMPD 100                                                                      RATE GM/HA  0016    0032    0064   0125  0250                                 ______________________________________                                        PRE                                                                           SOIL TYPE   TAM     TAM     TAM    TAM   TAM                                  G4646 CORN  0       0       0      0     20                                   WILLMS      0       25      40     70    80                                   SOYBEANS                                                                      GREEN       25      45      85     95    100                                  FOXTAIL                                                                       GIANT FOXTAIL                                                                             0       35      70     95    100                                  TALL PANICUM                                                                              40      85      100    100   100                                  LARGE       0       20      35     50    65                                   CRABGRASS                                                                     BARNYARD-   35      60      100    100   100                                  GRASS                                                                         JOHNSONGRASS                                                                              70      90      100    100   100                                  G522 SORGHUM                                                                              75      95      100    100   100                                  PURPLE      30      50      70     90    100                                  NUTSEDGE                                                                      VELVETLEAF  0       0       0      0     25                                   COCKLEBUR   0       0       20     35    50                                   LADY        40      70      95     100   100                                  SMARTWEED                                                                     LAMBSQUARTER                                                                              25      40      65     95    100                                  REDROOT     30      65      90     100   100                                  PIGWEED                                                                       IVY         0       0       0      0     35                                   MORNINGLORY                                                                   JIMSONWEED  0       0       30     45    70                                   ______________________________________                                        CMPD 100                                                                      RATE GM/HA  0002   0004   0008 0016 0032 0064 0125                            ______________________________________                                        POST                                                                          SOIL TYPE   SAS    SAS    SAS  SAS  SAS  SAS  SAS                             G4646 CORN  0      0      0    0    0    0    30                              WILLMS      65     75     90   100  100  100  100                             SOYBEANS                                                                      GREEN       50     65     80   95   100  100  100                             FOXTAIL                                                                       GIANT FOXTAIL                                                                             45     60     80   90   95   100  100                             FALL PANICUM                                                                              50     65     80   95   95   100  100                             LARGE       0      0      0    30   40   50   80                              CRABGRASS                                                                     BARNYARD-   50     60     70   80   100  100  100                             GRASS                                                                         JOHNSONGRASS                                                                              95     100    100  100  100  100  100                             G522 SORGHUM                                                                              100    100    100  100  100  100  100                             PURPLE      0      20     40   65   85   90   95                              NUTSEDGE                                                                      VELVETLEAF  0      40     70   80   90   100  100                             COCKLEBUR   45     95     100  100  100  100  100                             LADY        0      20     45   60   70   95   100                             SMARTWEED                                                                     LAMBSQUARTER                                                                              30     40     60   80   90   100  100                             REDROOT     65     90     100  100  100  100  100                             PIGWEED                                                                       IVY         30     70     85   100  100  100  100                             MORNINGLORY                                                                   JIMSONWEED  0      0      0    0    25   45   70                              PERLITE CORN                                                                              0      0      0    0    0    0    20                              ______________________________________                                    

Test D

Potatoes (Solanum tuberosum, cult. `Green Mountain`) were grown in Metro350 medium in 20 cm plastic pots. Potatoes were 17 days old at time ofspraying. Barnyardgrass (Echinochloa crus-galli), johnsongrass (Sorghumhalepense), giant foxtail (Setaria faberii), crabgrass (Digitariasanguinalis), purple nutsedge (Cyperus rotundus), jimsonweed (Daturastramonium), velvetleaf (Abutilon theophrasti), cocklebur (Xanthiumpensylvanicum), and morningglory (Ipomoea hederacea) were grown inSassafras sandy loam (pH 6.5, 1% organic matter) in plastic-lined 25 cmpots. These plants were 9 days old at the time of spraying.

Compound 21 was sprayed at 62, 16, 4, and 1 g/ha. The compound wassprayed at each rate on one pot containing potato plants and at the sametime on one pot containing the remaining species. Compound 21 wasdissolved in a non-phytotoxic solvent. The solvent was sprayed at 374l/ha. Plants were maintained in a greenhouse and were evaluated 11 daysafter spraying.

All sprayed plants were evaluated for injury as compared to controlplants. Injury was measured visually using a 0 to 100% scale where 0=noeffect and 100=complete control. Results are shown in Table D.

                  TABLE D                                                         ______________________________________                                        Compound 21                                                                               Rate (g/ha)                                                       Species       62     16         4    1                                        ______________________________________                                        Potato         0      0          0    0                                       Barnyardgrass 100    100        70   30                                       Johnsongrass  100    100        100  60                                       Giant foxtail 100    100        90   60                                       Crabgrass     90     85         60   50                                       Purple nutsedge                                                                             90     90         80   30                                       Jimsonweed    80     60         40   20                                       Velvetleaf    100    95         50   20                                       Cocklebur     90     50         30    0                                       Morningglory  90     70         40   20                                       ______________________________________                                    

Test E

Tomatoes (Lycopersicon esculentum cult. `Rutgers`) and peppers (Capsicumfrutescens cult. `Yolo`) were grown in Metro 350 medium in 10 cm plasticpots. Tomatoes and peppers were 19 days old at time of spraying. Purplenutsedge (Cyperus rotundus), crabgrass (Digitaria sanguinalis),sicklepod (Cassia tora), prickley sida (Sida spinosa), jimsonweed(Datura stramonium), velvetleaf (Abutilon theophrasti), lambsquarter(Chenopodium album), green foxtail (Setaria viridis), cocklebur(Xanthium pensylvanicum), morningglory (Ipomoea hederacea), johnsongrass(Sorghum halepense), barnyardgrass (Echinochloa crus-galli), giantfoxtail (Setaria faberii), wild buckwheat (Polygonum convolvulus), downybrome (Bromus tectorum), wild oat (Avena fatua), chickweed (Stellariaspp.), and blackgrass (Alopecurus myosuroides), were grown in Sassafrassandy loam (pH 6.5, 1% organic matter) in plastic-lined 25 cm pots.These plants were 7 to 11 days old at the time of spraying.

Compound 21 was sprayed at 62, 16, 4, and 1 g/ha. The compound wassprayed at each rate on one pot containing tomatoes, one pot containingpeppers, and on three pots containing the remaining species. Thecompound was dissolved in a non-phytotoxic solvent, and the solvent wassprayed at 374 l/ha. Plants were maintained in a greenhouse and wereevaluated 16 days after spraying.

All sprayed plants were evaluated for injury as compared to controlplants. Injury was measured visually using a 0 to 100% scale where 0=noeffect and 100=complete control. Results are shown in Table E.

                  TABLE E                                                         ______________________________________                                        Compound 20                                                                                Rage (g/ha)                                                      Species        62     16        4    1                                        ______________________________________                                        Tomatoes        10     0         0    0                                       Peppers         80     70       50   30                                       Nutsedge       100    100       30    0                                       Crabgrass       90     80       50   30                                       Sicklepod      100    100       90   40                                       Prickley sida  100    100       50   20                                       Jimsonweed     100     50       10    0                                       Velvetleaf     100    100       70   50                                       Lambsquarter    60     50       40    0                                       Green foxtail  100    100       100  50                                       Cocklebur      100     80       50   20                                       Morningglory    90     85       50   20                                       Johnsongrass   100    100       100  50                                       Barnyardgrass  100    100       100  40                                       Giant foxtail  100    100       90   40                                       Wild buckwheat 100     90       90   40                                       Downy brome    100    100       80   20                                       Wild oats      100     70       30   20                                       Chickweed      100    100       90   90                                       Blackgrass     100    100       100  70                                       ______________________________________                                    

What is claimed is:
 1. A compound selected from ##STR58## wherein J is##STR59## R is H or CH₃ ; W is O or S;R₁ is R_(f) or R_(g) ; R_(f) is H,C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, NO₂, C₁ -C₃ alkoxy, C₁ -C₃alkylthio or CN; R_(g) is C₁ -C₃ haloalkyl, cyclopropyl, C₁ -C₃ alkylsubstituted by C₁ -C₃ alkoxy, OH, C₁ -C₂ alkylthio or CN, CN, W₂ R₁₁,amino, C₁ -C₃ alkylamino or C₁ -C₃ dialkylamino; R₂ is C₁ -C₄alkylsulfinyl, C₁ -C₄ alkylsulfonyl, C₃ -C₅ cycloalkylthio, C₃ -C₅cycloalkylsulfinyl, C₃ -C₅ cycloalkylsulfonyl, SO₂ NH₂, SO₂ NR_(d)R_(e), SO₂ NR'₇ R₈, SO₂ NR₇ R₈, OSO₂ R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂alkyl)₂, CN, CO₂ R₉, CO₂ R'₉, CH₂ F, CF₂ H, CH₂ Cl, CCl₂ H or C₂ -C₄haloalkyl; R₇ is H, C₂ -C₃ cyanoalkyl, C₃ -C₄ alkenyl or C₃ -C₄ alkynyl;R'₇ is C₁ -C₄ alkyl; R₈ is C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, C₃ -C₄alkenyl, C₃ -C₄ alkynyl, C₂ -C₄ alkoxyalkyl or cyclopropyl; or R₇ and R₈may be taken together as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ -- or --CH₂CH₂ OCH₂ CH₂ --; R₉ is CH₂ CH₂ R₁₀, CH₂ CF₃, C₃ -C₄ haloalkyl, C₃ -C₄alknyl, C₂ -C₄ alkylthioalkyl, C₃ -C₅ cycloalkyl or C₄ -C₇cycloalkylalkyl; R'₉ is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, CH₂ CH₂ Cl, CH₂CH₂ Br, CH₂ CH₂ OCH₃ or CH₂ CH₂ OC₂ H₅ ; R₁₀ is OH, F, CN, OSO₂ (C₁ -C₃alkyl) or OSO₂ (C₁ -C₃ haloalkyl); R₁₁ is C₁ -C₃ alkyl, C₁ -C₃haloalkyl, C₃ -C₄ alkenyl or C₃ -C₄ alkynyl; W₁ is O or S; W₂ is O or S;A is ##STR60## X is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₂ -C₄ haloalkoxy,C₁ -C₄ haloalkyl, C₂ -C₄ haloalkylthio, C₁ -C₄ alkylthio, halogen, C₂-C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino or di(C₁-C₃ alkyl)amino; Y is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₂ -C₄ haloalkoxy,C₂ -C₄ haloalkylthio, C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino, C₃ -C₄alkenyloxy, C₃ -C₄ alkynyloxy, C₂ -C₅ alkylthioalkyl, C₂ -C₅alkylsulfinylalkyl, C₂ -C₅ alkylsulfonylalkyl, C₁ -C₄ haloalkyl, C₂ -C₄alkynyl, C₃ -C₅ cycloalkyl, azido, ##STR61## N(OCH₃)CH₃ ; m is 2 or 3;Q₁ and Q₂ are independently O or S; R_(a) is H or C₁ -C₃ alkyl; R_(b)and R_(c) are independently C₁ -C₃ alkyl; R_(d) is H or C₁ -C₂ alkyl;R_(e) is C₁ -C₂ alkoxy; Z is CH;and their agriculturally suitable salts;provided that 1) when X is halogen, then Y is OCH₃, OC₂ H₅, NH₂, NHCH₃,N(CH₃)₂ or N(OCH₃)CH₃ ; 2) when W is S, then R is H and Y is CH₃, OCH₃,OC₂ H₅, CH₂ OCH₃, C₂ H₅, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂OCH₃, ##STR62## 3) when the total number of carbon atoms of X and Y isgreater than four, then the combined number of carbons of R₁ or R₂ isless than or equal to six; 4) when R₂ is C₁ -C₄ alkylsulfinyl, C₁ -C₄alkylsulfonyl, SO₂ NR_(d) R_(e), SO₂ NR'₇ R₈ or CO₂ R'₉, then Y is otherthan C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, C₂ -C₅ alkylthioalkyl, C₂-C₅ alkylsulfinylalkyl, C₂ -C₅ alkylsulfonylalkyl, ##STR63## 5) when R₂is CO₂ R'₉ or SO₂ NR'₇ R, then R₁ is R_(g) and when R₂ is other than CO₂R'₉ or SO₂ NR'₇ R₈, then R₁ is R_(f) ; 6) when J is J-1;R is H or CH₃ ;X is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, Cl, F, Br, I, CH₂ F, CF₃, OCH₂ CH₂ F,OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; Y is H, C₁ -C₂ alkyl, C₁ -C₂alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃, N(OCH₃)CH₃, N(CH₃)₂, CF₃, SCH₃,OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, C(O)R_(a), cyclopropyl,C.tbd.CH or C.tbd.CCH₃ ; R_(a) is H or CH₃ ; Z is CH; W is O; R₁ isR_(f) ; and R_(f) is H, C₁ -C₂ alkyl, C₁ haloalkyl, C₁ -C₂ alkoxy or C₁-C₂ thioalkyl; then R₂ is other than C₁ -C₄ alkylsulfinyl or C₁ -C₄alkylsulfonyl and 7) when J is J-1;W is O; R is H or CH₃ ; R₁ is R_(f)or R_(g) ; R_(f) is C₁ haloalkyl, halogen or OCH₃ ; R_(g) is C₁ -C₂haloalkyl or W₂ R₁₁ ; W₂ is O or S; R₉ is CH₂ CH₂ R₁₀, CH₂ CF₃, C₃ -C₄haloalkyl, C₃ -C₄ alkynyl, C₂ -C₄ alkylthioalkyl, C₃ -C₅ cycloalkyl orC₄ -C₇ cycloalkylalkyl; R'₉ is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, CH₂ CH₂ Cl,CH₂ CH₂ Br, CH₂ CH₂ OCH₃ or CH₂ CH₂ OC₂ H₅ ; R₁₀ is OH, F, CN, OSO₂ (C₁-C₃ alkyl) or OSO₂ (C₁ -C₃ haloalkyl); R₁₁ is C₁ -C₃ alkyl or C₁ -C₃haloalkyl; A is A-1; X is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, Cl, F, Br, I, CH₂F, CF₃, OCH₂ CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; Y is H, C₁-C₂ alkyl, C₁ -C₂ alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃, N(OCH₃)CH₃,N(CH₃)₂, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ .tbd.CH, OCH₂ CH₂ OCH₃, C(O)R_(a),cyclopropyl, C.tbd.CH or C.tbd.CCH₃ ; R_(a) is H or CH₃ ; and Z is CH;then R₂ is other than CN, CO₂ R₉, CO₂ R'₉.
 2. A compound of claim 1whereX is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, Cl, F, Br, I, CH₂ F, CF₃, OCH₂CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; and Y is H, C₁ -C₂ alkyl,C₁ -C₂ alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃, N(OCH₃)CH₃, N(CH₃)₂, CF₃,SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, ##STR64## CH₂ SCH₃,cyclopropyl, C.tbd.CH or C.tbd.CCH₃ ; and R_(a) is H or CH₃.
 3. Acompound claim 2 whereW is O; R_(f) is H, CH₃, C₁ haloalkyl, halogen orOCH₃ ; R_(g) is C₁ -C₂ haloalkyl, ethyl, W₂ R₁₁, CH₂ OCH₃, CH₂ SCH₃, CH₂CN, C₁ -C₂ alkylamino or N(CH₃)₂ ; R₂ is C₁ -C₄ alkylsulfinyl, C₁ -C₄alkylsulfonyl, SO₂ NH₂, SO₂ NR_(d) R_(e), SO₂ NR₇ R₈, SO₂ NR'₇ R₈, OSO₂R₈, SO₂ OR₈, N₃, P(W₁)(OC₁ -C₂ alkyl)₂, CN, CO₂ R₉, CO₂ R'₉, CHF₂, CF₂H, CH₂ Cl, CCl₂ H or C₂ -C₄ haloalkyl; R₇ is H, C₂ -C₃ cyanoalkyl, C₃-C₄ alkenyl or C₃ -C₄ alkynyl; R₈ is C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, C₃-C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄ alkoxyalkyl or cyclopropyl; and R₁₁is C₁ -C₃ alkyl, C₁ -C₂ haloalkyl, allyl or propargyl.
 4. A compound ofclaim 3 whereR₇ is H, C₂ -C₃ cyanoalkyl, allyl or propargyl; R'₇ is C₁-C₃ alkyl; R₈ is C₁ -C₃ alkyl, allyl, propargyl or cyclopropyl; R₉ isCH₂ CH₂ R₁₀, CH₂ CH₂ SCH₃, propargyl or cyclopropylmethyl; R'₉ is C₁ -C₃alkyl, allyl, CH₂ CH₂ OCH₃ or CH₂ CH₂ Cl; and R₁₀ is OH, CN or OSO₂ CH₃.5. A compound of claim 4 whereX is CH₃, OCH₃, OCH₂ CH₃, Cl or OCH₂ CF₃ ;and Y is CH₃, OCH₃, CH₂ CH₃, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 6. Thecompound of claim 1 which isN2-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-N3-ethyl-2,3-pyridinedisulfonamide.7. The compound of claim 1 which isN-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-3-(methylsulfonyloxy)-2-pyridinesulfonamide.8. The compound of claim 1 which isN2-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-N3-methyl-2,3-pyridinedisulfonamide.9. A composition suitable for controlling the growth of undesiredvegetation which comprises an effective amount of a compound of claim 1and at least one of the following: surfactant, solid inert diluent orliquid inert diluent and mixtures of the foregoing.
 10. A method forcontrolling the growth of undesired vegetation which comprises applyingto the locus to be protected an effective amount of a compound of claim1.